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—— (6S)-6-(4-chlorophenyl)-3-cyclopropyl-N,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxamide —— C16H18ClN3OS
(6S)-6-(4-chlorophenyl)-3-cyclopropyl-N,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxamide
—— 6-[[(3S,8aR)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one —— C17H23N3O3S
6-[[(3S,8aR)-3-methyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(3R)-3-(4-ethyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C16H20N4O2S
6-[(3R)-3-(4-ethyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— [6-(dimethylamino)pyridazin-3-yl]-[(3S)-3-(4-ethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C17H23N5OS
[6-(dimethylamino)pyridazin-3-yl]-[(3S)-3-(4-ethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— [6-(dimethylamino)pyridazin-3-yl]-[(3R)-3-(4-ethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C17H23N5OS
[6-(dimethylamino)pyridazin-3-yl]-[(3R)-3-(4-ethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— 6-[(3S)-3-(4-ethyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C16H20N4O2S
6-[(3S)-3-(4-ethyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— 6-ethyl-N-[(2S)-2-morpholin-4-yl-2-thiophen-2-ylethyl]pyrimidin-4-amine —— C16H22N4OS
6-ethyl-N-[(2S)-2-morpholin-4-yl-2-thiophen-2-ylethyl]pyrimidin-4-amine
—— 6-[(3R)-3-(4-ethyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]-2-methylpyridine-3-carbonitrile —— C18H20N4OS
6-[(3R)-3-(4-ethyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]-2-methylpyridine-3-carbonitrile
—— 6-[2-[(S)-benzylsulfinyl]ethylamino]-5-chloropyridine-3-carboxamide —— C15H16ClN3O2S
6-[2-[(S)-benzylsulfinyl]ethylamino]-5-chloropyridine-3-carboxamide
—— 6-ethyl-N-methyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-2-ylethyl]pyrimidin-4-amine —— C17H24N4OS
6-ethyl-N-methyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-2-ylethyl]pyrimidin-4-amine
—— 6-[2-[(R)-benzylsulfinyl]ethylamino]-5-chloropyridine-3-carboxamide —— C15H16ClN3O2S
6-[2-[(R)-benzylsulfinyl]ethylamino]-5-chloropyridine-3-carboxamide
—— 6-ethyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-2-ylethyl]pyrimidin-4-amine —— C16H22N4OS
6-ethyl-N-[(2R)-2-morpholin-4-yl-2-thiophen-2-ylethyl]pyrimidin-4-amine
—— 6-[(3S)-3-carbamoylpiperidin-1-yl]-N-(4-methylphenyl)pyridine-3-carboxamide —— C19H22N4O2
6-[(3S)-3-carbamoylpiperidin-1-yl]-N-(4-methylphenyl)pyridine-3-carboxamide
—— 6-[(3R)-3-carbamoylpiperidin-1-yl]-N-(4-methylphenyl)pyridine-3-carboxamide —— C19H22N4O2
6-[(3R)-3-carbamoylpiperidin-1-yl]-N-(4-methylphenyl)pyridine-3-carboxamide
—— 6-bromo-N-ethoxy-4-oxo-1H-quinoline-2-carboxamide —— C12H11BrN2O3
6-bromo-N-ethoxy-4-oxo-1H-quinoline-2-carboxamide
—— 6-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]pyridine-3-carboxamide —— C18H23N5O2
6-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]pyridine-3-carboxamide
—— 6-[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]pyridine-3-carboxamide —— C18H23N5O2
6-[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]pyridine-3-carboxamide
—— 6-[[(3S)-3-ethyl-4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C16H28N4O3
6-[[(3S)-3-ethyl-4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[[(3R)-3-ethyl-4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C16H28N4O3
6-[[(3R)-3-ethyl-4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C16H19N5O
6-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[(2R)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C14H15N5O
6-[(2R)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— 6-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C16H19N5O
6-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[(2S)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C14H15N5O
6-[(2S)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— 6-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C14H15N5O
6-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile —— C14H15N5O
6-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
—— 6-(cyclopropylamino)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide —— C16H19N5O
6-(cyclopropylamino)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide
—— 6-(azepan-1-yl)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide —— C19H25N5O
6-(azepan-1-yl)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide
—— 6-(azepan-1-yl)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide —— C19H25N5O
6-(azepan-1-yl)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide
—— 6-(cyclopropylamino)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide —— C16H19N5O
6-(cyclopropylamino)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide
—— 6-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-3-methyl-1,3-benzoxazol-2-one —— C15H19N3O4S
6-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-3-methyl-1,3-benzoxazol-2-one
—— 6-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one —— C16H21N3O3S
6-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidine-1-carbonyl]-2-ethylpyridazin-3-one —— C16H22N6O2
6-[(3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidine-1-carbonyl]-2-ethylpyridazin-3-one
—— 6-[(3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidine-1-carbonyl]-2-ethylpyridazin-3-one —— C16H22N6O2
6-[(3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidine-1-carbonyl]-2-ethylpyridazin-3-one
—— 6-[[(2R)-4-methylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile —— C12H16N4O
6-[[(2R)-4-methylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile
—— 6-[(2R)-2-[(1R)-1-phenylpropyl]pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine —— C17H20N6
6-[(2R)-2-[(1R)-1-phenylpropyl]pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine
—— 6-[[(2S)-4-methylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile —— C12H16N4O
6-[[(2S)-4-methylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile
—— 6-[(2R)-2-[(1S)-1-phenylpropyl]pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine —— C17H20N6
6-[(2R)-2-[(1S)-1-phenylpropyl]pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine
—— 6-[(2S)-2-[[(3,5-dimethyl-1,2-oxazol-4-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine —— C16H24N6O
6-[(2S)-2-[[(3,5-dimethyl-1,2-oxazol-4-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine
—— 6-[(2R)-2-[[(3,5-dimethyl-1,2-oxazol-4-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine —— C16H24N6O
6-[(2R)-2-[[(3,5-dimethyl-1,2-oxazol-4-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine
—— 6-methyl-2-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole —— C14H18N6S
6-methyl-2-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole
—— 6-[(2S)-2-[[(1-ethylimidazol-2-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine —— C16H25N7
6-[(2S)-2-[[(1-ethylimidazol-2-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine
—— 6-[(2R)-2-[[(1-ethylimidazol-2-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine —— C16H25N7
6-[(2R)-2-[[(1-ethylimidazol-2-yl)methylamino]methyl]pyrrolidin-1-yl]-N-methylpyrimidin-4-amine
—— 6-[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C16H19N5O
6-[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— 6-[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C16H19N5O
6-[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— 6-[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine —— C13H15ClN8
6-[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine
—— 6-[(2S)-2-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]morpholin-4-yl]pyridine-3-carbonitrile —— C15H18N6O
6-[(2S)-2-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]morpholin-4-yl]pyridine-3-carbonitrile
—— 6-methyl-N-[(6S)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C14H19N7S
6-methyl-N-[(6S)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— 6-[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine —— C13H15ClN8
6-[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]tetrazolo[1,5-b]pyridazine
—— 6-[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C15H16ClN5
6-[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— 6-[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]pyridine-3-carbonitrile —— C14H16N6
6-[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]pyridine-3-carbonitrile