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—— 6-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— 6-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— 6-Chloro-2-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methylsulfanyl]-3-(2-methylpropyl)quinazolin-4-one —— C20H18ClN3O3S
6-Chloro-2-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methylsulfanyl]-3-(2-methylpropyl)quinazolin-4-one
—— 6-Chloro-3-prop-2-enyl-2-[(1-propyltetrazol-5-yl)methylsulfanyl]quinazolin-4-one —— C16H17ClN6OS
6-Chloro-3-prop-2-enyl-2-[(1-propyltetrazol-5-yl)methylsulfanyl]quinazolin-4-one
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (3aS)-4-oxo-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoxaline-7-carboxylate —— C21H19ClN2O5
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (3aS)-4-oxo-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoxaline-7-carboxylate
—— 6-chloro-8-[(4-chloro-2-nitrophenoxy)methyl]-4H-1,3-benzodioxine —— C15H11Cl2NO5
6-chloro-8-[(4-chloro-2-nitrophenoxy)methyl]-4H-1,3-benzodioxine
—— 6-methyl-N-[6-[(2S)-pyrrolidin-2-yl]pyridin-3-yl]pyridin-2-amine —— C15H18N4
6-methyl-N-[6-[(2S)-pyrrolidin-2-yl]pyridin-3-yl]pyridin-2-amine
—— 6-N-methyl-4-N-[4-[(2R)-piperidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C14H19N7
6-N-methyl-4-N-[4-[(2R)-piperidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 6-methyl-N-[5-[(2S)-piperidin-2-yl]pyridin-2-yl]pyridin-2-amine —— C16H20N4
6-methyl-N-[5-[(2S)-piperidin-2-yl]pyridin-2-yl]pyridin-2-amine
—— 6-methyl-N-[6-[(2R)-pyrrolidin-2-yl]pyridin-3-yl]pyridin-2-amine —— C15H18N4
6-methyl-N-[6-[(2R)-pyrrolidin-2-yl]pyridin-3-yl]pyridin-2-amine
—— (6R)-6-(methoxymethyl)-1-methyl-4-pyrazin-2-yl-1,4-diazepane —— C12H20N4O
(6R)-6-(methoxymethyl)-1-methyl-4-pyrazin-2-yl-1,4-diazepane
—— 6-N-methyl-4-N-[4-[(2S)-piperidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C14H19N7
6-N-methyl-4-N-[4-[(2S)-piperidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 6-N-methyl-4-N-[4-[(2R)-pyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C13H17N7
6-N-methyl-4-N-[4-[(2R)-pyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 6-[(2S)-1-[(3-chlorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine —— C19H19ClN6O2S
6-[(2S)-1-[(3-chlorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine —— C19H20N6O3S
6-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-[(6-methoxy-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C24H26N6O
6-[(2S)-1-[(6-methoxy-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine —— C23H28N6O
6-[(2R)-1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-[(1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine —— C24H26N6
6-[(2R)-1-[(1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2S)-1-[(3-fluorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C20H20FN5O2S
6-[(2S)-1-[(3-fluorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine —— C22H24N6O3
6-[(2S)-1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine —— C19H20N6O3S
6-[(2S)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine
—— 6-N-methyl-4-N-[4-[(2S)-pyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C13H17N7
6-N-methyl-4-N-[4-[(2S)-pyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 6-[(2S)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C24H25FN6
6-[(2S)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2S)-1-[(3,4-dimethylphenyl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C23H27N5
6-[(2S)-1-[(3,4-dimethylphenyl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2S)-1-(4-fluoro-3-methylphenyl)sulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C20H20FN5O2S
6-[(2S)-1-(4-fluoro-3-methylphenyl)sulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-(3,4-dimethylphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine —— C20H22N6O2S
6-[(2S)-1-(3,4-dimethylphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine
—— 6-methyl-N-[5-[(2R)-piperidin-2-yl]pyridin-2-yl]pyridin-2-amine —— C16H20N4
6-methyl-N-[5-[(2R)-piperidin-2-yl]pyridin-2-yl]pyridin-2-amine
—— 6-[(2S)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine —— C24H25FN6
6-[(2S)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2R)-1-[(3,4-dimethylphenyl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C23H27N5
6-[(2R)-1-[(3,4-dimethylphenyl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2S)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C24H27N5O
6-[(2S)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-[(6-methoxy-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C24H26N6O
6-[(2R)-1-[(6-methoxy-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-(2-methoxy-5-methylphenyl)sulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine —— C20H22N6O3S
6-[(2R)-1-(2-methoxy-5-methylphenyl)sulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine —— C24H25FN6
6-[(2R)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2S)-1-[(5-methoxy-1-propan-2-ylindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C26H30N6O
6-[(2S)-1-[(5-methoxy-1-propan-2-ylindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine —— C19H20N6O3S
6-[(2S)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C21H23N5O3S
6-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2R)-1-[(3,4-dimethylphenyl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C22H25N5
6-[(2R)-1-[(3,4-dimethylphenyl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-[(1-ethyl-5-methoxyindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C25H28N6O
6-[(2S)-1-[(1-ethyl-5-methoxyindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-[(1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine —— C24H26N6
6-[(2S)-1-[(1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-N-(6-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2S)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C21H23N5O3S
6-[(2S)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2R)-1-(2-methoxy-5-methylphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine —— C20H22N6O3S
6-[(2R)-1-(2-methoxy-5-methylphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-[(1-propan-2-yl-2,3-dihydroindol-5-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C25H30N6
6-[(2R)-1-[(1-propan-2-yl-2,3-dihydroindol-5-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C24H27N5O3
6-[(2R)-1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine
—— 6-[(2R)-1-[(1-ethyl-5-methoxyindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C25H28N6O
6-[(2R)-1-[(1-ethyl-5-methoxyindol-3-yl)methyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-(3,4-dimethylphenyl)sulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C21H23N5O2S
6-[(2R)-1-(3,4-dimethylphenyl)sulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine —— C19H20N6O3S
6-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrazin-2-amine
—— 6-[(2S)-1-(4-methoxy-2,5-dimethylphenyl)sulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C22H25N5O3S
6-[(2S)-1-(4-methoxy-2,5-dimethylphenyl)sulfonylpyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— 6-[(2R)-1-[[3-(methoxymethyl)-4-propan-2-yloxyphenyl]methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C26H33N5O2
6-[(2R)-1-[[3-(methoxymethyl)-4-propan-2-yloxyphenyl]methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine
—— 6-methyl-N-[6-[(2R)-pyrrolidin-2-yl]pyridin-2-yl]pyridin-2-amine —— C15H18N4
6-methyl-N-[6-[(2R)-pyrrolidin-2-yl]pyridin-2-yl]pyridin-2-amine
—— 6-[(2S)-1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine —— C24H27N5O3
6-[(2S)-1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]pyrrolidin-2-yl]-N-(3-methylpyridin-2-yl)pyrazin-2-amine