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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-Butanoyl-2-[1-(3-fluorobenzoyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H27FN4O3
6-Butanoyl-2-[1-(3-fluorobenzoyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(2,4-difluorophenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H28F2N4O2
6-Butanoyl-2-[1-[(2,4-difluorophenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(5-Methylthiophen-3-yl)methyl]-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27N5O2S
6-[(5-Methylthiophen-3-yl)methyl]-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N4O3
6-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-Ethyl-1,2-oxazole-3-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H31N5O4
6-(5-Ethyl-1,2-oxazole-3-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-(2-ethylpyrazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H30N6O3
6-Butanoyl-2-[1-(2-ethylpyrazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-hydroxyphenyl)methyl]-2-[1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H30N4O3
6-[(4-hydroxyphenyl)methyl]-2-[1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(pyridin-3-ylmethyl)-2-[(2R)-1-(2-thiophen-3-ylacetyl)piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27N5O2S
6-(pyridin-3-ylmethyl)-2-[(2R)-1-(2-thiophen-3-ylacetyl)piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylbenzoyl)-2-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H29N5O2
6-(4-Methylbenzoyl)-2-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(2-hydroxy-4-methylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H32N4O3
6-Butanoyl-2-[1-[(2-hydroxy-4-methylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butanoyl-2-[(2S)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O2S
6-butanoyl-2-[(2S)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-(cyclopropanecarbonyl)-2-[1-[(2R)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylbenzoyl)-2-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H28N4O2S
6-(4-Methylbenzoyl)-2-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[1-[(2S)-2-methylbutanoyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H38N4O2
6-(cyclohexylmethyl)-2-[1-[(2S)-2-methylbutanoyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclopropanecarbonyl)-2-[1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N6O2
6-(Cyclopropanecarbonyl)-2-[1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclobutanecarbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H32N4O3
6-(Cyclobutanecarbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-Methylthiophene-2-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O3S
6-(5-Methylthiophene-2-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O2
6-Butanoyl-2-[1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-(2-pyridin-2-ylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H29N5O3
6-Butanoyl-2-[1-(2-pyridin-2-ylacetyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H34N4O3
6-Butanoyl-2-[1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Oxane-4-carbonyl)-2-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O3S
6-(Oxane-4-carbonyl)-2-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H32N6O2
6-(Cyclohexylmethyl)-2-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-hydroxyphenyl)methyl]-2-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H30N4O3
6-[(4-hydroxyphenyl)methyl]-2-[1-[(1S,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylbenzoyl)-2-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H28N4O2S
6-(4-Methylbenzoyl)-2-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H32N4O3
6-(cyclopentanecarbonyl)-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(5-Methylthiophen-3-yl)methyl]-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27N5O2S
6-[(5-Methylthiophen-3-yl)methyl]-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butanoyl-2-[1-(2H-chromen-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-butanoyl-2-[1-(2H-chromen-3-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(1-Ethylpyrazole-3-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O3
6-(1-Ethylpyrazole-3-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclopropanecarbonyl)-2-[1-[(2-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H32N4O3
6-(Cyclopropanecarbonyl)-2-[1-[(2-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(2,5-dimethylthiophen-3-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O2S
6-Butanoyl-2-[1-[(2,5-dimethylthiophen-3-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-Hydroxyphenyl)methyl]-2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H27N5O3
6-[(4-Hydroxyphenyl)methyl]-2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Methylsulfonyl-2-[1-[(4-propan-2-ylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O3S
6-Methylsulfonyl-2-[1-[(4-propan-2-ylphenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(3S)-1-(cyclopropanecarbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O3
6-(cyclopropanecarbonyl)-2-[(3S)-1-(cyclopropanecarbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(5-Methylthiophene-3-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N4O3S
6-(5-Methylthiophene-3-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butanoyl-2-[(2R)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O2S
6-butanoyl-2-[(2R)-1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(Cyclohexylmethyl)-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Butanoyl-2-[1-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H32N6O2
6-Butanoyl-2-[1-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexylmethyl)-2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O3
6-(Cyclohexylmethyl)-2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylcyclohexyl)-2-[1-(1-methylpyrazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-(4-Methylcyclohexyl)-2-[1-(1-methylpyrazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylcyclohexyl)-2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O3
6-(4-Methylcyclohexyl)-2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butanoyl-2-[(2S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H30N4O3
6-butanoyl-2-[(2S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclohexanecarbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H36N4O3
6-(Cyclohexanecarbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Cyclopropanecarbonyl)-2-[1-[(2,4-difluorophenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H26F2N4O2
6-(Cyclopropanecarbonyl)-2-[1-[(2,4-difluorophenyl)methyl]piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Propan-2-yl-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H27N5O2
6-Propan-2-yl-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylcyclohexyl)-2-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-(4-Methylcyclohexyl)-2-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-Methylcyclohexyl)-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(4-Methylcyclohexyl)-2-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(1-Ethylpyrazole-4-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N6O3
6-(1-Ethylpyrazole-4-carbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-(cyclopropanecarbonyl)-2-[1-[(2S)-2-(4-methylphenyl)propanoyl]piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2S)-2-methylbutanoyl]-2-[1-(oxan-4-yl)piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H34N4O3
6-[(2S)-2-methylbutanoyl]-2-[1-(oxan-4-yl)piperidin-4-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-butanoyl-2-[(2R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H30N4O3
6-butanoyl-2-[(2R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one