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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-cyclopentyl-1-methyl-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C18H25N7
6-cyclopentyl-1-methyl-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-[(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)sulfanylmethyl]-1,3,5-triazine-2,4-diamine —— C11H13N9S
6-[(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)sulfanylmethyl]-1,3,5-triazine-2,4-diamine
—— (6S)-8-(2-amino-2-methylpropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6S)-8-(2-amino-2-methylpropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-butoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O3
(6S)-8-(2-butoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-butoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O3
(6R)-8-(2-butoxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6-aminohexanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-8-(6-aminohexanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(6R)-2-benzyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile —— C22H24N4O
6-[(6R)-2-benzyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile
—— (6S)-2-ethyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O3
(6S)-2-ethyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-(1H-pyrrolo[2,3-b]pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N4O2
(6R)-2-ethyl-8-(1H-pyrrolo[2,3-b]pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O3
(6R)-2-ethyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-aminohexanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6R)-8-(6-aminohexanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(4-aminopyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N6O
(6S)-8-(4-aminopyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(4-aminopyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N6O
(6R)-8-(4-aminopyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]amino]pyridine-2-carbonitrile —— C17H19N5
6-[[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]amino]pyridine-2-carbonitrile
—— (6S)-2-(3-methoxypropyl)-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3
(6S)-2-(3-methoxypropyl)-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(1H-pyrrolo[2,3-b]pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N4O2
(6S)-2-ethyl-8-(1H-pyrrolo[2,3-b]pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-pyridin-4-ylacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6R)-8-(2-pyridin-4-ylacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O2
(6R)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(4-chlorobenzoyl)amino]acetate —— C19H17Cl2NO5
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(4-chlorobenzoyl)amino]acetate
—— [6-[(3R)-3-(2-phenylethyl)piperidin-1-yl]pyridin-3-yl]-piperidin-1-ylmethanone —— C24H31N3O
[6-[(3R)-3-(2-phenylethyl)piperidin-1-yl]pyridin-3-yl]-piperidin-1-ylmethanone
—— (6S)-8-(2-morpholin-4-ylethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-8-(2-morpholin-4-ylethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-pyridin-4-ylacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6S)-8-(2-pyridin-4-ylacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C18H17ClN4O4
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate
—— 6-[2-[5-(2-chlorophenyl)tetrazol-2-yl]acetyl]-3,4-dihydro-1H-quinolin-2-one —— C18H14ClN5O2
6-[2-[5-(2-chlorophenyl)tetrazol-2-yl]acetyl]-3,4-dihydro-1H-quinolin-2-one
—— [6-[(3S)-3-(2-phenylethyl)piperidin-1-yl]pyridin-3-yl]-piperidin-1-ylmethanone —— C24H31N3O
[6-[(3S)-3-(2-phenylethyl)piperidin-1-yl]pyridin-3-yl]-piperidin-1-ylmethanone
—— 6-[(2-cyanophenyl)methylsulfanyl]-N-cyclohexyl-N-methylpyridine-3-sulfonamide —— C20H23N3O2S2
6-[(2-cyanophenyl)methylsulfanyl]-N-cyclohexyl-N-methylpyridine-3-sulfonamide
—— (6S)-2-benzyl-8-[[5-(hydroxymethyl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N2O3
(6S)-2-benzyl-8-[[5-(hydroxymethyl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methoxypropyl)-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O2
(6R)-2-(3-methoxypropyl)-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6S)-8-(6-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-7-methyl-8-oxo-N-[(2R)-pentan-2-yl]imidazo[1,2-a]pyrazine-2-carboxamide —— C19H21ClN4O2
6-(2-chlorophenyl)-7-methyl-8-oxo-N-[(2R)-pentan-2-yl]imidazo[1,2-a]pyrazine-2-carboxamide
—— 6-[(2S)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C15H16N4O3
6-[(2S)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-(4-fluorophenyl)-2-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxylic acid —— C18H19FN2O4
6-(4-fluorophenyl)-2-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxylic acid
—— (6R)-2-ethyl-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6R)-2-ethyl-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2R)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C19H22N4O4
6-(2,5-dimethylfuran-3-yl)-N-[(2R)-2-hydroxypropyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-2-benzyl-8-[[5-(hydroxymethyl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N2O3
(6R)-2-benzyl-8-[[5-(hydroxymethyl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(pyridin-2-ylmethyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H24N4O2
(6R)-2-(pyridin-2-ylmethyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-8-[2-[methyl(propan-2-yl)amino]acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6R)-8-(6-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2R)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C15H16N4O3
6-[(2R)-2-pyridin-2-ylpiperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (6R)-2-[2-(dimethylamino)ethyl]-8-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O
(6R)-2-[2-(dimethylamino)ethyl]-8-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-oxo-1H-pyrimidine-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23N5O3
(6R)-8-(6-oxo-1H-pyrimidine-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N4O
(6R)-2-benzyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [6-[[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C22H29N5O2
[6-[[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— (6R)-8-hexanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6R)-8-hexanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2
(6S)-2-ethyl-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-hexanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6S)-8-hexanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O2
(6S)-2-(3-methoxypropyl)-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— [6-[[(3S)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C22H29N5O2
[6-[[(3S)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— (6S)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O2
(6S)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-fluorophenyl)-2-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxylic acid —— C18H19FN2O4
6-(4-fluorophenyl)-2-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxylic acid