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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-2-(3-methoxypropyl)-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O2
(6S)-2-(3-methoxypropyl)-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N5O
(6R)-8-(5-propylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-(4-methylnaphthalene-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H28N2O2
(6R)-2-ethyl-8-(4-methylnaphthalene-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-2-carbonitrile —— C20H24N6
6-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-2-carbonitrile
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethenylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O
(6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethenylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine-2,4-diamine —— C17H27N9
6-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine-2,4-diamine
—— (6S)-2-ethyl-8-(4-methylnaphthalene-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H28N2O2
(6S)-2-ethyl-8-(4-methylnaphthalene-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-8-(5-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-N-[2-(2-nitroanilino)ethyl]-4-oxo-1-phenylpyridazine-3-carboxamide —— C20H19N5O4
6-methyl-N-[2-(2-nitroanilino)ethyl]-4-oxo-1-phenylpyridazine-3-carboxamide
—— (6S)-2-ethyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O3
(6S)-2-ethyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-2-carbonitrile —— C20H24N6
6-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]pyridine-2-carbonitrile
—— (6S)-8-(5-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6S)-8-(5-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-pent-2-ynyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O
(6R)-8-pent-2-ynyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O3
(6S)-2-ethyl-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methoxypropyl)-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O2
(6R)-2-(3-methoxypropyl)-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O3
(6R)-2-ethyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-chloro-3-fluoropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H26ClFN4O
(6S)-8-(5-chloro-3-fluoropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-4-oxo-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-1-phenylpyridazine-3-carboxamide —— C22H20N4O3
6-methyl-4-oxo-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-1-phenylpyridazine-3-carboxamide
—— (6S)-2-ethyl-8-(2-pyridin-4-ylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25N5O2
(6S)-2-ethyl-8-(2-pyridin-4-ylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-1-[3-oxo-3-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]propyl]pyridin-2-one —— C20H31N3O2
6-methyl-1-[3-oxo-3-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]propyl]pyridin-2-one
—— (6R)-8-(5-chloro-3-fluoropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H26ClFN4O
(6R)-8-(5-chloro-3-fluoropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-5-[2-oxo-2-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione —— C18H28N4O3
6-methyl-5-[2-oxo-2-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione
—— 6-methyl-5-[2-oxo-2-[4-[(1S)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione —— C18H28N4O3
6-methyl-5-[2-oxo-2-[4-[(1S)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione
—— 6-[(2R)-1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile —— C18H24N4O2
6-[(2R)-1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile
—— 6-[(6R)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C21H23N5O
6-[(6R)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— 6-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyrimidin-4-amine —— C20H29N5O2
6-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyrimidin-4-amine
—— (6R)-8-(4-ethyl-5-methylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6R)-8-(4-ethyl-5-methylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O3
(6R)-2-ethyl-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-pent-2-ynyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O
(6S)-8-pent-2-ynyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyrimidin-4-amine —— C20H29N5O2
6-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyrimidin-4-amine
—— 6-[(2S)-1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile —— C18H24N4O2
6-[(2S)-1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile
—— 6-methyl-2-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C20H27N7
6-methyl-2-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-methyl-4-oxo-N-[2-oxo-2-(propan-2-ylamino)ethyl]-1-[3-(trifluoromethyl)phenyl]pyridazine-3-carboxamide —— C18H19F3N4O3
6-methyl-4-oxo-N-[2-oxo-2-(propan-2-ylamino)ethyl]-1-[3-(trifluoromethyl)phenyl]pyridazine-3-carboxamide
—— 6-[(6S)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C21H23N5O
6-[(6S)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— (6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(2S)-2-pyridin-2-ylpiperidin-1-yl]methanone —— C17H16ClN5O
(6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(2S)-2-pyridin-2-ylpiperidin-1-yl]methanone
—— 6-methyl-1-[3-oxo-3-[4-[(1S)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]propyl]pyridin-2-one —— C20H31N3O2
6-methyl-1-[3-oxo-3-[4-[(1S)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]propyl]pyridin-2-one
—— (6S)-8-[4-(methylamino)pyrimidin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N6O
(6S)-8-[4-(methylamino)pyrimidin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6S)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-1-(2-nitrophenyl)-4-oxo-N-[2-oxo-2-(propan-2-ylamino)ethyl]pyridazine-3-carboxamide —— C17H19N5O5
6-methyl-1-(2-nitrophenyl)-4-oxo-N-[2-oxo-2-(propan-2-ylamino)ethyl]pyridazine-3-carboxamide
—— (6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(2R)-2-pyridin-2-ylpiperidin-1-yl]methanone —— C17H16ClN5O
(6-chloroimidazo[1,2-a]pyrimidin-2-yl)-[(2R)-2-pyridin-2-ylpiperidin-1-yl]methanone
—— 6-methyl-2-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C20H27N7
6-methyl-2-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— (6R)-8-[4-(methylamino)pyrimidin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N6O
(6R)-8-[4-(methylamino)pyrimidin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6S)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-8-(5-methyl-1H-imidazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(4,6-dimethylquinolin-2-yl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N3O
(6S)-8-(4,6-dimethylquinolin-2-yl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl]pyridine-2-carbonitrile —— C21H26N4O3
6-[(3S)-4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl]pyridine-2-carbonitrile
—— (6R)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O
(6R)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1H-pyrrolo[2,3-b]pyridine —— C20H23N3O2
6-[(3S)-3-[(3-methoxyphenoxy)methyl]piperidin-1-yl]-1H-pyrrolo[2,3-b]pyridine
—— (6S)-8-(3-fluoropyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23FN4O
(6S)-8-(3-fluoropyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one