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—— 6-(4-Methylcyclohexyl)-2-(1-propan-2-ylsulfonylpiperidin-4-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H36N4O3S
6-(4-Methylcyclohexyl)-2-(1-propan-2-ylsulfonylpiperidin-4-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(3R)-1-(cyclopropanecarbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O3
6-(cyclopropanecarbonyl)-2-[(3R)-1-(cyclopropanecarbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2R)-2-methylbutanoyl]-2-[1-(oxan-4-yl)piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H34N4O3
6-[(2R)-2-methylbutanoyl]-2-[1-(oxan-4-yl)piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-Hydroxyphenyl)methyl]-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H27N5O3
6-[(4-Hydroxyphenyl)methyl]-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(1-ethylpyrazol-4-yl)methyl]-2-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O3
6-[(1-ethylpyrazol-4-yl)methyl]-2-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H36N4O2
6-(cyclohexylmethyl)-2-[1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(2-methylpyrazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-(Cyclohexylmethyl)-2-[1-(2-methylpyrazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H31N5O2S
6-(Cyclohexylmethyl)-2-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Propan-2-yl-2-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H25N5O2S
6-Propan-2-yl-2-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H36N4O2
6-(cyclohexylmethyl)-2-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(2-pyrazol-1-ylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-(Cyclohexylmethyl)-2-[1-(2-pyrazol-1-ylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Propan-2-yl-2-[1-(5-propan-2-yl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H31N5O3
6-Propan-2-yl-2-[1-(5-propan-2-yl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylcyclohexyl)-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(4-Methylcyclohexyl)-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylcyclohexyl)-2-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H32N6O2
6-(4-Methylcyclohexyl)-2-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O2S2
6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Methyl-2-[1-[1-(4-methylphenyl)cyclopentanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H34N4O2
6-Methyl-2-[1-[1-(4-methylphenyl)cyclopentanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H36N4O2
6-(cyclohexylmethyl)-2-[1-[(1S,2S)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O2S2
6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Methyl-2-[1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H30N4O2
6-Methyl-2-[1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butanoyl-2-[(2S)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O2S
6-butanoyl-2-[(2S)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H36N4O2
6-(cyclohexylmethyl)-2-[1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H35N5O2
6-(Cyclohexylmethyl)-2-[1-(2-methylpyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-(butylamino)-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one —— C15H17N3O2S
6-[2-(butylamino)-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one
—— 6-(Cyclohexylmethyl)-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(Cyclohexylmethyl)-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butanoyl-2-[(2R)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O2S
6-butanoyl-2-[(2R)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-(quinoxalin-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H30N6O2
6-Butanoyl-2-[1-(quinoxalin-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-Butanoyl-2-[1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Oxane-4-carbonyl)-2-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H31N5O3
6-(Oxane-4-carbonyl)-2-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Propan-2-yl-2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H27N5O2
6-Propan-2-yl-2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-methylcyclohexyl)-2-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O2
6-(4-methylcyclohexyl)-2-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O2S2
6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(1-methylbenzimidazol-2-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H32N6O2
6-Butanoyl-2-[1-[(1-methylbenzimidazol-2-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O2S2
6-(5-methylthiophene-2-carbonyl)-2-[(2S)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Methyl-2-[1-(2-thiophen-3-ylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H24N4O2S
6-Methyl-2-[1-(2-thiophen-3-ylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Propan-2-yl-2-[1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H31N5O3
6-Propan-2-yl-2-[1-(3-propan-2-yl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Pyridine-3-carbonyl)-2-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H26N6O2
6-(Pyridine-3-carbonyl)-2-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Oxane-4-carbonyl)-2-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H31N5O3
6-(Oxane-4-carbonyl)-2-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Methyl-2-[1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H32N6O2
6-Methyl-2-[1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-(quinoxalin-6-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H30N6O2
6-Butanoyl-2-[1-(quinoxalin-6-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-(Cyclohexylmethyl)-2-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Methyl-2-[1-(2-phenylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H26N4O2
6-Methyl-2-[1-(2-phenylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(Cyclohexylmethyl)-2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-fluoro-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]-1H-indole-2-carboxamide —— C14H14FN5O
6-fluoro-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]-1H-indole-2-carboxamide
—— 6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-(3-fluorophenyl)methanone —— C12H11FN4O
6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-(3-fluorophenyl)methanone
—— 6-Methyl-2-[1-(4-piperidin-1-ylbenzoyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-Methyl-2-[1-(4-piperidin-1-ylbenzoyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-(6-methyl-1H-indol-2-yl)methanone —— C15H15N5O
6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-(6-methyl-1H-indol-2-yl)methanone
—— 6-methoxy-N-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]pyridine-3-carboxamide —— C14H21N3O2
6-methoxy-N-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]pyridine-3-carboxamide
—— 6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-[4-(dimethylamino)phenyl]methanone —— C14H17N5O
6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl-[4-(dimethylamino)phenyl]methanone
—— 6-methoxy-N-[(2R)-1-pyrrolidin-1-ylpropan-2-yl]pyridine-3-carboxamide —— C14H21N3O2
6-methoxy-N-[(2R)-1-pyrrolidin-1-ylpropan-2-yl]pyridine-3-carboxamide
—— 6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl(quinolin-6-yl)methanone —— C15H13N5O
6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl(quinolin-6-yl)methanone