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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6R)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3,6-dimethylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N5O
(6R)-8-(3,6-dimethylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-cyclopentyl-N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-N,1-dimethylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H32N6O
6-cyclopentyl-N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-N,1-dimethylpyrazolo[3,4-d]pyrimidin-4-amine
—— (6S)-2-ethyl-8-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6S)-2-ethyl-8-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2,5-dimethylfuran-3-yl)-8-oxo-N-[(3S)-2-oxopiperidin-3-yl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C21H23N5O4
6-(2,5-dimethylfuran-3-yl)-8-oxo-N-[(3S)-2-oxopiperidin-3-yl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-2-ethyl-8-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6R)-2-ethyl-8-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6-oxo-1H-pyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H24N4O3
(6S)-8-(6-oxo-1H-pyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-fluorophenyl)-7-(3-methylbut-2-enyl)-2-[(2R)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one —— C23H25FN4O2
6-(4-fluorophenyl)-7-(3-methylbut-2-enyl)-2-[(2R)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one
—— (6S)-2-benzyl-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O2
(6S)-2-benzyl-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-pentanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O2
(6R)-8-pentanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O2
(6R)-2-benzyl-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-N,2-dimethyl-3-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C19H21N5O2S
(6S)-N,2-dimethyl-3-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-8-(4-aminopyrimidin-2-yl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O
(6R)-8-(4-aminopyrimidin-2-yl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-pentanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O2
(6S)-8-pentanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-propoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6S)-8-(2-propoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-propoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6R)-8-(2-propoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-2-[(2R)-2-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O2
6-(2-chlorophenyl)-2-[(2R)-2-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— 6-(2-chlorophenyl)-2-[(2S)-2-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O2
6-(2-chlorophenyl)-2-[(2S)-2-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-cyclopentylacetate —— C19H22O5
(6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-cyclopentylacetate
—— 6-(4-fluorophenyl)-7-(3-methylbut-2-enyl)-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one —— C23H25FN4O2
6-(4-fluorophenyl)-7-(3-methylbut-2-enyl)-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-cyclopentylacetate —— C19H22O4
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-cyclopentylacetate
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2,3-dichlorobenzoate —— C16H11Cl3O4
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2,3-dichlorobenzoate
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate —— C20H16ClFO4
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate
—— (6S)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C21H24N2O4
(6S)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-chloro-4-nitrobenzoate —— C16H11Cl2NO6
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-chloro-4-nitrobenzoate
—— (6R)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C21H24N2O4
(6R)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 6-[2-(2-chloro-4-fluorophenoxy)acetyl]-4H-1,4-benzoxazin-3-one —— C16H11ClFNO4
6-[2-(2-chloro-4-fluorophenoxy)acetyl]-4H-1,4-benzoxazin-3-one
—— (6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate —— C20H16ClFO5
(6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(hydroxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C23H22N4O5
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(hydroxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O5
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H19F3N4O3
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylsulfanyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C28H30N4O3S
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylsulfanyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C29H32N4O3
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C30H34N4O3S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-methylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-methylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-2-[(4-chlorophenyl)methylsulfanyl]-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H25ClN4O3S
(6S,9S)-2-[(4-chlorophenyl)methylsulfanyl]-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H26N4O3S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H24N4O3
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H24N4O3S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C23H22N4O4
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H25ClN4O4
(6S,9R)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-pyridin-4-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H23N5O4
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-pyridin-4-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C25H21F3N4O3
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(hydroxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C23H22N4O5
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(hydroxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H19F3N4O3
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C23H19F3N4O4
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H25ClN4O4
(6R,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-2-pyridin-4-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C29H25N5O3
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-2-pyridin-4-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one