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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-2-ethyl-N-(2-methylsulfonylethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C11H20N4O2S
(6S)-2-ethyl-N-(2-methylsulfonylethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-(2-methylsulfonylethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H22N4O2S
(6R)-N-(2-methylsulfonylethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-(2-methylsulfonylethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H22N4O2S
(6S)-N-(2-methylsulfonylethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6,8-Dichloro-3-[(2-nitrophenyl)methylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine —— C13H8Cl2N4O2S
6,8-Dichloro-3-[(2-nitrophenyl)methylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine
—— 6,8-dichloro-3-[(1R)-1-phenylethyl]sulfanyl-[1,2,4]triazolo[4,3-a]pyridine —— C14H11Cl2N3S
6,8-dichloro-3-[(1R)-1-phenylethyl]sulfanyl-[1,2,4]triazolo[4,3-a]pyridine
—— 6,8-Dichloro-3-[2-(3-methylphenoxy)ethylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine —— C15H13Cl2N3OS
6,8-Dichloro-3-[2-(3-methylphenoxy)ethylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine
—— 6-Chloro-4-[[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-7-methylchromen-2-one —— C20H17ClN4O2S
6-Chloro-4-[[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-7-methylchromen-2-one
—— 6-Chloro-2-[[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]imidazo[1,2-a]pyridine —— C17H15ClN6S
6-Chloro-2-[[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]imidazo[1,2-a]pyridine
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate —— C18H15ClFNO5
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate
—— (6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate —— C20H15ClFNO5
(6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate —— C21H18FNO5
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate
—— 6-fluoro-8-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]quinoline —— C18H20FN5
6-fluoro-8-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]quinoline
—— 6-fluoro-8-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]quinoline —— C18H20FN5
6-fluoro-8-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]quinoline
—— 6-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C14H18N6S
6-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— 6-methyl-5-[(2S)-2-methylbutyl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3H-thieno[2,3-d]pyrimidin-4-one —— C20H27N5OS2
6-methyl-5-[(2S)-2-methylbutyl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C14H18N6S
6-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate —— C18H15FN2O7
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 2-[(4-fluorobenzoyl)amino]acetate
—— 6-acetyl-5-methyl-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3H-thieno[2,3-d]pyrimidin-4-one —— C17H19N5O2S2
6-acetyl-5-methyl-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-chloro-2-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine —— C16H19ClN6
6-chloro-2-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine
—— 6-chloro-2-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine —— C16H19ClN6
6-chloro-2-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine
—— [6-(dimethylamino)pyridazin-3-yl]-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C14H23N5O2
[6-(dimethylamino)pyridazin-3-yl]-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 6-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C15H19N5S
6-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— 6-methyl-5-[(2R)-2-methylbutyl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3H-thieno[2,3-d]pyrimidin-4-one —— C20H27N5OS2
6-methyl-5-[(2R)-2-methylbutyl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-chloro-7-methyl-4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)chromen-2-one —— C18H18ClN3O2S
6-chloro-7-methyl-4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)chromen-2-one
—— [6-(dimethylamino)pyridazin-3-yl]-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C14H23N5O2
[6-(dimethylamino)pyridazin-3-yl]-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— 6-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C15H19N5S
6-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— 6-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C14H17N5S
6-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— 6-fluoro-8-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline —— C18H19FN4
6-fluoro-8-[[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline
—— 6-fluoro-8-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline —— C18H19FN4
6-fluoro-8-[[(2S)-2-(pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline
—— (6S)-2-methyl-N-(6-pyrazol-1-ylpyrazin-2-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H16N8
(6S)-2-methyl-N-(6-pyrazol-1-ylpyrazin-2-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[6-(3,5-dimethylpyrazol-1-yl)pyrazin-2-yl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H20N8
(6R)-N-[6-(3,5-dimethylpyrazol-1-yl)pyrazin-2-yl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pyridine-3-carbonitrile —— C13H14N6
6-[[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]pyridine-3-carbonitrile
—— (6R)-2-methyl-N-[(2-methyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H17N5S
(6R)-2-methyl-N-[(2-methyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-2-methyl-N-[(2-methyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H17N5S
(6S)-2-methyl-N-[(2-methyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-(4-methoxypyrimidin-2-yl)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H16N6O
(6R)-N-(4-methoxypyrimidin-2-yl)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-ethyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine —— C15H18N6S
6-ethyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine
—— (6S)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H19N7
(6S)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-ethyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine —— C15H18N6S
6-ethyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]thieno[2,3-d]pyrimidin-4-amine
—— (6R)-2-methyl-N-(6-pyrazol-1-ylpyrazin-2-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H16N8
(6R)-2-methyl-N-(6-pyrazol-1-ylpyrazin-2-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-(4-methoxypyrimidin-2-yl)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H16N6O
(6S)-N-(4-methoxypyrimidin-2-yl)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[6-(3,5-dimethylpyrazol-1-yl)pyrazin-2-yl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H20N8
(6S)-N-[6-(3,5-dimethylpyrazol-1-yl)pyrazin-2-yl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H19N7
(6R)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-6-methyl-2-[[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H25N5O2S2
(6S)-6-methyl-2-[[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-6-methyl-2-[[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H25N5O2S2
(6R)-6-methyl-2-[[2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R,9S)-6-(3-ethoxy-4-methoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H26N2O3S
(6R,9S)-6-(3-ethoxy-4-methoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-6-(3-ethoxy-4-methoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H26N2O3S
(6S,9S)-6-(3-ethoxy-4-methoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-6-(3-ethoxy-4-methoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H26N2O3S
(6S,9R)-6-(3-ethoxy-4-methoxyphenyl)-9-thiophen-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-acetamido-N-[(1R)-1-(3-bromophenyl)ethyl]hexanamide —— C16H23BrN2O2
6-acetamido-N-[(1R)-1-(3-bromophenyl)ethyl]hexanamide
—— 6-(2,3-dihydroindole-1-carbonyl)-2-[(3S)-1,1-dioxothiolan-3-yl]-4,5-dihydropyridazin-3-one —— C17H19N3O4S
6-(2,3-dihydroindole-1-carbonyl)-2-[(3S)-1,1-dioxothiolan-3-yl]-4,5-dihydropyridazin-3-one
—— (6R)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C19H23N5O
(6R)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine