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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-8-(6-oxo-1H-pyrimidine-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23N5O3
(6S)-8-(6-oxo-1H-pyrimidine-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N4O
(6S)-2-benzyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-2-[(3S)-3-(methoxymethyl)pyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O3
6-(2-chlorophenyl)-2-[(3S)-3-(methoxymethyl)pyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6R)-8-(5-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-8-(5-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-7-methyl-8-oxo-N-[(2S)-pentan-2-yl]imidazo[1,2-a]pyrazine-2-carboxamide —— C19H21ClN4O2
6-(2-chlorophenyl)-7-methyl-8-oxo-N-[(2S)-pentan-2-yl]imidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2-chlorophenyl)-2-[(3R)-3-(methoxymethyl)pyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O3
6-(2-chlorophenyl)-2-[(3R)-3-(methoxymethyl)pyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— [6-[[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C21H33N5O
[6-[[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— (6S)-8-(5-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6S)-8-(5-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-cyclopentyl-1-methyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C18H25N7
6-cyclopentyl-1-methyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— [6-[[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C21H33N5O
[6-[[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— 6-cyclopentyl-1-methyl-N-[(2S)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C18H25N7
6-cyclopentyl-1-methyl-N-[(2S)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2S)-4-hydroxybutan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C19H24N4O4
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-4-hydroxybutan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N5O
(6R)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N5O
(6S)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O
(6S)-2-[2-(dimethylamino)ethyl]-8-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-acetylpyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6R)-8-(5-acetylpyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-acetylpyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6S)-8-(5-acetylpyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-fluorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C20H17FN4O3
6-(4-fluorophenyl)-N-[(1R)-1-(furan-2-yl)ethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2R)-4-hydroxybutan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C19H24N4O4
6-(2,5-dimethylfuran-3-yl)-N-[(2R)-4-hydroxybutan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(4-fluorophenyl)-N-[(1S)-1-(furan-2-yl)ethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C20H17FN4O3
6-(4-fluorophenyl)-N-[(1S)-1-(furan-2-yl)ethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-[(3S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl]-1H-pyrimidin-4-one —— C21H27N3O3
6-[(3S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl]-1H-pyrimidin-4-one
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(2-fluorobenzoyl)amino]acetate —— C19H17ClFNO5
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(2-fluorobenzoyl)amino]acetate
—— 6-(2-chlorophenyl)-N-[(1R)-1-cyclopropylethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C19H19ClN4O2
6-(2-chlorophenyl)-N-[(1R)-1-cyclopropylethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-[(3R)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl]-1H-pyrimidin-4-one —— C21H27N3O3
6-[(3R)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl]-1H-pyrimidin-4-one
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2R)-1-hydroxypropan-2-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C19H22N4O4
6-(2,5-dimethylfuran-3-yl)-N-[(2R)-1-hydroxypropan-2-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2-chlorophenyl)-N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C21H23ClN4O3
6-(2-chlorophenyl)-N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2-chlorophenyl)-N-[(1S)-1-cyclopropylethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C19H19ClN4O2
6-(2-chlorophenyl)-N-[(1S)-1-cyclopropylethyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-2-benzyl-8-[2-(1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O
(6S)-2-benzyl-8-[2-(1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-(2-propyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N3O2S
(6R)-2-ethyl-8-(2-propyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(2-propyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N3O2S
(6S)-2-ethyl-8-(2-propyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-(cyclohexanecarbonylamino)acetate —— C19H24ClNO5
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-(cyclohexanecarbonylamino)acetate
—— (6R)-8-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O3
(6R)-8-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-methyl-2-(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)-2,8-diazaspiro[5.5]undecane —— C20H31N5
(6R)-8-methyl-2-(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)-2,8-diazaspiro[5.5]undecane
—— 6-[[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine —— C12H10ClN7OS
6-[[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine
—— (6S)-8-methyl-2-(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)-2,8-diazaspiro[5.5]undecane —— C20H31N5
(6S)-8-methyl-2-(2-methyl-5-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl)-2,8-diazaspiro[5.5]undecane
—— (6S)-8-(5,6-dimethylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N5O
(6S)-8-(5,6-dimethylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3S)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino]-N,N-dimethylpyrazine-2-carboxamide —— C21H27N5O
6-[[(3S)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino]-N,N-dimethylpyrazine-2-carboxamide
—— (6S)-8-(6-methylpyridazin-3-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O
(6S)-8-(6-methylpyridazin-3-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino]-N,N-dimethylpyrazine-2-carboxamide —— C21H27N5O
6-[[(3R)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino]-N,N-dimethylpyrazine-2-carboxamide
—— 6-[(2R)-1-morpholin-4-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile —— C16H21N3O2
6-[(2R)-1-morpholin-4-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile
—— (6R)-8-(5-acetylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6R)-8-(5-acetylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2,2-dimethylbutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6R)-8-(2,2-dimethylbutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2,2-dimethylbutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6S)-8-(2,2-dimethylbutanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[(4-oxo-1H-quinolin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N3O2
(6R)-2-ethyl-8-[(4-oxo-1H-quinolin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-acetylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6S)-8-(5-acetylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[4-Cyclohexyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine —— C19H24N8OS
6-[[4-Cyclohexyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3,5-triazine-2,4-diamine
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H35N5O
(6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[(4-oxo-1H-quinolin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N3O2
(6S)-2-ethyl-8-[(4-oxo-1H-quinolin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-methylpyridazin-3-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O
(6R)-8-(6-methylpyridazin-3-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(4-methylpentanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6S)-8-(4-methylpentanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one