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—— 6-(benzotriazol-1-ylmethyl)-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]-2-methylpyrimidin-4-amine —— C22H23FN6
6-(benzotriazol-1-ylmethyl)-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]-2-methylpyrimidin-4-amine
—— 6-[2-(1H-benzimidazol-2-yl)ethyl]-2-methyl-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]pyrimidin-4-amine —— C26H30N6O
6-[2-(1H-benzimidazol-2-yl)ethyl]-2-methyl-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]pyrimidin-4-amine
—— 6-(benzotriazol-1-ylmethyl)-N-[(2R)-4-(4-fluorophenyl)butan-2-yl]-2-methylpyrimidin-4-amine —— C22H23FN6
6-(benzotriazol-1-ylmethyl)-N-[(2R)-4-(4-fluorophenyl)butan-2-yl]-2-methylpyrimidin-4-amine
—— 6-(5-ethyl-2-methylpyrazol-3-yl)-2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]pyrimidin-4-amine —— C24H31N5O
6-(5-ethyl-2-methylpyrazol-3-yl)-2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]pyrimidin-4-amine
—— 6-(1-ethylpyrazol-4-yl)-4-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine —— C19H23FN6
6-(1-ethylpyrazol-4-yl)-4-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine
—— 6-(benzotriazol-1-ylmethyl)-N-[(2S)-1-(4-chlorophenoxy)propan-2-yl]-2-methylpyrimidin-4-amine —— C21H21ClN6O
6-(benzotriazol-1-ylmethyl)-N-[(2S)-1-(4-chlorophenoxy)propan-2-yl]-2-methylpyrimidin-4-amine
—— 6-(1-ethylpyrazol-4-yl)-4-N-[(2R)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine —— C19H23FN6
6-(1-ethylpyrazol-4-yl)-4-N-[(2R)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine
—— 6-(2,4-Difluorophenyl)-2,3-dimethylimidazo[1,2-b][1,2,4]triazine —— C13H10F2N4
6-(2,4-Difluorophenyl)-2,3-dimethylimidazo[1,2-b][1,2,4]triazine
—— 6-(5-ethyl-2-methylpyrazol-3-yl)-N-[(2S)-1-(2-methoxyphenyl)propan-2-yl]-2-methylpyrimidin-4-amine —— C21H27N5O
6-(5-ethyl-2-methylpyrazol-3-yl)-N-[(2S)-1-(2-methoxyphenyl)propan-2-yl]-2-methylpyrimidin-4-amine
—— (6-aminopyridin-3-yl)-[(2R)-2-[4-[(5-fluoropyridin-2-yl)amino]-6-methylpyridin-2-yl]pyrrolidin-1-yl]methanone —— C21H21FN6O
(6-aminopyridin-3-yl)-[(2R)-2-[4-[(5-fluoropyridin-2-yl)amino]-6-methylpyridin-2-yl]pyrrolidin-1-yl]methanone
—— (6-aminopyridin-3-yl)-[(2S)-2-[4-[(5-fluoropyridin-2-yl)amino]-6-methylpyridin-2-yl]pyrrolidin-1-yl]methanone —— C21H21FN6O
(6-aminopyridin-3-yl)-[(2S)-2-[4-[(5-fluoropyridin-2-yl)amino]-6-methylpyridin-2-yl]pyrrolidin-1-yl]methanone
—— 6-methyl-2-[2-[(2S)-2-[6-methyl-4-[(4-methyl-1,3-thiazol-2-yl)amino]pyridin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C21H24N6O2S
6-methyl-2-[2-[(2S)-2-[6-methyl-4-[(4-methyl-1,3-thiazol-2-yl)amino]pyridin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— (6-methoxy-2H-chromen-3-yl)-[(2S)-2-[6-methyl-4-(pyridin-2-ylamino)pyridin-2-yl]pyrrolidin-1-yl]methanone —— C26H26N4O3
(6-methoxy-2H-chromen-3-yl)-[(2S)-2-[6-methyl-4-(pyridin-2-ylamino)pyridin-2-yl]pyrrolidin-1-yl]methanone
—— 6-methyl-2-[2-[(2R)-2-[6-methyl-4-[(4-methyl-1,3-thiazol-2-yl)amino]pyridin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C21H24N6O2S
6-methyl-2-[2-[(2R)-2-[6-methyl-4-[(4-methyl-1,3-thiazol-2-yl)amino]pyridin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— (6-methoxy-2H-chromen-3-yl)-[(2R)-2-[6-methyl-4-(pyridin-2-ylamino)pyridin-2-yl]pyrrolidin-1-yl]methanone —— C26H26N4O3
(6-methoxy-2H-chromen-3-yl)-[(2R)-2-[6-methyl-4-(pyridin-2-ylamino)pyridin-2-yl]pyrrolidin-1-yl]methanone
—— 6-(4-fluorophenyl)sulfonyl-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C20H26FN5O2S
6-(4-fluorophenyl)sulfonyl-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,3,6-trichlorobenzoate —— C17H11Cl3N2O3
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,3,6-trichlorobenzoate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(4-methylphenyl)sulfonylpropanoate —— C20H20N2O5S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(4-methylphenyl)sulfonylpropanoate
—— (6-bromo-1,3-benzodioxol-5-yl)methyl 3-(1H-indol-3-yl)propanoate —— C19H16BrNO4
(6-bromo-1,3-benzodioxol-5-yl)methyl 3-(1H-indol-3-yl)propanoate
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(1H-indol-3-yl)propanoate —— C21H19N3O3
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(1H-indol-3-yl)propanoate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[methyl-(4-methylphenyl)sulfonylamino]acetate —— C20H21N3O5S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[methyl-(4-methylphenyl)sulfonylamino]acetate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2-phenoxyacetyl)amino]acetate —— C20H19N3O5
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2-phenoxyacetyl)amino]acetate
—— 6-(4-fluorophenyl)sulfonyl-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C20H26FN5O2S
6-(4-fluorophenyl)sulfonyl-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— (6-aminopyridin-3-yl)-[(3S)-3-[5-[2-[3-(trifluoromethyl)phenoxy]ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C22H22F3N5O2
(6-aminopyridin-3-yl)-[(3S)-3-[5-[2-[3-(trifluoromethyl)phenoxy]ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— (6-aminopyridin-3-yl)-[(3R)-3-[5-[2-[3-(trifluoromethyl)phenoxy]ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C22H22F3N5O2
(6-aminopyridin-3-yl)-[(3R)-3-[5-[2-[3-(trifluoromethyl)phenoxy]ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— (6-fluoro-1H-indol-2-yl)-[(3R)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C25H25FN4O3
(6-fluoro-1H-indol-2-yl)-[(3R)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— (6-fluoro-1H-indol-2-yl)-[(3S)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone —— C25H25FN4O3
(6-fluoro-1H-indol-2-yl)-[(3S)-3-[5-[2-(4-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methanone
—— 6-[[(3S)-3-[5-[2-(4-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25ClN4O
6-[[(3S)-3-[5-[2-(4-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3S)-3-[5-[2-(3-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C26H28N4O2
6-[[(3S)-3-[5-[2-(3-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3R)-3-[5-[2-(4-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25ClN4O
6-[[(3R)-3-[5-[2-(4-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3S)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25FN4O
6-[[(3S)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3R)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25ClN4O
6-[[(3R)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3R)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25FN4O
6-[[(3R)-3-[5-[2-(4-fluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3R)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H24F2N4O
6-[[(3R)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3S)-3-[5-[2-(2-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25ClN4O
6-[[(3S)-3-[5-[2-(2-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3S)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25ClN4O
6-[[(3S)-3-[5-[2-(3-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3S)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H24F2N4O
6-[[(3S)-3-[5-[2-(3,4-difluorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3R)-3-[5-[2-(3-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C26H28N4O2
6-[[(3R)-3-[5-[2-(3-methoxyphenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— 6-[[(3R)-3-[5-[2-(2-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline —— C25H25ClN4O
6-[[(3R)-3-[5-[2-(2-chlorophenoxy)ethyl]-1H-pyrazol-3-yl]pyrrolidin-1-yl]methyl]quinoline
—— (6S)-6-[1-[(3-fluoro-4-morpholin-4-ylphenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C25H36FN3O3
(6S)-6-[1-[(3-fluoro-4-morpholin-4-ylphenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C21H29FN2O4S
(6S)-6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-benzyl-6-[1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C27H34N2O3
(6R)-1-benzyl-6-[1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-[(2R)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H28FN5O
6-[(2R)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— (6R)-6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C21H29FN2O4S
(6R)-6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6S)-1-(2-methoxyethyl)-6-[1-[[2-(2-methylpropoxy)phenyl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C25H38N2O3
(6S)-1-(2-methoxyethyl)-6-[1-[[2-(2-methylpropoxy)phenyl]methyl]piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one
—— 6-[(2S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H28FN5O
6-[(2S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— (6R)-6-[1-(5-methoxy-1-benzofuran-2-carbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C24H30N2O5
(6R)-6-[1-(5-methoxy-1-benzofuran-2-carbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one —— C24H32N4O
(6R)-6-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-1-(2-phenylethyl)-5,6-dihydro-2H-azepin-7-one
—— (6R)-6-[1-[(3-fluoro-4-morpholin-4-ylphenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one —— C25H36FN3O3
(6R)-6-[1-[(3-fluoro-4-morpholin-4-ylphenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-5,6-dihydro-2H-azepin-7-one
—— (6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one —— C24H30N4O3
(6R)-1-[(3-methoxyphenyl)methyl]-6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydro-2H-azepin-7-one