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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-8-[3-(benzotriazol-1-yl)propanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O2
(6S)-8-[3-(benzotriazol-1-yl)propanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C20H27N7
6-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[(6R)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile —— C17H22N4O
6-[(6R)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile
—— (6S)-8-(6-methylpyridazin-3-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O
(6S)-8-(6-methylpyridazin-3-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O2
(6R)-2-benzyl-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(6S)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile —— C17H22N4O
6-[(6S)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile
—— (6S)-2-ethyl-8-[2-(4-methoxyphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O3
(6S)-2-ethyl-8-[2-(4-methoxyphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-butyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O
(6R)-8-butyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O2
(6S)-2-benzyl-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6S)-2-ethyl-8-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[4-[6-(2-methoxyethylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C21H21N5O2
6-[4-[6-(2-methoxyethylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-fluoro-4-[(2R)-2-(pyrrolidine-1-carbonyl)morpholine-4-carbonyl]-1H-quinolin-2-one —— C19H20FN3O4
6-fluoro-4-[(2R)-2-(pyrrolidine-1-carbonyl)morpholine-4-carbonyl]-1H-quinolin-2-one
—— 6-fluoro-4-[(2S)-2-(pyrrolidine-1-carbonyl)morpholine-4-carbonyl]-1H-quinolin-2-one —— C19H20FN3O4
6-fluoro-4-[(2S)-2-(pyrrolidine-1-carbonyl)morpholine-4-carbonyl]-1H-quinolin-2-one
—— (6S)-2-ethyl-8-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6S)-2-ethyl-8-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[3-(benzotriazol-1-yl)propanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O2
(6R)-8-[3-(benzotriazol-1-yl)propanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6R)-2-ethyl-8-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide —— C21H34N4O2
6-[(3R)-4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
—— (6S)-8-pyridin-2-yl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H24N4O
(6S)-8-pyridin-2-yl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(3-methoxybenzoyl)amino]acetate —— C20H20ClNO6
(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)methyl 2-[(3-methoxybenzoyl)amino]acetate
—— (6R)-8-pyridin-2-yl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H24N4O
(6R)-8-pyridin-2-yl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N4O
(6R)-2-benzyl-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2,6-dimethylpyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N4O
(6R)-8-(2,6-dimethylpyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C23H28N2O2
(6S)-2-benzyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-methoxyphenyl)-7-methyl-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one —— C20H22N4O3
6-(4-methoxyphenyl)-7-methyl-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one
—— 6-(3-chlorophenyl)-8-oxo-N-[[(3R)-oxolan-3-yl]methyl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C21H21ClN4O3
6-(3-chlorophenyl)-8-oxo-N-[[(3R)-oxolan-3-yl]methyl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-2-benzyl-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N4O
(6S)-2-benzyl-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-methoxyphenyl)-7-methyl-N-[(3S)-oxan-3-yl]-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C20H22N4O4
6-(4-methoxyphenyl)-7-methyl-N-[(3S)-oxan-3-yl]-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyridine-3-carboxylic acid —— C22H29N3O4
6-[(3S)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyridine-3-carboxylic acid
—— (6R)-2-benzyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C23H28N2O2
(6R)-2-benzyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperazin-2-one —— C17H23N3O4
(6R)-6-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperazin-2-one
—— (6S)-8-(2,6-dimethylpyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N4O
(6S)-8-(2,6-dimethylpyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperazin-2-one —— C17H23N3O4
(6S)-6-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperazin-2-one
—— (6R)-8-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H32N6O2
(6R)-8-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-pent-4-enoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O2
(6S)-8-pent-4-enoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-cyclopentyl-1-methyl-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C19H24N6
6-cyclopentyl-1-methyl-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-methyl-N-[(3R)-1-(3-phenylpropyl)piperidin-3-yl]pyridazin-3-amine —— C19H26N4
6-methyl-N-[(3R)-1-(3-phenylpropyl)piperidin-3-yl]pyridazin-3-amine
—— (6S)-8-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H32N6O2
(6S)-8-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(3-chlorophenyl)-8-oxo-N-[[(3S)-oxolan-3-yl]methyl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C21H21ClN4O3
6-(3-chlorophenyl)-8-oxo-N-[[(3S)-oxolan-3-yl]methyl]-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-8-(2-propan-2-yloxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6S)-8-(2-propan-2-yloxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyridine-3-carboxylic acid —— C22H29N3O4
6-[(3R)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]piperidin-1-yl]pyridine-3-carboxylic acid
—— (6R)-2-[2-(dimethylamino)ethyl]-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O3
(6R)-2-[2-(dimethylamino)ethyl]-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23ClN4O
(6R)-8-(5-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-N-[(3S)-1-(3-phenylpropyl)piperidin-3-yl]pyridazin-3-amine —— C19H26N4
6-methyl-N-[(3S)-1-(3-phenylpropyl)piperidin-3-yl]pyridazin-3-amine
—— (6R)-8-pent-4-enoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O2
(6R)-8-pent-4-enoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [6-[(2S)-1-(dimethylamino)hex-5-en-2-yl]oxypyridin-3-yl]-pyrrolidin-1-ylmethanone —— C18H27N3O2
[6-[(2S)-1-(dimethylamino)hex-5-en-2-yl]oxypyridin-3-yl]-pyrrolidin-1-ylmethanone
—— (6R)-8-(2-propan-2-yloxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6R)-8-(2-propan-2-yloxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-cyclopentyl-1-methyl-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[3,4-d]pyrimidin-4-amine —— C19H24N6
6-cyclopentyl-1-methyl-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-(2,5-dimethylfuran-3-yl)-7-methyl-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one —— C19H22N4O3
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-[(2S)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one
—— [(6R)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]-(1,3-oxazol-4-yl)methanone —— C20H25N3O2
[(6R)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]-(1,3-oxazol-4-yl)methanone
—— 6-(4-methoxyphenyl)-7-methyl-2-[(2R)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one —— C20H22N4O3
6-(4-methoxyphenyl)-7-methyl-2-[(2R)-2-methylpyrrolidine-1-carbonyl]imidazo[1,2-a]pyrazin-8-one