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—— (6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H30N2O4S
(6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-methyl-2-[(2R)-2-methyl-1-(1-methylpyrazol-4-yl)sulfonylpyrrolidin-2-yl]pyrimidin-4-amine —— C14H20N6O2S
6-methyl-2-[(2R)-2-methyl-1-(1-methylpyrazol-4-yl)sulfonylpyrrolidin-2-yl]pyrimidin-4-amine
—— (6-methylpyridin-2-yl)-[(2R)-2-(4-methylsulfonyl-1H-pyrazol-5-yl)pyrrolidin-1-yl]methanone —— C15H18N4O3S
(6-methylpyridin-2-yl)-[(2R)-2-(4-methylsulfonyl-1H-pyrazol-5-yl)pyrrolidin-1-yl]methanone
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (E)-3-(4-methylphenyl)prop-2-enoate —— C20H18N2O3
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (E)-3-(4-methylphenyl)prop-2-enoate
—— 6-methyl-2-[(2S)-2-methyl-1-(1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C15H17N5O2S
6-methyl-2-[(2S)-2-methyl-1-(1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— (6-methylpyridin-2-yl)-[(2S)-2-(4-methylsulfonyl-1H-pyrazol-5-yl)pyrrolidin-1-yl]methanone —— C15H18N4O3S
(6-methylpyridin-2-yl)-[(2S)-2-(4-methylsulfonyl-1H-pyrazol-5-yl)pyrrolidin-1-yl]methanone
—— 6-methyl-2-[(2R)-2-methyl-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C16H20N6O2
6-methyl-2-[(2R)-2-methyl-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2S)-2-methyl-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C16H20N6O2
6-methyl-2-[(2S)-2-methyl-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2S)-2-methyl-1-(piperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrimidin-4-one —— C16H24N4O2
6-methyl-2-[(2S)-2-methyl-1-(piperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrimidin-4-one
—— 6-[[(2S)-2-methyl-2-(4-methylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]-1H-indole —— C19H22N4
6-[[(2S)-2-methyl-2-(4-methylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]-1H-indole
—— 6-methyl-2-[(2R)-2-methyl-1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C15H17N5O2S
6-methyl-2-[(2R)-2-methyl-1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2R)-2-methyl-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C16H19N5O2S
6-methyl-2-[(2R)-2-methyl-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2S)-2-methyl-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C16H19N5O2S
6-methyl-2-[(2S)-2-methyl-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2R)-2-methyl-1-(1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C15H17N5O2S
6-methyl-2-[(2R)-2-methyl-1-(1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2R)-2-methyl-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C16H20N6O2
6-methyl-2-[(2R)-2-methyl-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2S)-2-methyl-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C16H20N6O2
6-methyl-2-[(2S)-2-methyl-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-[[(2R)-2-methyl-2-(4-methylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]-1H-indole —— C19H22N4
6-[[(2R)-2-methyl-2-(4-methylpyrimidin-2-yl)pyrrolidin-1-yl]methyl]-1H-indole
—— 6-methyl-2-[(2S)-2-methyl-1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C15H17N5O2S
6-methyl-2-[(2S)-2-methyl-1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2S)-2-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-amine —— C15H21N5S
6-methyl-2-[(2S)-2-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-amine
—— [(6S)-6-[[5-(methylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-(1-methylpyrazol-3-yl)methanone —— C16H22N6O2
[(6S)-6-[[5-(methylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-(1-methylpyrazol-3-yl)methanone
—— 6-[[(6S)-4-benzyl-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide —— C18H22N4O2
6-[[(6S)-4-benzyl-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide
—— (6-methylpyridin-2-yl)-[(6R)-6-[(6-methylpyrimidin-4-yl)methyl]-1,4-oxazepan-4-yl]methanone —— C18H22N4O2
(6-methylpyridin-2-yl)-[(6R)-6-[(6-methylpyrimidin-4-yl)methyl]-1,4-oxazepan-4-yl]methanone
—— 6-methyl-2-[(2S)-2-methyl-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C15H18N6O2
6-methyl-2-[(2S)-2-methyl-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— (6R)-4-[2-(4-fluorophenyl)ethyl]-6-(pyrazin-2-ylmethyl)-1,4-oxazepane —— C18H22FN3O
(6R)-4-[2-(4-fluorophenyl)ethyl]-6-(pyrazin-2-ylmethyl)-1,4-oxazepane
—— [(6R)-6-(pyrimidin-4-ylmethyl)-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone —— C14H16N4O2S
[(6R)-6-(pyrimidin-4-ylmethyl)-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone
—— 6-methyl-2-[(2R)-2-methyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-amine —— C14H20N6O
6-methyl-2-[(2R)-2-methyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-amine
—— 6-methyl-2-[(2R)-2-methyl-1-pyridin-2-ylpyrrolidin-2-yl]pyrimidin-4-amine —— C15H19N5
6-methyl-2-[(2R)-2-methyl-1-pyridin-2-ylpyrrolidin-2-yl]pyrimidin-4-amine
—— [(6S)-6-[[5-(methylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-phenylmethanone —— C18H22N4O2
[(6S)-6-[[5-(methylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-phenylmethanone
—— 6-methyl-2-[(2R)-2-methyl-1-(piperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrimidin-4-one —— C16H24N4O2
6-methyl-2-[(2R)-2-methyl-1-(piperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrimidin-4-one
—— 6-[[(6S)-4-[(4-methylphenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide —— C19H24N4O2
6-[[(6S)-4-[(4-methylphenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide
—— [(6S)-6-[(5-methylpyrazin-2-yl)methyl]-1,4-oxazepan-4-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C16H20N4O2S
[(6S)-6-[(5-methylpyrazin-2-yl)methyl]-1,4-oxazepan-4-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 6-methyl-2-[(2S)-2-methyl-1-methylsulfonylpyrrolidin-2-yl]pyrimidine-4-carboxamide —— C12H18N4O3S
6-methyl-2-[(2S)-2-methyl-1-methylsulfonylpyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-[[(6R)-4-[(4-methylphenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide —— C19H24N4O2
6-[[(6R)-4-[(4-methylphenyl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide
—— [(6S)-6-(pyrimidin-4-ylmethyl)-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone —— C14H16N4O2S
[(6S)-6-(pyrimidin-4-ylmethyl)-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone
—— [(6R)-6-[[5-(dimethylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-(5-methyl-1H-pyrazol-4-yl)methanone —— C17H24N6O2
[(6R)-6-[[5-(dimethylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-(5-methyl-1H-pyrazol-4-yl)methanone
—— [(6S)-6-[(6-methylpyrimidin-4-yl)methyl]-1,4-oxazepan-4-yl]-pyrimidin-5-ylmethanone —— C16H19N5O2
[(6S)-6-[(6-methylpyrimidin-4-yl)methyl]-1,4-oxazepan-4-yl]-pyrimidin-5-ylmethanone
—— [(6R)-6-[[6-(dimethylamino)pyrimidin-4-yl]methyl]-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone —— C16H21N5O2S
[(6R)-6-[[6-(dimethylamino)pyrimidin-4-yl]methyl]-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone
—— [(6R)-6-[(5-methylpyrazin-2-yl)methyl]-1,4-oxazepan-4-yl]-(1-methylpyrazol-4-yl)methanone —— C16H21N5O2
[(6R)-6-[(5-methylpyrazin-2-yl)methyl]-1,4-oxazepan-4-yl]-(1-methylpyrazol-4-yl)methanone
—— [(6R)-6-[(6-methylpyrimidin-4-yl)methyl]-1,4-oxazepan-4-yl]-pyrimidin-5-ylmethanone —— C16H19N5O2
[(6R)-6-[(6-methylpyrimidin-4-yl)methyl]-1,4-oxazepan-4-yl]-pyrimidin-5-ylmethanone
—— 6-methyl-2-[(2S)-2-methyl-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C16H20N6O2
6-methyl-2-[(2S)-2-methyl-1-(1-methylimidazole-2-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— 6-Chloro-4-[[5-(4-ethylphenyl)tetrazol-2-yl]methyl]-7-methylchromen-2-one —— C20H17ClN4O2
6-Chloro-4-[[5-(4-ethylphenyl)tetrazol-2-yl]methyl]-7-methylchromen-2-one
—— 6-methyl-2-[(2R)-2-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-amine —— C15H21N5S
6-methyl-2-[(2R)-2-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-2-yl]pyrimidin-4-amine
—— [(6R)-6-[[5-(methylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-(1-methylpyrazol-3-yl)methanone —— C16H22N6O2
[(6R)-6-[[5-(methylamino)pyrazin-2-yl]methyl]-1,4-oxazepan-4-yl]-(1-methylpyrazol-3-yl)methanone
—— 6-[[(6S)-4-[(6-methylpyridin-2-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide —— C18H23N5O2
6-[[(6S)-4-[(6-methylpyridin-2-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide
—— 6-methyl-2-[(2R)-2-methyl-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide —— C15H18N6O2
6-methyl-2-[(2R)-2-methyl-1-(1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]pyrimidine-4-carboxamide
—— [(6R)-6-(pyrazin-2-ylmethyl)-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone —— C14H16N4O2S
[(6R)-6-(pyrazin-2-ylmethyl)-1,4-oxazepan-4-yl]-(1,3-thiazol-5-yl)methanone
—— 6-[[(6R)-4-[(6-methylpyridin-2-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide —— C18H23N5O2
6-[[(6R)-4-[(6-methylpyridin-2-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrimidine-4-carboxamide
—— (6R)-4-(1H-indol-6-ylmethyl)-6-(pyrazin-2-ylmethyl)-1,4-oxazepane —— C19H22N4O
(6R)-4-(1H-indol-6-ylmethyl)-6-(pyrazin-2-ylmethyl)-1,4-oxazepane
—— [(6S)-6-[[6-(dimethylamino)pyrimidin-4-yl]methyl]-1,4-oxazepan-4-yl]-(1,3-thiazol-4-yl)methanone —— C16H21N5O2S
[(6S)-6-[[6-(dimethylamino)pyrimidin-4-yl]methyl]-1,4-oxazepan-4-yl]-(1,3-thiazol-4-yl)methanone
—— 6-methyl-2-[(2S)-2-methyl-1-(1-methylpyrazol-4-yl)sulfonylpyrrolidin-2-yl]pyrimidin-4-amine —— C14H20N6O2S
6-methyl-2-[(2S)-2-methyl-1-(1-methylpyrazol-4-yl)sulfonylpyrrolidin-2-yl]pyrimidin-4-amine