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—— 6-[[(1R,3R)-3-ethoxy-2,2-diethylcyclobutyl]-methylamino]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C17H27N5O2
6-[[(1R,3R)-3-ethoxy-2,2-diethylcyclobutyl]-methylamino]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-ethyl-2-[(1S)-2-oxocyclohexyl]sulfanyl-3-(2-phenylethyl)thieno[2,3-d]pyrimidin-4-one —— C22H24N2O2S2
6-ethyl-2-[(1S)-2-oxocyclohexyl]sulfanyl-3-(2-phenylethyl)thieno[2,3-d]pyrimidin-4-one
—— 6-Ethyl-7-hydroxy-4-[[4-methyl-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one —— C20H19N3O4S
6-Ethyl-7-hydroxy-4-[[4-methyl-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one
—— 6-methyl-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-2-pyridin-2-ylpyrimidin-4-amine —— C22H22N6
6-methyl-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-2-pyridin-2-ylpyrimidin-4-amine
—— 6-[[(1S,3R)-3-ethoxy-2,2-diethylcyclobutyl]-methylamino]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C17H27N5O2
6-[[(1S,3R)-3-ethoxy-2,2-diethylcyclobutyl]-methylamino]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[(2S)-2-butyl-3-oxopiperazine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H22N4O3
6-[(2S)-2-butyl-3-oxopiperazine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-chloro-N-[(1R)-2,2-dimethylcyclopentyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide —— C17H22ClNO3
6-chloro-N-[(1R)-2,2-dimethylcyclopentyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide
—— 6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]hexan-1-ol —— C12H25NO2
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]hexan-1-ol
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]hexan-1-ol —— C12H25NO2
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]hexan-1-ol
—— 6-(cyclopropylamino)-N-[(2S,3S)-2-(1-methylpyrazol-4-yl)-6-oxopiperidin-3-yl]pyridine-3-carboxamide —— C18H22N6O2
6-(cyclopropylamino)-N-[(2S,3S)-2-(1-methylpyrazol-4-yl)-6-oxopiperidin-3-yl]pyridine-3-carboxamide
—— 6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]hexan-1-ol —— C12H25NO2
6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]hexan-1-ol
—— 6-chloro-7-ethyl-4-[[methyl-[[(3S)-oxolan-3-yl]methyl]amino]methyl]chromen-2-one —— C18H22ClNO3
6-chloro-7-ethyl-4-[[methyl-[[(3S)-oxolan-3-yl]methyl]amino]methyl]chromen-2-one
—— 6-chloro-N-[(1S)-2,2-dimethylcyclopentyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide —— C17H22ClNO3
6-chloro-N-[(1S)-2,2-dimethylcyclopentyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide
—— 6-chloro-7-ethyl-4-[[methyl-[[(3R)-oxolan-3-yl]methyl]amino]methyl]chromen-2-one —— C18H22ClNO3
6-chloro-7-ethyl-4-[[methyl-[[(3R)-oxolan-3-yl]methyl]amino]methyl]chromen-2-one
—— 6-(cyclopropylamino)-N-[(2R,3S)-2-(1-methylpyrazol-4-yl)-6-oxopiperidin-3-yl]pyridine-3-carboxamide —— C18H22N6O2
6-(cyclopropylamino)-N-[(2R,3S)-2-(1-methylpyrazol-4-yl)-6-oxopiperidin-3-yl]pyridine-3-carboxamide
—— 6-Chloro-7-methyl-4-[[4-methyl-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one —— C19H16ClN3O3S
6-Chloro-7-methyl-4-[[4-methyl-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one
—— 6-[(4S,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C21H25N5O
6-[(4S,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-chloro-N-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]pyrazin-2-amine —— C16H16ClN5O
6-chloro-N-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]pyrazin-2-amine
—— 6-N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-N,4-N-dimethylpyrimidine-4,5,6-triamine —— C18H25FN6O
6-N-[(2R)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-N,4-N-dimethylpyrimidine-4,5,6-triamine
—— 6-fluoro-4-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]quinazoline —— C17H21FN4O
6-fluoro-4-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]quinazoline
—— 6-Ethyl-4-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-7-hydroxychromen-2-one —— C21H18FN3O3S
6-Ethyl-4-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-7-hydroxychromen-2-one
—— 6-N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-N,4-N-dimethylpyrimidine-4,5,6-triamine —— C18H25FN6O
6-N-[(2S)-2-(4-fluorophenyl)-2-morpholin-4-ylethyl]-4-N,4-N-dimethylpyrimidine-4,5,6-triamine
—— 6-[(4R,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C21H25N5O
6-[(4R,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-fluoro-4-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]quinazoline —— C17H21FN4O
6-fluoro-4-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]quinazoline
—— 6-(2,3-Dihydropyrrolo[3,2-c]pyridin-1-yl)pyridine-3-carbonitrile —— C13H10N4
6-(2,3-Dihydropyrrolo[3,2-c]pyridin-1-yl)pyridine-3-carbonitrile
—— 6-[[(4R)-2-oxo-3,4-dihydro-1H-quinolin-4-yl]methylamino]pyridine-3-carbonitrile —— C16H14N4O
6-[[(4R)-2-oxo-3,4-dihydro-1H-quinolin-4-yl]methylamino]pyridine-3-carbonitrile
—— 6-chloro-N-[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]pyrazin-2-amine —— C16H16ClN5O
6-chloro-N-[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]pyrazin-2-amine
—— 6-Amino-5-[2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione —— C18H19FN6O3S
6-Amino-5-[2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione
—— 6-[(2S)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C17H18FN5O
6-[(2S)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[(2R)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C17H18FN5O
6-[(2R)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[(2R)-2-[(2-methoxyphenyl)methyl]pyrrolidin-1-yl]-7H-purine —— C17H19N5O
6-[(2R)-2-[(2-methoxyphenyl)methyl]pyrrolidin-1-yl]-7H-purine
—— 6-[(2R)-2-[(2-chlorophenyl)methyl]pyrrolidin-1-yl]pyridazine-3-carboxamide —— C16H17ClN4O
6-[(2R)-2-[(2-chlorophenyl)methyl]pyrrolidin-1-yl]pyridazine-3-carboxamide
—— 6-Chloro-4-[(4,5-dimethyl-1,2,4-triazol-3-yl)sulfanylmethyl]-7-methylchromen-2-one —— C15H14ClN3O2S
6-Chloro-4-[(4,5-dimethyl-1,2,4-triazol-3-yl)sulfanylmethyl]-7-methylchromen-2-one
—— (6S)-3-methyl-6-(trichloromethyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C12H9Cl3N4O
(6S)-3-methyl-6-(trichloromethyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— (6R)-3-methyl-6-(trichloromethyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C12H9Cl3N4O
(6R)-3-methyl-6-(trichloromethyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— 6-[2-[(1R)-2-oxocyclopentyl]ethyl]-3-prop-2-enyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C15H17N3O2S2
6-[2-[(1R)-2-oxocyclopentyl]ethyl]-3-prop-2-enyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 6-methoxy-5-[[[(2R)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]amino]methyl]pyrimidin-4-amine —— C19H27N5O2
6-methoxy-5-[[[(2R)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]amino]methyl]pyrimidin-4-amine
—— 6-chloro-2-ethyl-5-methyl-N-[(3S)-1-methylsulfonylpiperidin-3-yl]pyrimidin-4-amine —— C13H21ClN4O2S
6-chloro-2-ethyl-5-methyl-N-[(3S)-1-methylsulfonylpiperidin-3-yl]pyrimidin-4-amine
—— (6S)-2,2,6-trimethyl-4-[5-methyl-2-[(6S)-2,2,6-trimethylmorpholin-4-yl]pyrimidin-4-yl]morpholine —— C19H32N4O2
(6S)-2,2,6-trimethyl-4-[5-methyl-2-[(6S)-2,2,6-trimethylmorpholin-4-yl]pyrimidin-4-yl]morpholine
—— 6-[2-[(1S)-2-oxocyclopentyl]ethyl]-3-prop-2-enyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C15H17N3O2S2
6-[2-[(1S)-2-oxocyclopentyl]ethyl]-3-prop-2-enyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— (6R)-2,2,6-trimethyl-4-[5-methyl-2-[(6S)-2,2,6-trimethylmorpholin-4-yl]pyrimidin-4-yl]morpholine —— C19H32N4O2
(6R)-2,2,6-trimethyl-4-[5-methyl-2-[(6S)-2,2,6-trimethylmorpholin-4-yl]pyrimidin-4-yl]morpholine
—— 6-methoxy-5-[[[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]amino]methyl]pyrimidin-4-amine —— C19H27N5O2
6-methoxy-5-[[[(2S)-2-(4-methoxyphenyl)-2-pyrrolidin-1-ylethyl]amino]methyl]pyrimidin-4-amine
—— 6-chloro-2-ethyl-5-methyl-N-[(3R)-1-methylsulfonylpiperidin-3-yl]pyrimidin-4-amine —— C13H21ClN4O2S
6-chloro-2-ethyl-5-methyl-N-[(3R)-1-methylsulfonylpiperidin-3-yl]pyrimidin-4-amine
—— 6-methyl-3-[(2Z)-2-[1-(4-methylsulfonylphenyl)ethylidene]hydrazinyl]-4H-1,2,4-triazin-5-one —— C13H15N5O3S
6-methyl-3-[(2Z)-2-[1-(4-methylsulfonylphenyl)ethylidene]hydrazinyl]-4H-1,2,4-triazin-5-one
—— 6-fluoro-N-[[3-[(1R)-1-methoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylquinazolin-4-amine —— C15H16FN5O2
6-fluoro-N-[[3-[(1R)-1-methoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylquinazolin-4-amine
—— 6-fluoro-N-[[3-[(1S)-1-methoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylquinazolin-4-amine —— C15H16FN5O2
6-fluoro-N-[[3-[(1S)-1-methoxyethyl]-1,2,4-oxadiazol-5-yl]methyl]-N-methylquinazolin-4-amine
—— 6-methyl-3-[(2Z)-2-[(5-phenylthiophen-2-yl)methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one —— C15H13N5OS
6-methyl-3-[(2Z)-2-[(5-phenylthiophen-2-yl)methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one
—— 6-(4-fluorophenyl)-2-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]pyridazin-3-one —— C17H16FN3O2S
6-(4-fluorophenyl)-2-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]pyridazin-3-one
—— 6-chloro-N-[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]pyrazin-2-amine —— C16H14ClN5
6-chloro-N-[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]pyrazin-2-amine
—— 6-ethylsulfanyl-N-[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]pyrazin-2-amine —— C18H19N5S
6-ethylsulfanyl-N-[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]pyrazin-2-amine