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—— 6-chloro-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1,4-benzodioxine-7-sulfonamide —— C14H15ClN2O5S
6-chloro-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1,4-benzodioxine-7-sulfonamide
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3R)-3-acetamido-3-phenylpropanoate —— C21H21N3O4
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3R)-3-acetamido-3-phenylpropanoate
—— 6-(2-Hydroxy-4-phenylmethoxyphenyl)-9-methyl-2-(4-morpholin-4-ylphenyl)-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone —— C40H36N2O7
6-(2-Hydroxy-4-phenylmethoxyphenyl)-9-methyl-2-(4-morpholin-4-ylphenyl)-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone
—— (6S)-1-[2-(4-ethoxyphenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C28H30N2O3
(6S)-1-[2-(4-ethoxyphenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-butoxy-3-methoxybenzoate —— C22H24N2O5
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-butoxy-3-methoxybenzoate
—— (6R)-1-[2-(4-ethoxyphenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C28H30N2O3
(6R)-1-[2-(4-ethoxyphenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(4-hydroxy-3-methoxyphenyl)-2-(4-iodophenyl)-6a,9-diphenyl-4,6,10a,11,11a,11b-hexahydro-3aH-naphtho[6,7-e]isoindole-1,3,7,10-tetrone —— C41H32INO6
6-(4-hydroxy-3-methoxyphenyl)-2-(4-iodophenyl)-6a,9-diphenyl-4,6,10a,11,11a,11b-hexahydro-3aH-naphtho[6,7-e]isoindole-1,3,7,10-tetrone
—— (6-Bromo-1,3-benzodioxol-5-yl)methyl 4-(4-methylphenyl)-4-oxobutanoate —— C19H17BrO5
(6-Bromo-1,3-benzodioxol-5-yl)methyl 4-(4-methylphenyl)-4-oxobutanoate
—— 6-[(E)-hydroxyiminomethyl]-8-methyl-3-phenylpteridine-2,4-dione —— C14H11N5O3
6-[(E)-hydroxyiminomethyl]-8-methyl-3-phenylpteridine-2,4-dione
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-hexoxy-3-methoxybenzoate —— C24H28N2O5
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-hexoxy-3-methoxybenzoate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(4-chlorophenyl)sulfanylbutanoate —— C20H19ClN2O3S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(4-chlorophenyl)sulfanylbutanoate
—— 6-[2-(Cyclohexen-1-yl)ethyl]-3-(4-fluorophenyl)-[1,2]thiazolo[4,5-d]pyrimidin-7-one —— C19H18FN3OS
6-[2-(Cyclohexen-1-yl)ethyl]-3-(4-fluorophenyl)-[1,2]thiazolo[4,5-d]pyrimidin-7-one
—— 6-[(6-Methyl-4-oxochromen-3-yl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O3
6-[(6-Methyl-4-oxochromen-3-yl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H37N5O2
6-[[2,5-dimethyl-1-[[(2R)-oxolan-2-yl]methyl]pyrrol-3-yl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H37N5O2
6-[[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-Methylphenyl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H24N4O
6-[(3-Methylphenyl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,4-Dimethoxyphenyl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O3
6-[(3,4-Dimethoxyphenyl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-hydroxy-4-methoxyphenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H28N4O3
6-[(3-hydroxy-4-methoxyphenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(1-methylimidazol-2-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H26N6O
6-[(1-methylimidazol-2-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H30N4O3
6-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(1-methylimidazol-2-yl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H26N6O
6-[(1-methylimidazol-2-yl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(4-Methylphenyl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H24N4O
6-[(4-Methylphenyl)methyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H30N4O3
6-[[3-(hydroxymethyl)-4-methoxyphenyl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2H-chromen-3-ylmethyl)-2-(4-methylpiperidin-1-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H28N4O2
6-(2H-chromen-3-ylmethyl)-2-(4-methylpiperidin-1-yl)-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-hydroxy-4-methoxyphenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H28N4O3
6-[(3-hydroxy-4-methoxyphenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(4-methylphenyl)-4-oxobutanoate —— C21H20N2O4
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(4-methylphenyl)-4-oxobutanoate
—— 6-Cyclopropyl-2-[1-[1-(4-methoxyphenyl)cyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one —— C26H33N3O3
6-Cyclopropyl-2-[1-[1-(4-methoxyphenyl)cyclohexanecarbonyl]piperidin-4-yl]pyridazin-3-one
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(1-benzyltriazol-4-yl)prop-2-enoate —— C21H18ClN3O4
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(1-benzyltriazol-4-yl)prop-2-enoate
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(4-ethoxyphenoxy)butanoate —— C22H24N2O5
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(4-ethoxyphenoxy)butanoate
—— 6-tert-butyl-3-[[(4-methyl-2-oxo-1H-pyridin-3-yl)amino]methyl]-1H-quinolin-2-one —— C20H23N3O2
6-tert-butyl-3-[[(4-methyl-2-oxo-1H-pyridin-3-yl)amino]methyl]-1H-quinolin-2-one
—— 6-tert-butyl-3-[[(3-methoxypyridin-2-yl)amino]methyl]-1H-quinolin-2-one —— C20H23N3O2
6-tert-butyl-3-[[(3-methoxypyridin-2-yl)amino]methyl]-1H-quinolin-2-one
—— (6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H30N2O4S
(6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O2
(6R)-1-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1,3-benzothiazole-6-carboxylate —— C18H13N3O3S
(6-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1,3-benzothiazole-6-carboxylate
—— (6R)-1-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O2
(6R)-1-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1S,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one —— C24H28N2O3
(6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1S,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one
—— (6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H29FN2O4S
(6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-methyl-1-[(2S)-2-phenylpropyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H31N3O
(6R)-4-methyl-1-[(2S)-2-phenylpropyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (E)-3-(1-benzyltriazol-4-yl)prop-2-enoate —— C22H19N5O3
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (E)-3-(1-benzyltriazol-4-yl)prop-2-enoate
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(1S,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one —— C24H28N2O3
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(1S,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one
—— (6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H30N2O4S
(6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H30N2O4S
(6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(1R,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one —— C24H28N2O3
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-[(1R,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one
—— (6R)-1-[(2S)-2-phenylpropyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O
(6R)-1-[(2S)-2-phenylpropyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1,4-diazepan-5-one —— C22H26F2N2O3S
(6R)-1-[(2R)-butan-2-yl]sulfonyl-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1R,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one —— C24H28N2O3
(6R)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1-[(1R,2R)-2-methylcyclopropanecarbonyl]-1,4-diazepan-5-one
—— (6R)-4-methyl-1-[(2R)-2-phenylpropyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H31N3O
(6R)-4-methyl-1-[(2R)-2-phenylpropyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2R)-2-phenylpropyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O
(6R)-1-[(2R)-2-phenylpropyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1,4-diazepan-5-one —— C22H26F2N2O3S
(6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(3,4-difluorophenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H29FN2O4S
(6R)-1-[(2S)-butan-2-yl]sulfonyl-6-[[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one