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—— (6-methyl-1H-indol-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H20N4O
(6-methyl-1H-indol-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 6-methyl-5-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-3H-furo[2,3-d]pyrimidin-4-one —— C16H17N5O3
6-methyl-5-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-3H-furo[2,3-d]pyrimidin-4-one
—— 6-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H15N5O2S
6-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6R)-6-(3-methoxy-4-propoxyphenyl)-9,9-dimethyl-5-propanoyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H34N2O4
(6R)-6-(3-methoxy-4-propoxyphenyl)-9,9-dimethyl-5-propanoyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6-morpholin-4-ylpyridin-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone —— C18H23N5O2
(6-morpholin-4-ylpyridin-3-yl)-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methanone
—— 6,7-dihydro-4H-thieno[3,2-c]pyran-2-yl-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C18H23N3O2S
6,7-dihydro-4H-thieno[3,2-c]pyran-2-yl-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (6R)-5-hexanoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C34H38N2O3
(6R)-5-hexanoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— [6-(cyclopropylamino)pyridin-3-yl]-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C19H25N5O
[6-(cyclopropylamino)pyridin-3-yl]-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (6S)-5-hexanoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C34H38N2O3
(6S)-5-hexanoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(3-methoxy-4-propoxyphenyl)-9,9-dimethyl-5-propanoyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H34N2O4
(6S)-6-(3-methoxy-4-propoxyphenyl)-9,9-dimethyl-5-propanoyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-[(Z)-1-bromo-2-phenylethenyl]-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C23H23BrN2O
(6S)-6-[(Z)-1-bromo-2-phenylethenyl]-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-6-[(Z)-1-bromo-2-phenylethenyl]-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C23H23BrN2O
(6R)-6-[(Z)-1-bromo-2-phenylethenyl]-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-benzoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C35H32N2O3
(6S)-5-benzoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6,7-dihydro-4H-thieno[3,2-c]pyran-2-yl-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C18H23N3O2S
6,7-dihydro-4H-thieno[3,2-c]pyran-2-yl-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (6R)-5-benzoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C35H32N2O3
(6R)-5-benzoyl-9,9-dimethyl-6-(2-phenylmethoxyphenyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-2-benzoyl-6-(3,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C28H24Cl2N2O2
(6R)-2-benzoyl-6-(3,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H15N5O2S
6-[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6R)-5-(4-bromobenzoyl)-6-(4-fluorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H24BrFN2O2
(6R)-5-(4-bromobenzoyl)-6-(4-fluorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(3,4-dichlorophenyl)-9,9-dimethyl-5-(3-methylbutanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H28Cl2N2O2
(6S)-6-(3,4-dichlorophenyl)-9,9-dimethyl-5-(3-methylbutanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6-fluoro-1H-benzimidazol-4-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C18H20FN5O
(6-fluoro-1H-benzimidazol-4-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— [6-(dimethylamino)pyridin-3-yl]-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C18H25N5O
[6-(dimethylamino)pyridin-3-yl]-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (6-fluoro-1H-benzimidazol-4-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C18H20FN5O
(6-fluoro-1H-benzimidazol-4-yl)-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— [6-(cyclopropylamino)pyridin-3-yl]-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C19H25N5O
[6-(cyclopropylamino)pyridin-3-yl]-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— [6-(dimethylamino)pyridin-3-yl]-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone —— C18H25N5O
[6-(dimethylamino)pyridin-3-yl]-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methanone
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-(3,5-dimethyl-4-nitropyrazol-1-yl)acetate —— C19H19N3O6
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-(3,5-dimethyl-4-nitropyrazol-1-yl)acetate
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-(3,5-dimethyl-4-nitropyrazol-1-yl)acetate —— C16H16ClN3O6
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-(3,5-dimethyl-4-nitropyrazol-1-yl)acetate
—— 6-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-propylpyridazin-3-one —— C18H25N5O2
6-[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-propylpyridazin-3-one
—— 6-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-methylpyridine-3-carbonitrile —— C19H23N5O
6-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-methylpyridine-3-carbonitrile
—— 6-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-propylpyridazin-3-one —— C18H25N5O2
6-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-propylpyridazin-3-one
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl (E)-3-(5-bromofuran-2-yl)prop-2-enoate —— C19H15BrO5
(6,7-dimethyl-2-oxochromen-4-yl)methyl (E)-3-(5-bromofuran-2-yl)prop-2-enoate
—— 6-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C17H23N5O2
6-[(2R)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— [6-(dimethylamino)pyridin-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H23N5O
[6-(dimethylamino)pyridin-3-yl]-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 6-[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-methylpyridine-3-carbonitrile —— C19H23N5O
6-[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]piperidine-1-carbonyl]-2-methylpyridine-3-carbonitrile
—— [6-(dimethylamino)pyridin-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C17H23N5O
[6-(dimethylamino)pyridin-3-yl]-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(5-bromofuran-2-yl)prop-2-enoate —— C16H12BrClO5
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(5-bromofuran-2-yl)prop-2-enoate
—— 6-[(2S)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H17N5O2S
6-[(2S)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— [(6R)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone —— C18H24N4OS
[(6R)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone
—— 6-[(2R)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H17N5O2S
6-[(2R)-2-(pyrazol-1-ylmethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-[[(3S)-4-(2-methoxyethyl)-3-methylpiperazin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C14H22N4OS
6-[[(3S)-4-(2-methoxyethyl)-3-methylpiperazin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— [(6S)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone —— C18H24N4OS
[(6S)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl]-(3-propan-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)methanone
—— 6-[[(3R)-4-(2-methoxyethyl)-3-methylpiperazin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C14H22N4OS
6-[[(3R)-4-(2-methoxyethyl)-3-methylpiperazin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— (6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl benzoate —— C19H16O5
(6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl benzoate
—— 6-[4-[(2S)-2-hydroxy-3,3-dimethylbutyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one —— C16H26N4O3
6-[4-[(2S)-2-hydroxy-3,3-dimethylbutyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one
—— 6-[4-[(2R)-2-hydroxy-3,3-dimethylbutyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one —— C16H26N4O3
6-[4-[(2R)-2-hydroxy-3,3-dimethylbutyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one
—— (6-chloro-7-methyl-2-oxochromen-4-yl)methyl (E)-2-cyano-3-(4-methoxyphenyl)prop-2-enoate —— C22H16ClNO5
(6-chloro-7-methyl-2-oxochromen-4-yl)methyl (E)-2-cyano-3-(4-methoxyphenyl)prop-2-enoate
—— 6-[[(3S)-3-methyl-4-(4-methyl-1,3-thiazol-2-yl)piperazin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C15H19N5S2
6-[[(3S)-3-methyl-4-(4-methyl-1,3-thiazol-2-yl)piperazin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— 6-[4-[(1R)-1-(3-fluorophenyl)ethyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine —— C18H21FN6
6-[4-[(1R)-1-(3-fluorophenyl)ethyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(4-chlorophenyl)prop-2-enoate —— C18H14Cl2O4
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(4-chlorophenyl)prop-2-enoate
—— 6-[4-[(1S)-1-(4-fluorophenyl)ethyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine —— C18H21FN6
6-[4-[(1S)-1-(4-fluorophenyl)ethyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine
—— 6-[4-[(1R)-1-(4-fluorophenyl)ethyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine —— C18H21FN6
6-[4-[(1R)-1-(4-fluorophenyl)ethyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine