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—— 6-(2-chlorophenyl)-7-methyl-2-[(2R)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one —— C19H19ClN4O2
6-(2-chlorophenyl)-7-methyl-2-[(2R)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one
—— [(6R)-8-ethyl-2,8-diazaspiro[5.5]undecan-2-yl]-[3-(3-hydroxy-3-methylbutyl)phenyl]methanone —— C23H36N2O2
[(6R)-8-ethyl-2,8-diazaspiro[5.5]undecan-2-yl]-[3-(3-hydroxy-3-methylbutyl)phenyl]methanone
—— 6-(2-chlorophenyl)-7-methyl-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one —— C19H19ClN4O2
6-(2-chlorophenyl)-7-methyl-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one
—— 6-[(6R)-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C21H23N5O
6-[(6R)-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— 6-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carboxylic acid —— C20H25N5O2
6-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carboxylic acid
—— (6R)-2-benzyl-8-(3-imidazol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N4O
(6R)-2-benzyl-8-(3-imidazol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-8-ethyl-2,8-diazaspiro[5.5]undecan-2-yl]-[3-(3-hydroxy-3-methylbutyl)phenyl]methanone —— C23H36N2O2
[(6S)-8-ethyl-2,8-diazaspiro[5.5]undecan-2-yl]-[3-(3-hydroxy-3-methylbutyl)phenyl]methanone
—— 6-[(6S)-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C21H23N5O
6-[(6S)-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— 6-(2,5-dimethylfuran-3-yl)-N-[(3R)-1-methyl-2-oxopyrrolidin-3-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C21H23N5O4
6-(2,5-dimethylfuran-3-yl)-N-[(3R)-1-methyl-2-oxopyrrolidin-3-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-[(2-Methoxyanilino)methyl]-1,3,5-triazine-2,4-diamine —— C11H14N6O
6-[(2-Methoxyanilino)methyl]-1,3,5-triazine-2,4-diamine
—— 6-[(3R)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1H-pyrrolo[2,3-b]pyridine —— C20H23N3O2
6-[(3R)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1H-pyrrolo[2,3-b]pyridine
—— 6-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carboxylic acid —— C20H25N5O2
6-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-3-carboxylic acid
—— (6S)-8-[(4-methoxy-2-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C24H31N3O2
(6S)-8-[(4-methoxy-2-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-N-[(2R)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C19H19ClN4O3
6-(2-chlorophenyl)-N-[(2R)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— [(6R)-4-[(4-phenylphenyl)methyl]-1,4-oxazepan-6-yl]methanol —— C19H23NO2
[(6R)-4-[(4-phenylphenyl)methyl]-1,4-oxazepan-6-yl]methanol
—— 6-[(1S)-1-[2-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl)imidazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole —— C16H18N8S
6-[(1S)-1-[2-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl)imidazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole
—— (6S)-N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C15H21N5O2S
(6S)-N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-4-[(6-chloro-1,3-benzodioxol-5-yl)methyl]-1,4-oxazepan-6-ol —— C13H16ClNO4
(6R)-4-[(6-chloro-1,3-benzodioxol-5-yl)methyl]-1,4-oxazepan-6-ol
—— (6R)-2-ethyl-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O3
(6R)-2-ethyl-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O3
(6R)-8-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O2
(6S)-2-benzyl-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]amino]-N,N-dimethylpyridine-3-carboxamide —— C20H32N4O
6-[[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]amino]-N,N-dimethylpyridine-3-carboxamide
—— (6R)-8-[(4-methoxy-2-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C24H31N3O2
(6R)-8-[(4-methoxy-2-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2,5-dimethylfuran-3-yl)-N-[(3S)-1-methyl-2-oxopyrrolidin-3-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C21H23N5O4
6-(2,5-dimethylfuran-3-yl)-N-[(3S)-1-methyl-2-oxopyrrolidin-3-yl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-8-(3-methylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O
(6R)-8-(3-methylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O
(6S)-2-ethyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-cyclopentyl-N-[(1R)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H29N7
6-cyclopentyl-N-[(1R)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— 6-[[(6R)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1H-pyrimidine-2,4-dione —— C18H29N5O3
6-[[(6R)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1H-pyrimidine-2,4-dione
—— [(6S)-4-[(4-phenylphenyl)methyl]-1,4-oxazepan-6-yl]methanol —— C19H23NO2
[(6S)-4-[(4-phenylphenyl)methyl]-1,4-oxazepan-6-yl]methanol
—— (6S)-2-benzyl-8-(3-imidazol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N4O
(6S)-2-benzyl-8-(3-imidazol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6R)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O
(6R)-2-ethyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(1R)-1-[2-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl)imidazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole —— C16H18N8S
6-[(1R)-1-[2-(5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl)imidazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole
—— 6-[[(6S)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1H-pyrimidine-2,4-dione —— C18H29N5O3
6-[[(6S)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]methyl]-1H-pyrimidine-2,4-dione
—— (6R)-8-(5-fluoropyrimidin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H22FN5O
(6R)-8-(5-fluoropyrimidin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]amino]-N,N-dimethylpyridine-3-carboxamide —— C20H32N4O
6-[[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]amino]-N,N-dimethylpyridine-3-carboxamide
—— 6-(2-chlorophenyl)-N-[(2S)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C19H19ClN4O3
6-(2-chlorophenyl)-N-[(2S)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-8-(3-methylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O
(6S)-8-(3-methylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-fluoropyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23FN4O
(6R)-8-(3-fluoropyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-cyclopentyl-N-[(1S)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H29N7
6-cyclopentyl-N-[(1S)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— (6R)-8-[(2-hydroxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N3O2
(6R)-8-[(2-hydroxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-methoxypropyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O2
(6R)-8-(3-methoxypropyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C15H21N5O2S
(6R)-N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-2-ethyl-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O3
(6S)-2-ethyl-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-(4-propan-2-ylthiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H26N4O2S
(6R)-2-ethyl-8-(4-propan-2-ylthiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide —— C21H28N4O2
6-[(3R)-4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
—— (6-aminopyridin-3-yl)-[(3R)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone —— C18H20FN3O2
(6-aminopyridin-3-yl)-[(3R)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone
—— (6R)-8-(3-acetyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25N5O3
(6R)-8-(3-acetyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(1-benzoxepine-4-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N2O3
(6R)-8-(1-benzoxepine-4-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O2
(6R)-2-benzyl-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one