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—— 6-(2,5-dimethylfuran-3-yl)-N-[(2S)-2-hydroxypropyl]-N-methyl-7-(3-methylbut-2-enyl)-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C22H28N4O4
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-2-hydroxypropyl]-N-methyl-7-(3-methylbut-2-enyl)-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-fluoro-2-[(2R)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C17H18FN3S
6-fluoro-2-[(2R)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-8-(3-acetyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25N5O3
(6S)-8-(3-acetyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(2-hydroxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N3O2
(6S)-8-[(2-hydroxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(1-benzoxepine-4-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N2O3
(6S)-8-(1-benzoxepine-4-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6-aminopyridin-3-yl)-[(3S)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone —— C18H20FN3O2
(6-aminopyridin-3-yl)-[(3S)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]methanone
—— (6R)-2-ethyl-8-[5-(tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C16H22N8O2
(6R)-2-ethyl-8-[5-(tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C16H26N4O2
(6S)-2-ethyl-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]amino]pyridine-3-carbonitrile —— C17H16F3N5
6-[[(3R)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]amino]pyridine-3-carbonitrile
—— (6S)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6S)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]amino]pyridine-3-carbonitrile —— C17H16F3N5
6-[[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]amino]pyridine-3-carbonitrile
—— 6-fluoro-2-[(2S)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C17H18FN3S
6-fluoro-2-[(2S)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6R)-2-ethyl-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C16H26N4O2
(6R)-2-ethyl-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(4-propan-2-ylthiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H26N4O2S
(6S)-2-ethyl-8-(4-propan-2-ylthiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-[(E)-pent-3-enoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N2O2
(6S)-2-benzyl-8-[(E)-pent-3-enoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2S)-1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile —— C17H23N3O2
6-[(2S)-1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile
—— (6S)-8-[(6-chloropyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28ClN3O2
(6S)-8-[(6-chloropyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2R)-2-hydroxypropyl]-N-methyl-7-(3-methylbut-2-enyl)-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C22H28N4O4
6-(2,5-dimethylfuran-3-yl)-N-[(2R)-2-hydroxypropyl]-N-methyl-7-(3-methylbut-2-enyl)-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(6-chloropyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28ClN3O2
(6R)-8-[(6-chloropyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]-N,N-dimethylpyrimidin-4-amine —— C22H33N5O2
6-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]-N,N-dimethylpyrimidin-4-amine
—— (6S)-8-(3-amino-1H-pyrazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N6O2
(6S)-8-(3-amino-1H-pyrazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-5-[4-[(1S)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile —— C19H26N4O3
6-methyl-5-[4-[(1S)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile
—— (6S)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6S)-8-(4-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-[(E)-pent-3-enoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N2O2
(6R)-2-benzyl-8-[(E)-pent-3-enoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6S)-8-(5-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6S)-2-ethyl-8-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6R)-8-(5-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-N-[(2R)-2-hydroxypropyl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C18H19ClN4O3
6-(2-chlorophenyl)-N-[(2R)-2-hydroxypropyl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2-chlorophenyl)-2-[(3S)-3-ethylpiperazine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H24ClN5O2
6-(2-chlorophenyl)-2-[(3S)-3-ethylpiperazine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6S)-8-(2-methoxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N3O2
(6S)-8-(2-methoxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-5-[4-[(1R)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile —— C19H26N4O3
6-methyl-5-[4-[(1R)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile
—— 6-(2-chlorophenyl)-2-[(3R)-3-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O2
6-(2-chlorophenyl)-2-[(3R)-3-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— 6-(2-chlorophenyl)-2-[(3S)-3-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H23ClN4O2
6-(2-chlorophenyl)-2-[(3S)-3-methylpiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— (6R)-2-ethyl-8-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6R)-2-ethyl-8-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-2-[(3R)-3-ethylpiperazine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H24ClN5O2
6-(2-chlorophenyl)-2-[(3R)-3-ethylpiperazine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— 6-[(2R)-1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile —— C17H23N3O2
6-[(2R)-1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile
—— (6R)-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H25N5O2
(6R)-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-(diethylamino)acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-8-[2-(diethylamino)acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[2-(diethylamino)acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6R)-8-[2-(diethylamino)acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-methoxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N3O2
(6R)-8-(2-methoxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-N-[(2S)-2-hydroxypropyl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C18H19ClN4O3
6-(2-chlorophenyl)-N-[(2S)-2-hydroxypropyl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-8-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N5O2
(6S)-8-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(1,3-benzoxazol-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O3
(6S)-8-(1,3-benzoxazol-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(1,3-benzoxazol-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O3
(6R)-8-(1,3-benzoxazol-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-methoxypyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-8-(6-methoxypyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-cyclopentylpropyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H35N3O
(6R)-8-(3-cyclopentylpropyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-(2-propan-2-yloxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6S)-2-benzyl-8-(2-propan-2-yloxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-N-(2-methylphenyl)-3-oxo-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C21H31N3O3
(6S)-2-(3-methoxypropyl)-N-(2-methylphenyl)-3-oxo-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— 6-(4-fluorophenyl)-N-[(2R)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C19H19FN4O3
6-(4-fluorophenyl)-N-[(2R)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide