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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H22N4O4
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-(4-methylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H28N4O4
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-(4-methylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C25H20ClF3N4O3
(6R,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H26N4O3S
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C25H23ClN4O4
(6S,9R)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C28H27F3N4O3
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H28N4O3
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C25H24N4O3
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylsulfanyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C25H24N4O3S
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylsulfanyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C28H30N4O4
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C28H30N4O4S
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H25ClN4O4
(6S,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-pyridin-3-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H23N5O4
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-pyridin-3-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C23H19F3N4O4
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(trifluoromethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H26N4O3
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S)-2-[[2-(3,4-difluorophenyl)sulfanylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C18H18F2N2O2S2
(6S)-2-[[2-(3,4-difluorophenyl)sulfanylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H22N4O3
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C29H32N4O3S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O5
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-(methoxymethyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O3S
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4S
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(furan-2-yl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H24N4O4S
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(furan-2-yl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C28H30N4O4S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H28N4O4S
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C29H32N4O4
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C29H32N4O3
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O3
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H26N4O3
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylsulfanyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C28H30N4O3S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylsulfanyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H26N4O3S
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-2-propylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C29H32N4O4
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C25H24N4O4
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H24N4O3S
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C28H30N4O4
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H28N4O3
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C29H32N4O3
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C24H22N4O3
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R)-2-[[2-(3,4-difluorophenyl)sulfanylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C18H18F2N2O2S2
(6R)-2-[[2-(3,4-difluorophenyl)sulfanylacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-pyridin-3-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H23N5O4
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(furan-2-yl)-2-pyridin-3-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4
(6S,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-6-phenyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,6-dimethyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H22N4O3
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,6-dimethyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-2-benzylsulfanyl-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O3S
(6S,9R)-2-benzylsulfanyl-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-methoxyphenyl)-2-methylsulfanyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C25H23ClN4O3
(6S,9S)-6-(4-chlorophenyl)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methyl-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H28N4O4S
(6R,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-6-(4-methoxyphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-methylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C26H26N4O4
(6R,9R)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-6-(4-methylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C27H28N4O3
(6S,9S)-9-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-1H-[1,2,4]triazolo[5,1-b]quinazolin-8-one