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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-6-[4-(4-methylphenyl)sulfanylpiperidine-1-carbonyl]piperazin-2-one —— C17H23N3O2S
(6R)-6-[4-(4-methylphenyl)sulfanylpiperidine-1-carbonyl]piperazin-2-one
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl 2-(4-methylphenyl)acetate —— C18H17NO6
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl 2-(4-methylphenyl)acetate
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H29N5O2
(6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H29N5O2
(6R)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(pyridine-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H24N4O2
(6R)-8-(pyridine-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carboxylic acid —— C17H24N6O2
6-[(3R)-3-[5-[(dimethylamino)methyl]-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carboxylic acid
—— (6R)-2-ethyl-8-(2-ethylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N4O2
(6R)-2-ethyl-8-(2-ethylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H31N3O2
(6R)-2-benzyl-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2S)-2-hydroxybutyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C18H22N4O4
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-2-hydroxybutyl]-7-methyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H25N5O2
(6S)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(pyridin-3-ylmethyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H24N4O2
(6S)-2-(pyridin-3-ylmethyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(3-fluoropyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H23FN4O
(6S)-8-(3-fluoropyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[4-(4-methylphenyl)sulfanylpiperidine-1-carbonyl]piperazin-2-one —— C17H23N3O2S
(6S)-6-[4-(4-methylphenyl)sulfanylpiperidine-1-carbonyl]piperazin-2-one
—— (6S)-2-ethyl-8-(2-ethylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N4O2
(6S)-2-ethyl-8-(2-ethylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methoxypropyl)-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C17H28N4O2S
(6R)-2-(3-methoxypropyl)-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C17H28N4O2S
(6S)-2-(3-methoxypropyl)-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(6R)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C22H25N5O
6-methyl-2-[(6R)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— (6S)-8-[(E)-pent-3-enoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O2
(6S)-8-[(E)-pent-3-enoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-cyclopentyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine —— C18H24N6O
6-cyclopentyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methylpyrazolo[3,4-d]pyrimidin-4-amine
—— (6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H29N5OS
(6S)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(E)-pent-3-enoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N3O2
(6R)-8-[(E)-pent-3-enoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H29N5OS
(6R)-2-[2-(dimethylamino)ethyl]-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(8-hydroxyquinoline-7-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25N3O3
(6S)-2-ethyl-8-(8-hydroxyquinoline-7-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6-propan-2-ylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H30N4O
(6S)-8-(6-propan-2-ylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-chlorophenyl)-7-[[(3R)-3-methoxypiperidin-1-yl]methyl]-[1,3]dioxolo[4,5-g]quinoline —— C23H23ClN2O3
6-(4-chlorophenyl)-7-[[(3R)-3-methoxypiperidin-1-yl]methyl]-[1,3]dioxolo[4,5-g]quinoline
—— (6R)-2-ethyl-8-(8-hydroxyquinoline-7-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25N3O3
(6R)-2-ethyl-8-(8-hydroxyquinoline-7-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4-chlorophenyl)-7-[[(3S)-3-methoxypiperidin-1-yl]methyl]-[1,3]dioxolo[4,5-g]quinoline —— C23H23ClN2O3
6-(4-chlorophenyl)-7-[[(3S)-3-methoxypiperidin-1-yl]methyl]-[1,3]dioxolo[4,5-g]quinoline
—— 6-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C18H18FN5O2
6-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— 6-methyl-2-[(6S)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C22H25N5O
6-methyl-2-[(6S)-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— 6-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C18H18FN5O2
6-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— (6R)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H25N5O2
(6R)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6S)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6R)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(4,6-dimethylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O2
(6R)-8-(4,6-dimethylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-propan-2-ylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H30N4O
(6R)-8-(6-propan-2-ylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-4-[1-(2-phenylethyl)piperidin-4-yl]-1,4-oxazepan-6-yl]methanol —— C19H30N2O2
[(6S)-4-[1-(2-phenylethyl)piperidin-4-yl]-1,4-oxazepan-6-yl]methanol
—— 6-(3-chlorophenyl)-2-[(2S)-2-methylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C21H21ClN4O2
6-(3-chlorophenyl)-2-[(2S)-2-methylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— 6-(3-chlorophenyl)-2-[(2R)-2-methylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C21H21ClN4O2
6-(3-chlorophenyl)-2-[(2R)-2-methylpyrrolidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— [(6R)-4-[1-(2-phenylethyl)piperidin-4-yl]-1,4-oxazepan-6-yl]methanol —— C19H30N2O2
[(6R)-4-[1-(2-phenylethyl)piperidin-4-yl]-1,4-oxazepan-6-yl]methanol
—— (6S)-8-(3-methylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O
(6S)-8-(3-methylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N4O
(6R)-2-ethyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-methylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O
(6R)-8-(3-methylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[4-methyl-5-(morpholin-4-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C19H25N7O
6-[(3R)-3-[4-methyl-5-(morpholin-4-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— (6S)-2-(pyridin-3-ylmethyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H22N6O2
(6S)-2-(pyridin-3-ylmethyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[3-(2-methylimidazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O
(6R)-2-ethyl-8-[3-(2-methylimidazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile —— C20H27N7
6-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile
—— (6R)-2-(pyridin-3-ylmethyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H22N6O2
(6R)-2-(pyridin-3-ylmethyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(6-chloropyridin-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25ClN4O
(6S)-8-[(6-chloropyridin-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(6-chloropyridin-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25ClN4O
(6R)-8-[(6-chloropyridin-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-pentanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O2
(6S)-8-pentanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one