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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(2R)-1-[2-(2-fluorophenoxy)acetyl]pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C21H19FN4O3S
6-[(2R)-1-[2-(2-fluorophenoxy)acetyl]pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 6-[(3R)-1-[(3-methylphenyl)methyl]piperidin-3-yl]-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazolo[3,4-b]pyridin-3-amine —— C26H30N6
6-[(3R)-1-[(3-methylphenyl)methyl]piperidin-3-yl]-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazolo[3,4-b]pyridin-3-amine
—— 6-[1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C22H28N4O3S
6-[1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— 6-[1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine —— C25H28N4O3
6-[1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine
—— 6-[(3R)-1-methylsulfonylpiperidin-3-yl]-N-(1-phenylcyclopentyl)pyridine-3-carboxamide —— C23H29N3O3S
6-[(3R)-1-methylsulfonylpiperidin-3-yl]-N-(1-phenylcyclopentyl)pyridine-3-carboxamide
—— 6-methyl-N-[6-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]pyridin-3-yl]pyridin-2-amine —— C21H26N6
6-methyl-N-[6-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]pyridin-3-yl]pyridin-2-amine
—— 6-methyl-N-[6-[1-(1-methylimidazol-4-yl)sulfonylpiperidin-4-yl]pyridin-3-yl]pyridin-2-amine —— C20H24N6O2S
6-methyl-N-[6-[1-(1-methylimidazol-4-yl)sulfonylpiperidin-4-yl]pyridin-3-yl]pyridin-2-amine
—— 6-[1-[[2-(2-methoxyethyl)pyrimidin-5-yl]methyl]piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine —— C23H28N6O
6-[1-[[2-(2-methoxyethyl)pyrimidin-5-yl]methyl]piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine
—— 6-[1-(cyclopropylmethyl)piperidin-4-yl]-N-(5-fluoropyridin-2-yl)pyridin-3-amine —— C19H23FN4
6-[1-(cyclopropylmethyl)piperidin-4-yl]-N-(5-fluoropyridin-2-yl)pyridin-3-amine
—— 6-[1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C22H28N6O3
6-[1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— [6-[1-(2,3-dimethyl-1H-indole-4-carbonyl)piperidin-4-yl]pyridin-3-yl]-piperidin-1-ylmethanone —— C27H32N4O2
[6-[1-(2,3-dimethyl-1H-indole-4-carbonyl)piperidin-4-yl]pyridin-3-yl]-piperidin-1-ylmethanone
—— 6-[(2R)-1-(2,2-dimethylpropyl)pyrrolidin-2-yl]-3-methyl-1-pyridin-2-ylpyrazolo[3,4-b]pyridine —— C21H27N5
6-[(2R)-1-(2,2-dimethylpropyl)pyrrolidin-2-yl]-3-methyl-1-pyridin-2-ylpyrazolo[3,4-b]pyridine
—— 6-[1-(6-methoxypyridine-3-carbonyl)piperidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C23H28N4O4
6-[1-(6-methoxypyridine-3-carbonyl)piperidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— 6-methyl-N-[6-[1-(2-phenylethylsulfonyl)piperidin-4-yl]pyridin-3-yl]pyridin-2-amine —— C24H28N4O2S
6-methyl-N-[6-[1-(2-phenylethylsulfonyl)piperidin-4-yl]pyridin-3-yl]pyridin-2-amine
—— [6-[(2S)-1-(2,3-dimethyl-1H-indole-4-carbonyl)pyrrolidin-2-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C26H31N5O2
[6-[(2S)-1-(2,3-dimethyl-1H-indole-4-carbonyl)pyrrolidin-2-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— 6-[1-(6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl)piperidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C24H28N6O3
6-[1-(6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl)piperidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— 6-[(3R)-1-methylsulfonylpiperidin-3-yl]-N-(3-pyrazol-1-ylpropyl)pyridine-3-carboxamide —— C18H25N5O3S
6-[(3R)-1-methylsulfonylpiperidin-3-yl]-N-(3-pyrazol-1-ylpropyl)pyridine-3-carboxamide
—— 6-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine —— C20H23N5O3S
6-[1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine
—— 6-[1-(1-methylimidazol-4-yl)sulfonylpiperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine —— C19H22N6O2S
6-[1-(1-methylimidazol-4-yl)sulfonylpiperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine
—— 6-[1-(1-ethyl-3-methylpyrazol-4-yl)sulfonylpiperidin-4-yl]-N-(5-fluoropyridin-2-yl)pyridin-3-amine —— C21H25FN6O2S
6-[1-(1-ethyl-3-methylpyrazol-4-yl)sulfonylpiperidin-4-yl]-N-(5-fluoropyridin-2-yl)pyridin-3-amine
—— (6S)-1-(1H-imidazol-2-ylmethyl)-4-phenyl-6-(pyridin-2-ylmethyl)-1,4-diazepane —— C21H25N5
(6S)-1-(1H-imidazol-2-ylmethyl)-4-phenyl-6-(pyridin-2-ylmethyl)-1,4-diazepane
—— 6-[1-[2-(1-ethylpiperidin-4-yl)acetyl]piperidin-4-yl]-N,N-dimethylpyridine-3-carboxamide —— C22H34N4O2
6-[1-[2-(1-ethylpiperidin-4-yl)acetyl]piperidin-4-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[(3S)-1-methylsulfonylpiperidin-3-yl]-N-(1-phenylcyclopentyl)pyridine-3-carboxamide —— C23H29N3O3S
6-[(3S)-1-methylsulfonylpiperidin-3-yl]-N-(1-phenylcyclopentyl)pyridine-3-carboxamide
—— 6-[(3R)-1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C23H23FN6O2
6-[(3R)-1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— 6-[1-(4-methoxy-3-methylphenyl)sulfonylpiperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine —— C23H26N4O3S
6-[1-(4-methoxy-3-methylphenyl)sulfonylpiperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine
—— 6-methyl-N-[6-[1-[(1-methylpyrazol-4-yl)methyl]piperidin-4-yl]pyridin-3-yl]pyridin-2-amine —— C21H26N6
6-methyl-N-[6-[1-[(1-methylpyrazol-4-yl)methyl]piperidin-4-yl]pyridin-3-yl]pyridin-2-amine
—— 6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(5-fluoropyridin-2-yl)pyridin-3-amine —— C21H23FN6
6-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(5-fluoropyridin-2-yl)pyridin-3-amine
—— 6-[(3S)-1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C23H23FN6O2
6-[(3S)-1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— (6-fluoro-1H-indol-2-yl)-[3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone —— C18H19FN6O
(6-fluoro-1H-indol-2-yl)-[3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone
—— 6-[[3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methyl]quinoline —— C20H24N6
6-[[3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methyl]quinoline
—— (6-fluoro-1H-indol-2-yl)-[3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone —— C18H19FN6O
(6-fluoro-1H-indol-2-yl)-[3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methanone
—— 6-[[3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methyl]quinoline —— C20H24N6
6-[[3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]methyl]quinoline
—— (6-chloro-1H-indol-2-yl)-[(2S)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)piperidin-1-yl]methanone —— C20H23ClN6O
(6-chloro-1H-indol-2-yl)-[(2S)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)piperidin-1-yl]methanone
—— 6-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine —— C21H24N6
6-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-N-pyridin-2-ylpyridin-3-amine
—— (6-chloro-1H-indol-2-yl)-[(2R)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)piperidin-1-yl]methanone —— C20H23ClN6O
(6-chloro-1H-indol-2-yl)-[(2R)-2-(7-methyl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)piperidin-1-yl]methanone
—— (6-aminopyridin-3-yl)-[(2R)-2-[4-methyl-8-(2-phenylethyl)-6,7-dihydro-5H-pyrido[2,3-d]pyrimidin-2-yl]pyrrolidin-1-yl]methanone —— C26H30N6O
(6-aminopyridin-3-yl)-[(2R)-2-[4-methyl-8-(2-phenylethyl)-6,7-dihydro-5H-pyrido[2,3-d]pyrimidin-2-yl]pyrrolidin-1-yl]methanone
—— (6-aminopyridin-3-yl)-[(2S)-2-[4-methyl-8-(2-phenylethyl)-6,7-dihydro-5H-pyrido[2,3-d]pyrimidin-2-yl]pyrrolidin-1-yl]methanone —— C26H30N6O
(6-aminopyridin-3-yl)-[(2S)-2-[4-methyl-8-(2-phenylethyl)-6,7-dihydro-5H-pyrido[2,3-d]pyrimidin-2-yl]pyrrolidin-1-yl]methanone
—— (6R)-8-[(4-fluorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one —— C17H16FN3O
(6R)-8-[(4-fluorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one
—— 6-Phenyl-8-(pyrrolidin-1-ylmethyl)tetrazolo[1,5-a]pyridine —— C16H17N5
6-Phenyl-8-(pyrrolidin-1-ylmethyl)tetrazolo[1,5-a]pyridine
—— (6S)-8-[(4-fluorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one —— C17H16FN3O
(6S)-8-[(4-fluorophenyl)methyl]-2,8,13-triazatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-7-one
—— 6-(3,4-Dimethylphenyl)-2,3-dimethylimidazo[1,2-b][1,2,4]triazine —— C15H16N4
6-(3,4-Dimethylphenyl)-2,3-dimethylimidazo[1,2-b][1,2,4]triazine
—— 6-(4-Methoxyphenyl)-2-(piperidin-4-ylmethyl)pyridazin-3-one —— C17H21N3O2
6-(4-Methoxyphenyl)-2-(piperidin-4-ylmethyl)pyridazin-3-one
—— 6-[2-(1H-benzimidazol-2-yl)ethyl]-2-methyl-N-[(1R)-2-morpholin-4-yl-1-phenylethyl]pyrimidin-4-amine —— C26H30N6O
6-[2-(1H-benzimidazol-2-yl)ethyl]-2-methyl-N-[(1R)-2-morpholin-4-yl-1-phenylethyl]pyrimidin-4-amine
—— 6-[(2-methylbenzimidazol-1-yl)methyl]-4-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]pyrimidine-2,4-diamine —— C24H28N6O
6-[(2-methylbenzimidazol-1-yl)methyl]-4-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]pyrimidine-2,4-diamine
—— 6-(benzotriazol-1-ylmethyl)-N-[(2R)-1-(4-chlorophenoxy)propan-2-yl]-2-methylpyrimidin-4-amine —— C21H21ClN6O
6-(benzotriazol-1-ylmethyl)-N-[(2R)-1-(4-chlorophenoxy)propan-2-yl]-2-methylpyrimidin-4-amine
—— 6-(5-Chlorothiophen-2-yl)-2,3-dimethylimidazo[1,2-b][1,2,4]triazine —— C11H9ClN4S
6-(5-Chlorothiophen-2-yl)-2,3-dimethylimidazo[1,2-b][1,2,4]triazine
—— 6-(5-ethyl-2-methylpyrazol-3-yl)-N-[(2R)-1-(2-methoxyphenyl)propan-2-yl]-2-methylpyrimidin-4-amine —— C21H27N5O
6-(5-ethyl-2-methylpyrazol-3-yl)-N-[(2R)-1-(2-methoxyphenyl)propan-2-yl]-2-methylpyrimidin-4-amine
—— 6-(5-Bromothiophen-2-yl)-2,3-dipyridin-2-ylimidazo[1,2-b][1,2,4]triazine —— C19H11BrN6S
6-(5-Bromothiophen-2-yl)-2,3-dipyridin-2-ylimidazo[1,2-b][1,2,4]triazine
—— 6-(2,3-Dihydro-1,4-benzodioxin-6-yl)-2,3-diethylimidazo[1,2-b][1,2,4]triazine —— C17H18N4O2
6-(2,3-Dihydro-1,4-benzodioxin-6-yl)-2,3-diethylimidazo[1,2-b][1,2,4]triazine
—— 6-[(2-methylbenzimidazol-1-yl)methyl]-4-N-[(1S)-1-(4-propan-2-yloxyphenyl)ethyl]pyrimidine-2,4-diamine —— C24H28N6O
6-[(2-methylbenzimidazol-1-yl)methyl]-4-N-[(1S)-1-(4-propan-2-yloxyphenyl)ethyl]pyrimidine-2,4-diamine