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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-2-ethyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N4O
(6S)-2-ethyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H31FN4O
(6S)-2-[2-(dimethylamino)ethyl]-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[3-(2-methylimidazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O
(6S)-2-ethyl-8-[3-(2-methylimidazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone —— C18H24ClN5O2
(6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone
—— (6S)-2-[[2-(2,5-difluorophenyl)sulfanylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C18H18F2N2O2S2
(6S)-2-[[2-(2,5-difluorophenyl)sulfanylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-Amino-3-methyl-1-propyl-5-(2-pyridin-2-ylsulfanylacetyl)pyrimidine-2,4-dione —— C15H18N4O3S
6-Amino-3-methyl-1-propyl-5-(2-pyridin-2-ylsulfanylacetyl)pyrimidine-2,4-dione
—— 6-[2-(2,5-difluorophenyl)sulfanylacetyl]-4H-1,4-benzoxazin-3-one —— C16H11F2NO3S
6-[2-(2,5-difluorophenyl)sulfanylacetyl]-4H-1,4-benzoxazin-3-one
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 2-hydroxy-5-methylbenzoate —— C17H15NO7
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 2-hydroxy-5-methylbenzoate
—— 6-(2-chlorophenyl)-N-[(2R)-2-hydroxybutyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C18H19ClN4O3
6-(2-chlorophenyl)-N-[(2R)-2-hydroxybutyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-6-[4-(3,4-dihydro-1H-isoquinolin-2-yl)piperidine-1-carbonyl]piperazin-2-one —— C19H26N4O2
(6S)-6-[4-(3,4-dihydro-1H-isoquinolin-2-yl)piperidine-1-carbonyl]piperazin-2-one
—— (6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone —— C18H24ClN5O2
(6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone
—— (6R)-8-pentanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O2
(6R)-8-pentanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-N-[(2S)-2-hydroxybutyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C18H19ClN4O3
6-(2-chlorophenyl)-N-[(2S)-2-hydroxybutyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-2-(3-methoxypropyl)-8-(7H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N6O2
(6R)-2-(3-methoxypropyl)-8-(7H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(dimethylamino)ethyl]-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H31FN4O
(6R)-2-[2-(dimethylamino)ethyl]-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(3-chlorophenyl)-N-[(2S)-2,3-dihydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C19H19ClN4O4
6-(3-chlorophenyl)-N-[(2S)-2,3-dihydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(3-chlorophenyl)-N-[(2R)-2,3-dihydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C19H19ClN4O4
6-(3-chlorophenyl)-N-[(2R)-2,3-dihydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[(3R)-2-oxopyrrolidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide —— C18H19N5O4
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[(3R)-2-oxopyrrolidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-8-(2-ethoxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O3
(6R)-8-(2-ethoxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[(3S)-2-oxopyrrolidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide —— C18H19N5O4
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[(3S)-2-oxopyrrolidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-8-(3-amino-1H-pyrazole-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C17H28N6O2
(6S)-8-(3-amino-1H-pyrazole-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-phenyl-3-[(2S)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyridin-2-one —— C22H21N3O2
6-phenyl-3-[(2S)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyridin-2-one
—— (6R)-8-[4-(hydroxymethyl)pyridin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O2
(6R)-8-[4-(hydroxymethyl)pyridin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6R)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-amino-1H-pyrazole-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C17H28N6O2
(6R)-8-(3-amino-1H-pyrazole-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [6-[(2S)-1-(dimethylamino)hex-5-en-2-yl]oxypyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C17H26N4O2
[6-[(2S)-1-(dimethylamino)hex-5-en-2-yl]oxypyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— (6S)-8-[(E)-pent-3-enoyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O2
(6S)-8-[(E)-pent-3-enoyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(pyridin-2-ylmethyl)-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N4O2
(6R)-2-(pyridin-2-ylmethyl)-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(E)-pent-3-enoyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O2
(6R)-8-[(E)-pent-3-enoyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [6-[(2R)-1-(dimethylamino)hex-5-en-2-yl]oxypyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C17H26N4O2
[6-[(2R)-1-(dimethylamino)hex-5-en-2-yl]oxypyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— 6-phenyl-3-[(2R)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyridin-2-one —— C22H21N3O2
6-phenyl-3-[(2R)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyridin-2-one
—— (6S)-2-(pyridin-2-ylmethyl)-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N4O2
(6S)-2-(pyridin-2-ylmethyl)-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[4-(hydroxymethyl)pyridin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O2
(6S)-8-[4-(hydroxymethyl)pyridin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-(diethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-8-[2-(diethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[2-(diethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6R)-8-[2-(diethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-ethoxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O3
(6S)-8-(2-ethoxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N5O
(6R)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N5O
(6S)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6S)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine-2,4-diamine —— C18H29N9
6-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine-2,4-diamine
—— (6S)-8-(2-amino-6-methoxypyrimidin-4-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N6O2
(6S)-8-(2-amino-6-methoxypyrimidin-4-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine-2,4-diamine —— C18H29N9
6-[(3S)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine-2,4-diamine
—— (6R)-8-(2-butoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O3
(6R)-8-(2-butoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-fluorophenyl)-2-[(5R)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]pyridine-3-carboxylic acid —— C20H20FN3O4
6-(4-fluorophenyl)-2-[(5R)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]pyridine-3-carboxylic acid
—— (6S)-8-(2-butoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O3
(6S)-8-(2-butoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(3-ethylsulfanylpropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O2S
(6S)-8-(3-ethylsulfanylpropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-fluorophenyl)-2-[(5S)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]pyridine-3-carboxylic acid —— C20H20FN3O4
6-(4-fluorophenyl)-2-[(5S)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.5]decan-9-yl]pyridine-3-carboxylic acid
—— (6R)-8-[3-(dimethylamino)propanoyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6R)-8-[3-(dimethylamino)propanoyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one