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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(2S)-1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxypyridine-3-carbonitrile —— C17H23N3O2
6-[(2S)-1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxypyridine-3-carbonitrile
—— (6S)-2-ethyl-8-[6-propan-2-yl-2-(trifluoromethyl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H27F3N4O
(6S)-2-ethyl-8-[6-propan-2-yl-2-(trifluoromethyl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-fluorophenyl)-7-methyl-8-oxo-N-[[(3S)-oxolan-3-yl]methyl]imidazo[1,2-a]pyrazine-2-carboxamide —— C19H19FN4O3
6-(4-fluorophenyl)-7-methyl-8-oxo-N-[[(3S)-oxolan-3-yl]methyl]imidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-8-benzyl-2-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecane —— C20H28N4
(6S)-8-benzyl-2-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecane
—— (6R)-2-(pyridin-3-ylmethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H24N4O2
(6R)-2-(pyridin-3-ylmethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C18H25F3N4O
(6S)-8-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-N-[(2S)-2-hydroxybutyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C20H21ClN4O3
6-(2-chlorophenyl)-N-[(2S)-2-hydroxybutyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-2-ethyl-8-[2-(2-hydroxyphenoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O4
(6S)-2-ethyl-8-[2-(2-hydroxyphenoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-hydroxybenzoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H25N3O3
(6R)-8-(2-hydroxybenzoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2-chlorophenyl)-N-[(2R)-2-hydroxybutyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C20H21ClN4O3
6-(2-chlorophenyl)-N-[(2R)-2-hydroxybutyl]-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-8-benzyl-2-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecane —— C20H28N4
(6R)-8-benzyl-2-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecane
—— (6-methylpyridin-2-yl)-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C20H28N6O
(6-methylpyridin-2-yl)-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (6S)-2-[2-(dimethylamino)ethyl]-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N5O2
(6S)-2-[2-(dimethylamino)ethyl]-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide —— C21H25F2N3O
6-[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[1-[[(3S)-3-hydroxypiperidin-3-yl]methyl]piperidin-4-yl]-2-methyl-1H-pyrimidin-4-one —— C16H26N4O2
6-[1-[[(3S)-3-hydroxypiperidin-3-yl]methyl]piperidin-4-yl]-2-methyl-1H-pyrimidin-4-one
—— 6-[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide —— C21H25F2N3O
6-[(3S)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
—— (6R)-8-[2-(dimethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6R)-8-[2-(dimethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(dimethylamino)ethyl]-8-[2-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H31N5O3
(6S)-2-[2-(dimethylamino)ethyl]-8-[2-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(dimethylamino)ethyl]-8-[2-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H31N5O3
(6R)-2-[2-(dimethylamino)ethyl]-8-[2-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6S)-2-(3-methoxypropyl)-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]pyridine-2-carbonitrile —— C13H18N4O
6-[(3S)-3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]pyridine-2-carbonitrile
—— (6R)-2-[2-(dimethylamino)ethyl]-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H33N5O
(6R)-2-[2-(dimethylamino)ethyl]-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H33N5O
(6S)-2-[2-(dimethylamino)ethyl]-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[1-[[(3R)-3-hydroxypiperidin-3-yl]methyl]piperidin-4-yl]-2-methyl-1H-pyrimidin-4-one —— C16H26N4O2
6-[1-[[(3R)-3-hydroxypiperidin-3-yl]methyl]piperidin-4-yl]-2-methyl-1H-pyrimidin-4-one
—— (6S)-8-[2-(benzylamino)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O2
(6S)-8-[2-(benzylamino)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[2-(2-hydroxyethoxy)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O3
(6R)-8-[2-(2-hydroxyethoxy)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(dimethylamino)ethyl]-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N5O2
(6R)-2-[2-(dimethylamino)ethyl]-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile —— C19H25N7
6-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile
—— 6-[(6S)-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile —— C21H23N5O
6-[(6S)-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile
—— 6-(3-chlorophenyl)-7-(cyclopropylmethyl)-N-[(2S)-2-hydroxybutyl]-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C21H23ClN4O3
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-N-[(2S)-2-hydroxybutyl]-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-2-benzyl-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N3O
(6R)-2-benzyl-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-chloro-2-[(3,5-dimethyl-4-nitropyrazol-1-yl)methyl]-3H-quinazolin-4-one —— C14H12ClN5O3
6-chloro-2-[(3,5-dimethyl-4-nitropyrazol-1-yl)methyl]-3H-quinazolin-4-one
—— 6-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile —— C19H25N7
6-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile
—— 6-ethyl-4-[(3S)-3-(3-methoxypropyl)piperidin-1-yl]-1-methylpyrazolo[3,4-d]pyrimidine —— C17H27N5O
6-ethyl-4-[(3S)-3-(3-methoxypropyl)piperidin-1-yl]-1-methylpyrazolo[3,4-d]pyrimidine
—— (6S)-8-[2-(dimethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6S)-8-[2-(dimethylamino)acetyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-chloro-2-[[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-quinazolin-4-one —— C18H13ClN4O3S
6-chloro-2-[[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-quinazolin-4-one
—— 6-cyclopentyl-1-methyl-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C19H28N8
6-cyclopentyl-1-methyl-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— (6S)-8-[2-(2-hydroxyethoxy)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O3
(6S)-8-[2-(2-hydroxyethoxy)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-chloro-2-[[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-3H-quinazolin-4-one —— C18H15ClN6OS
6-chloro-2-[[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-3H-quinazolin-4-one
—— 6-chloro-2-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3H-quinazolin-4-one —— C15H14ClN5OS
6-chloro-2-[(5-methyl-4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3H-quinazolin-4-one
—— 6-chloro-2-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-quinazolin-4-one —— C18H13ClFN5OS
6-chloro-2-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-quinazolin-4-one
—— 6-[(6R)-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile —— C21H23N5O
6-[(6R)-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile
—— 6-chloro-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-quinazolin-4-one —— C16H11ClN4O3S
6-chloro-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-3H-quinazolin-4-one
—— (6R)-N-(1,3-benzodioxol-5-ylmethyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C19H20N2O4
(6R)-N-(1,3-benzodioxol-5-ylmethyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (6S)-6-methyl-2-oxo-N-(2,3,4-trimethoxyphenyl)-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C20H24N2O5
(6S)-6-methyl-2-oxo-N-(2,3,4-trimethoxyphenyl)-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (6R)-N-(5-chloro-2-methylphenyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C18H19ClN2O2
(6R)-N-(5-chloro-2-methylphenyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (6R)-6-methyl-2-oxo-N-propan-2-yl-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C14H20N2O2
(6R)-6-methyl-2-oxo-N-propan-2-yl-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (6S)-6-methyl-2-oxo-N-pentyl-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C16H24N2O2
(6S)-6-methyl-2-oxo-N-pentyl-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (6S)-N-(2-ethylphenyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C19H22N2O2
(6S)-N-(2-ethylphenyl)-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— (6R)-N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C21H26N2O4
(6R)-N-[2-(3,4-dimethoxyphenyl)ethyl]-6-methyl-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide