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—— (6-aminopyridin-3-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone —— C20H22F3N3O
(6-aminopyridin-3-yl)-[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methanone
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate —— C17H17ClN2O6S
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-[2-[(5-methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]sulfanylacetate
—— 6-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione —— C21H28N4O3
6-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione
—— 6-[(3S)-oxolan-3-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C10H14N4OS
6-[(3S)-oxolan-3-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6-[(3R)-oxolan-3-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C10H14N4OS
6-[(3R)-oxolan-3-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— [6-[(2S)-2-(4-chlorophenyl)morpholin-4-yl]pyrazin-2-yl]-piperidin-1-ylmethanone —— C20H23ClN4O2
[6-[(2S)-2-(4-chlorophenyl)morpholin-4-yl]pyrazin-2-yl]-piperidin-1-ylmethanone
—— 6-[4-[(1R)-1-methoxyethyl]phenyl]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C21H24N4O3
6-[4-[(1R)-1-methoxyethyl]phenyl]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— [6-[(2R)-2-(4-chlorophenyl)morpholin-4-yl]pyrazin-2-yl]-piperidin-1-ylmethanone —— C20H23ClN4O2
[6-[(2R)-2-(4-chlorophenyl)morpholin-4-yl]pyrazin-2-yl]-piperidin-1-ylmethanone
—— 6-phenyl-3-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one —— C17H15F3N2O3
6-phenyl-3-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one
—— 6-[2-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one —— C15H14N4O3S2
6-[2-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one
—— [6-[(2R)-2-(4-chlorophenyl)morpholin-4-yl]pyridin-3-yl]-morpholin-4-ylmethanone —— C20H22ClN3O3
[6-[(2R)-2-(4-chlorophenyl)morpholin-4-yl]pyridin-3-yl]-morpholin-4-ylmethanone
—— 6-[4-[(1S)-1-methoxyethyl]phenyl]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C21H24N4O3
6-[4-[(1S)-1-methoxyethyl]phenyl]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— (6-methoxynaphthalen-2-yl)-[(3R)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]methanone —— C23H22N4O2
(6-methoxynaphthalen-2-yl)-[(3R)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]methanone
—— (6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-hydroxybenzoate —— C19H16O6
(6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-hydroxybenzoate
—— 6-phenyl-3-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one —— C17H15F3N2O3
6-phenyl-3-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one
—— [6-[(2S)-2-(4-chlorophenyl)morpholin-4-yl]pyridin-3-yl]-morpholin-4-ylmethanone —— C20H22ClN3O3
[6-[(2S)-2-(4-chlorophenyl)morpholin-4-yl]pyridin-3-yl]-morpholin-4-ylmethanone
—— [6-[[(3S)-oxolan-3-yl]methylamino]pyridin-3-yl]-(4-pyridin-3-yloxypiperidin-1-yl)methanone —— C21H26N4O3
[6-[[(3S)-oxolan-3-yl]methylamino]pyridin-3-yl]-(4-pyridin-3-yloxypiperidin-1-yl)methanone
—— 6-methyl-5-[1-[[(3S)-1-methylpyrrolidin-3-yl]methyl]imidazol-2-yl]quinoline —— C19H22N4
6-methyl-5-[1-[[(3S)-1-methylpyrrolidin-3-yl]methyl]imidazol-2-yl]quinoline
—— (6-methoxynaphthalen-2-yl)-[(3S)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]methanone —— C23H22N4O2
(6-methoxynaphthalen-2-yl)-[(3S)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]methanone
—— 6-Ethyl-7-hydroxy-4-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C17H17N3O3S2
6-Ethyl-7-hydroxy-4-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— 6-[(2R)-2-[2-(dimethylamino)ethyl]morpholin-4-yl]-N-ethylpyridine-3-carboxamide —— C16H26N4O2
6-[(2R)-2-[2-(dimethylamino)ethyl]morpholin-4-yl]-N-ethylpyridine-3-carboxamide
—— (6R)-6-(4,4-diphenylpiperidine-1-carbonyl)piperazin-2-one —— C22H25N3O2
(6R)-6-(4,4-diphenylpiperidine-1-carbonyl)piperazin-2-one
—— 6-[(3S)-3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile —— C19H18FN3O2
6-[(3S)-3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile
—— 6,7-Dimethyl-4-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C17H17N3O2S2
6,7-Dimethyl-4-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— (6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-hydroxybenzoate —— C18H13ClO5
(6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-hydroxybenzoate
—— [6-[[(3R)-oxolan-3-yl]methylamino]pyridin-3-yl]-(4-pyridin-3-yloxypiperidin-1-yl)methanone —— C21H26N4O3
[6-[[(3R)-oxolan-3-yl]methylamino]pyridin-3-yl]-(4-pyridin-3-yloxypiperidin-1-yl)methanone
—— 6-[(3R)-3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyrazine-2-carboxamide —— C18H19FN4O3
6-[(3R)-3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyrazine-2-carboxamide
—— (6S)-6-(4,4-diphenylpiperidine-1-carbonyl)piperazin-2-one —— C22H25N3O2
(6S)-6-(4,4-diphenylpiperidine-1-carbonyl)piperazin-2-one
—— 6-propan-2-yl-3-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one —— C14H17F3N2O3
6-propan-2-yl-3-[(2S)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one
—— 6-[(2S)-2-[2-(dimethylamino)ethyl]morpholin-4-yl]-N-ethylpyridine-3-carboxamide —— C16H26N4O2
6-[(2S)-2-[2-(dimethylamino)ethyl]morpholin-4-yl]-N-ethylpyridine-3-carboxamide
—— 6-propan-2-yl-3-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one —— C14H17F3N2O3
6-propan-2-yl-3-[(2R)-2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyridin-2-one
—— 6-[(3R)-3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile —— C19H18FN3O2
6-[(3R)-3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile
—— 6-methyl-2-[2-[2-[(3S)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one —— C14H19N5O2
6-methyl-2-[2-[2-[(3S)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one
—— (6R)-2,6-diamino-4-(phenylmethoxymethyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C18H20N4O
(6R)-2,6-diamino-4-(phenylmethoxymethyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— 6-methyl-2-[2-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one —— C14H19N5O2
6-methyl-2-[2-[2-[(3R)-oxolan-3-yl]imidazol-1-yl]ethylamino]-1H-pyrimidin-4-one
—— 6-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-3-[(2R)-oxolan-2-yl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C13H12N6OS2
6-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-3-[(2R)-oxolan-2-yl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— 6-Chloro-7-methyl-4-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C16H14ClN3O2S2
6-Chloro-7-methyl-4-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— (6S)-2,6-diamino-4-(phenylmethoxymethyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C18H20N4O
(6S)-2,6-diamino-4-(phenylmethoxymethyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— 6-(Furan-2-yl)-3-methyl-1-[2-(trifluoromethyl)phenyl]pyrazolo[3,4-b]pyridine-4-carboxylate —— C19H11F3N3O3-
6-(Furan-2-yl)-3-methyl-1-[2-(trifluoromethyl)phenyl]pyrazolo[3,4-b]pyridine-4-carboxylate
—— 6-[(2R)-2-(4-fluorophenyl)morpholin-4-yl]pyridine-3-carboxylic acid —— C16H15FN2O3
6-[(2R)-2-(4-fluorophenyl)morpholin-4-yl]pyridine-3-carboxylic acid
—— 6-[(2S)-2-(4-fluorophenyl)morpholin-4-yl]pyridine-3-carboxylic acid —— C16H15FN2O3
6-[(2S)-2-(4-fluorophenyl)morpholin-4-yl]pyridine-3-carboxylic acid
—— 6-[5-[4-(dimethylamino)-2-methyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C20H22N6O2
6-[5-[4-(dimethylamino)-2-methyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— (6R)-2-amino-4-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)-6-methyl-5,6,7,8-tetrahydro-1H-quinoline-3-carbonitrile —— C17H17N3O2
(6R)-2-amino-4-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)-6-methyl-5,6,7,8-tetrahydro-1H-quinoline-3-carbonitrile
—— (6S)-2-amino-4-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)-6-methyl-5,6,7,8-tetrahydro-1H-quinoline-3-carbonitrile —— C17H17N3O2
(6S)-2-amino-4-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)-6-methyl-5,6,7,8-tetrahydro-1H-quinoline-3-carbonitrile
—— 6-methyl-2-[(3R)-3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl]pyridine-3-carbonitrile —— C20H18F3N3O
6-methyl-2-[(3R)-3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-(6-methoxypyridin-3-yl)-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C21H28N4O2
6-(6-methoxypyridin-3-yl)-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— 6-(6-methoxypyridin-3-yl)-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C21H28N4O2
6-(6-methoxypyridin-3-yl)-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— (6R)-2,6-diamino-4-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C21H22N6O
(6R)-2,6-diamino-4-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— (6S)-6-[(3aS,4S,7R,7aR)-1,3,3a,4,5,6,7,7a-octahydro-4,7-epoxyisoindole-2-carbonyl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C16H22N4O3
(6S)-6-[(3aS,4S,7R,7aR)-1,3,3a,4,5,6,7,7a-octahydro-4,7-epoxyisoindole-2-carbonyl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— (6S)-2,6-diamino-4-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C21H22N6O
(6S)-2,6-diamino-4-[4-methoxy-3-(pyrazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile