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—— 6-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C21H24N6O
6-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[[5-(2-methylpropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-2-N-phenyl-1,3,5-triazine-2,4-diamine —— C16H20N8S2
6-[[5-(2-methylpropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-2-N-phenyl-1,3,5-triazine-2,4-diamine
—— 6-[(3S)-1-[(2,4-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C21H20F2N4O
6-[(3S)-1-[(2,4-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H27N5O2
6-[(3R)-1-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H24N4O3
6-[(3S)-1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-ethylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H24N6OS
6-[(3R)-1-[(2-ethylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H28N4O3
6-[(3R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(3-methoxy-4-propan-2-yloxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H30N4O3
6-[(3R)-1-[(3-methoxy-4-propan-2-yloxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H30N8O
6-[(3S)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C21H22N6OS
6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(4-methylsulfanylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H24N4OS
6-[(3S)-1-[(4-methylsulfanylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H28N4O3
6-[(3S)-1-[(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C23H26N4O3
6-[(3S)-1-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H26N6O
6-[(3R)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(4-methoxy-3-propan-2-yloxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H30N4O3
6-[(3S)-1-[(4-methoxy-3-propan-2-yloxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(4-methylsulfanylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H24N4OS
6-[(3R)-1-[(4-methylsulfanylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H26N6O
6-[(3S)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C21H24N6O
6-[(3S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C20H22N6O2
6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(3-methoxy-4-prop-2-ynoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H26N4O3
6-[(3S)-1-[(3-methoxy-4-prop-2-ynoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H28N4O3
6-[(3S)-1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C20H23N7O
6-[(3S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H24N4O3
6-[(3R)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(3,4-dimethoxy-5-prop-2-enylphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C26H30N4O3
6-[(3R)-1-[(3,4-dimethoxy-5-prop-2-enylphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H30N8O
6-[(3R)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H24N4O3
6-[(3R)-1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H28N4O3
6-[(3R)-1-[(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(4-methoxy-3-propan-2-yloxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H30N4O3
6-[(3R)-1-[(4-methoxy-3-propan-2-yloxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(3-methoxy-4-prop-2-ynoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H26N4O3
6-[(3R)-1-[(3-methoxy-4-prop-2-ynoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H28N4O3
6-[(3R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H28N4O3
6-[(3S)-1-[(4,5-dimethoxy-2-methylphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C20H22N6OS
6-[(3S)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C23H24N4O4
6-[(3R)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-methyl-5-(4-methylphenyl)-2-[(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C21H23N3O2S2
6-methyl-5-(4-methylphenyl)-2-[(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-[(3R)-1-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C23H26N4O3
6-[(3R)-1-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-propylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-4-one —— C22H26N6OS
6-[(3R)-1-[(2-propylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C20H22N6O2
6-[(3R)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H24N4O2
6-[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C23H24N4O4
6-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C25H27N5O2
6-[(3S)-1-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(3,5-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H20F2N4O
6-[(3R)-1-[(3,5-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C22H26N6O
6-[(3S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(3,5-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H20F2N4O
6-[(3S)-1-[(3,5-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H20F2N4O
6-[(3R)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H24N4O3
6-[(3S)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C22H23FN4O2
6-[(3S)-1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C22H24N4O3
6-[(3R)-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C20H22N6O2
6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H22N6OS
6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H20F2N4O
6-[(3S)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one