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—— [(6S)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone —— C18H21FN4O3
[(6S)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]-[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methanone
—— (6S)-3-ethyl-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-6-phenyl-1,6-dihydropyrimidin-2-one —— C22H22N2O3
(6S)-3-ethyl-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-6-phenyl-1,6-dihydropyrimidin-2-one
—— (6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 3-methoxybenzoate —— C20H18O6
(6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 3-methoxybenzoate
—— 6-fluoro-2-[(2S)-1-[3-(5-methyltetrazol-1-yl)propyl]pyrrolidin-2-yl]-1H-benzimidazole —— C16H20FN7
6-fluoro-2-[(2S)-1-[3-(5-methyltetrazol-1-yl)propyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-3-ethyl-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-4-methyl-6-phenyl-1,6-dihydropyrimidin-2-one —— C23H24N2O3
(6S)-3-ethyl-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-4-methyl-6-phenyl-1,6-dihydropyrimidin-2-one
—— (6R)-5-acetyl-4-methyl-6-phenyl-3-prop-2-enyl-1,6-dihydropyrimidin-2-one —— C16H18N2O2
(6R)-5-acetyl-4-methyl-6-phenyl-3-prop-2-enyl-1,6-dihydropyrimidin-2-one
—— (6R)-3-ethyl-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-6-phenyl-1,6-dihydropyrimidin-2-one —— C22H22N2O3
(6R)-3-ethyl-5-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-6-phenyl-1,6-dihydropyrimidin-2-one
—— 6-(chloromethyl)-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C12H9ClN4O
6-(chloromethyl)-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— (6S)-5-acetyl-3-ethyl-6-(4-methoxyphenyl)-4-methyl-1,6-dihydropyrimidin-2-one —— C16H20N2O3
(6S)-5-acetyl-3-ethyl-6-(4-methoxyphenyl)-4-methyl-1,6-dihydropyrimidin-2-one
—— (6S)-5-acetyl-3-ethyl-6-phenyl-1,6-dihydropyrimidin-2-one —— C14H16N2O2
(6S)-5-acetyl-3-ethyl-6-phenyl-1,6-dihydropyrimidin-2-one
—— (6S)-5-acetyl-4-methyl-6-phenyl-3-prop-2-enyl-1,6-dihydropyrimidin-2-one —— C16H18N2O2
(6S)-5-acetyl-4-methyl-6-phenyl-3-prop-2-enyl-1,6-dihydropyrimidin-2-one
—— (6R)-5-acetyl-3-ethyl-6-phenyl-1,6-dihydropyrimidin-2-one —— C14H16N2O2
(6R)-5-acetyl-3-ethyl-6-phenyl-1,6-dihydropyrimidin-2-one
—— 6-oxo-N-[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]-1H-pyrimidine-5-carboxamide —— C16H16F3N5O2
6-oxo-N-[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]-1H-pyrimidine-5-carboxamide
—— 6-cyclopentyl-1-methyl-N-[[(3S)-1-propylpiperidin-3-yl]methyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H32N6
6-cyclopentyl-1-methyl-N-[[(3S)-1-propylpiperidin-3-yl]methyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6R)-4-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C16H26N4O2
(6R)-4-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— (6-aminopyridin-3-yl)-[(2R)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone —— C19H21N3O2
(6-aminopyridin-3-yl)-[(2R)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone
—— 6-phenyl-N-(2,2,6,6-tetramethylpiperidin-1-ium-4-yl)thieno[2,3-d]pyrimidin-4-amine —— C21H27N4S+
6-phenyl-N-(2,2,6,6-tetramethylpiperidin-1-ium-4-yl)thieno[2,3-d]pyrimidin-4-amine
—— 6-fluoro-N-[(3S)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-1H-benzimidazole-2-carboxamide —— C20H20F2N4O
6-fluoro-N-[(3S)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-1H-benzimidazole-2-carboxamide
—— 6-[[(3S)-5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]amino]pyridine-2-carbonitrile —— C19H20N4O
6-[[(3S)-5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]amino]pyridine-2-carbonitrile
—— 6-fluoro-N-[(3R)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-1H-benzimidazole-2-carboxamide —— C20H20F2N4O
6-fluoro-N-[(3R)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-1H-benzimidazole-2-carboxamide
—— 6-methyl-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide —— C20H22N6O2
6-methyl-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
—— 6-methyl-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide —— C20H22N6O2
6-methyl-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
—— 6-cyclopentyl-1-methyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C16H22N8
6-cyclopentyl-1-methyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6-aminopyridin-3-yl)-[(2S)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone —— C19H21N3O2
(6-aminopyridin-3-yl)-[(2S)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone
—— 6-(methoxymethyl)-1-methyl-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C15H21N7O
6-(methoxymethyl)-1-methyl-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-(methoxymethyl)-1-methyl-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C15H21N7O
6-(methoxymethyl)-1-methyl-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-cyclopentyl-1-methyl-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C16H22N8
6-cyclopentyl-1-methyl-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-oxo-N-[(3R)-5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-propan-2-yl-1H-pyrimidine-5-carboxamide —— C20H24N4O3
6-oxo-N-[(3R)-5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-propan-2-yl-1H-pyrimidine-5-carboxamide
—— 6-ethyl-N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C16H20N6O
6-ethyl-N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— 6-oxa-9-azaspiro[4.5]decan-9-yl-[2-[(3R)-pyrrolidin-3-yl]phenyl]methanone —— C19H26N2O2
6-oxa-9-azaspiro[4.5]decan-9-yl-[2-[(3R)-pyrrolidin-3-yl]phenyl]methanone
—— 6-oxo-N-[(3S)-5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-propan-2-yl-1H-pyrimidine-5-carboxamide —— C20H24N4O3
6-oxo-N-[(3S)-5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-propan-2-yl-1H-pyrimidine-5-carboxamide
—— 6-cyclopentyl-N,1-dimethyl-N-[(3R)-3-pyrrolidin-1-ylbutyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H32N6
6-cyclopentyl-N,1-dimethyl-N-[(3R)-3-pyrrolidin-1-ylbutyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-oxa-9-azaspiro[4.5]decan-9-yl-[2-[(3S)-pyrrolidin-3-yl]phenyl]methanone —— C19H26N2O2
6-oxa-9-azaspiro[4.5]decan-9-yl-[2-[(3S)-pyrrolidin-3-yl]phenyl]methanone
—— 6-amino-1-[(3S)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]hexan-1-one —— C18H27N3O3
6-amino-1-[(3S)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]hexan-1-one
—— 6-cyclopentyl-N,1-dimethyl-N-[(3S)-3-pyrrolidin-1-ylbutyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C20H32N6
6-cyclopentyl-N,1-dimethyl-N-[(3S)-3-pyrrolidin-1-ylbutyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6R)-4-[[1-(1,3-thiazol-2-yl)pyrrol-2-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C16H22N4O2S
(6R)-4-[[1-(1,3-thiazol-2-yl)pyrrol-2-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— 6-[3-hydroxy-5-[2-[(2S)-piperidin-2-yl]ethyl]phenyl]-2H-isoquinolin-1-one —— C22H24N2O2
6-[3-hydroxy-5-[2-[(2S)-piperidin-2-yl]ethyl]phenyl]-2H-isoquinolin-1-one
—— 6-amino-1-[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]hexan-1-one —— C18H27N3O3
6-amino-1-[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]hexan-1-one
—— 6-[3-hydroxy-5-[2-[(2R)-piperidin-2-yl]ethyl]phenyl]-2H-isoquinolin-1-one —— C22H24N2O2
6-[3-hydroxy-5-[2-[(2R)-piperidin-2-yl]ethyl]phenyl]-2H-isoquinolin-1-one
—— [(6R)-4-(1-ethylpiperidin-4-yl)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-8-yl]-(2-methylphenyl)methanone —— C23H35N3O3
[(6R)-4-(1-ethylpiperidin-4-yl)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-8-yl]-(2-methylphenyl)methanone
—— (6R)-4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C19H30N2O3
(6R)-4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— (6S)-4-[[1-(1,3-thiazol-2-yl)pyrrol-2-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C16H22N4O2S
(6S)-4-[[1-(1,3-thiazol-2-yl)pyrrol-2-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— 6-[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-N,N-diethylpyridine-3-sulfonamide —— C20H24N4O2S2
6-[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-N,N-diethylpyridine-3-sulfonamide
—— 6-tert-butyl-N-[(1S)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C17H24N6O
6-tert-butyl-N-[(1S)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— (6R)-6-methyl-N-[[(2R)-oxolan-2-yl]methyl]-6,7,8,9-tetrahydro-5H-carbazole-3-carboxamide —— C19H24N2O2
(6R)-6-methyl-N-[[(2R)-oxolan-2-yl]methyl]-6,7,8,9-tetrahydro-5H-carbazole-3-carboxamide
—— (6S,9R)-9-(4-chlorophenyl)-6-propyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C19H18ClF3N4O
(6S,9R)-9-(4-chlorophenyl)-6-propyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— [(6S)-4-(1-ethylpiperidin-4-yl)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-8-yl]-(2-methylphenyl)methanone —— C23H35N3O3
[(6S)-4-(1-ethylpiperidin-4-yl)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-8-yl]-(2-methylphenyl)methanone
—— (6S)-4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C19H30N2O3
(6S)-4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— 6-tert-butyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C17H24N6O
6-tert-butyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— (6R,9S)-9-(4-chlorophenyl)-6-propyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C19H18ClF3N4O
(6R,9S)-9-(4-chlorophenyl)-6-propyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one