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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-8-hexanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6R)-8-hexanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-cyclopropylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O
(6R)-8-(6-cyclopropylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6S)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-benzyl-2-[(5-methyl-1H-imidazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecane —— C21H30N4
(6S)-8-benzyl-2-[(5-methyl-1H-imidazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecane
—— [(6S)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]-(2,5-dimethyl-1,3-oxazol-4-yl)methanone —— C22H29N3O2
[(6S)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]-(2,5-dimethyl-1,3-oxazol-4-yl)methanone
—— 6-[(2S)-1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxypyridine-3-carbonitrile —— C18H24N4O2
6-[(2S)-1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxypyridine-3-carbonitrile
—— (6S)-8-pyridin-2-yl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H24N4O
(6S)-8-pyridin-2-yl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6-cyclopropylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O
(6S)-8-(6-cyclopropylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-(2-pyrrolidin-1-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H33N3O
(6S)-2-benzyl-8-(2-pyrrolidin-1-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(dimethylamino)ethyl]-8-[4-(tetrazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H31N7O2
(6R)-2-[2-(dimethylamino)ethyl]-8-[4-(tetrazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O3
(6S)-2-ethyl-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6S)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-benzyl-8-(2-pyrrolidin-1-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H33N3O
(6R)-2-benzyl-8-(2-pyrrolidin-1-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H29N3O
(6S)-2-benzyl-8-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-1-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]piperidin-3-yl]-1H-pyrimidin-4-one —— C20H21ClN4O2
6-[(3S)-1-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]piperidin-3-yl]-1H-pyrimidin-4-one
—— 6-[(3R)-1-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]piperidin-3-yl]-1H-pyrimidin-4-one —— C20H21ClN4O2
6-[(3R)-1-[[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]piperidin-3-yl]-1H-pyrimidin-4-one
—— (6R)-8-pyridin-2-yl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H24N4O
(6R)-8-pyridin-2-yl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6R)-8-(1-aminocyclopropanecarbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(dimethylamino)ethyl]-8-[4-(tetrazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H31N7O2
(6S)-2-[2-(dimethylamino)ethyl]-8-[4-(tetrazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-hydroxy-4-methyl-5-[[(5R)-5-methyl-1,3-oxazolidin-3-ium-3-yl]methyl]-2-oxo-1-prop-2-enylpyridine-3-carbonitrile —— C15H20N3O3+
6-hydroxy-4-methyl-5-[[(5R)-5-methyl-1,3-oxazolidin-3-ium-3-yl]methyl]-2-oxo-1-prop-2-enylpyridine-3-carbonitrile
—— 6-hydroxy-4-methyl-5-[[(5S)-5-methyl-1,3-oxazolidin-3-ium-3-yl]methyl]-2-oxo-1-prop-2-enylpyridine-3-carbonitrile —— C15H20N3O3+
6-hydroxy-4-methyl-5-[[(5S)-5-methyl-1,3-oxazolidin-3-ium-3-yl]methyl]-2-oxo-1-prop-2-enylpyridine-3-carbonitrile
—— 6-[(3S)-3-[2-(2,5-dihydropyrrol-1-yl)-2-oxoethyl]morpholine-4-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one —— C18H20N4O4S
6-[(3S)-3-[2-(2,5-dihydropyrrol-1-yl)-2-oxoethyl]morpholine-4-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one
—— (6R)-2-ethyl-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O3
(6R)-2-ethyl-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-chloro-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]pyridine-3-carboxamide —— C14H15ClN2OS
6-chloro-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]pyridine-3-carboxamide
—— 6-(2-chlorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C18H19ClN4O3
6-(2-chlorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2-chlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide —— C18H19ClN4O3
6-(2-chlorophenyl)-N-[(2R)-1-hydroxypropan-2-yl]-N,7-dimethyl-8-oxoimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2,5-dimethylfuran-3-yl)-2-[(3R)-3-methoxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H26N4O4
6-(2,5-dimethylfuran-3-yl)-2-[(3R)-3-methoxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— 6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[[(3R)-oxolan-3-yl]methyl]imidazo[1,2-a]pyrazine-2-carboxamide —— C19H22N4O4
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[[(3R)-oxolan-3-yl]methyl]imidazo[1,2-a]pyrazine-2-carboxamide
—— (6S)-2-ethyl-8-(7H-purin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C16H22N6O
(6S)-2-ethyl-8-(7H-purin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N4O3
(6R)-2-ethyl-8-[2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-4-[4-[(1S)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-1H-quinolin-2-one —— C22H29N3O3
6-methyl-4-[4-[(1S)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-1H-quinolin-2-one
—— 6-(2,5-dimethylfuran-3-yl)-2-[(3S)-3-methoxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one —— C22H26N4O4
6-(2,5-dimethylfuran-3-yl)-2-[(3S)-3-methoxypiperidine-1-carbonyl]-7-prop-2-enylimidazo[1,2-a]pyrazin-8-one
—— 6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-[(3R)-2-oxopiperidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide —— C20H20FN5O4
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-[(3R)-2-oxopiperidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2-chlorophenyl)-N-[(2S)-4-hydroxybutan-2-yl]-N-methyl-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide —— C21H23ClN4O3
6-(2-chlorophenyl)-N-[(2S)-4-hydroxybutan-2-yl]-N-methyl-8-oxo-7-prop-2-enylimidazo[1,2-a]pyrazine-2-carboxamide
—— 6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-[(3S)-2-oxopiperidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide —— C20H20FN5O4
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-[(3S)-2-oxopiperidin-3-yl]imidazo[1,2-a]pyrazine-2-carboxamide
—— (6R)-2-ethyl-8-(7H-purin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C16H22N6O
(6R)-2-ethyl-8-(7H-purin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-[2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N4O3
(6S)-2-ethyl-8-[2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-4-[4-[(1R)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-1H-quinolin-2-one —— C22H29N3O3
6-methyl-4-[4-[(1R)-1-morpholin-4-ylethyl]piperidine-1-carbonyl]-1H-quinolin-2-one
—— (6R)-8-(5-acetylpyridin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6R)-8-(5-acetylpyridin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[(3-methoxy-4-phenylmethoxyphenyl)methyl]-1,4-oxazepan-6-ol —— C20H25NO4
(6S)-4-[(3-methoxy-4-phenylmethoxyphenyl)methyl]-1,4-oxazepan-6-ol
—— (6R)-8-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O4
(6R)-8-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-amino-2-methylpropanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6S)-8-(2-amino-2-methylpropanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-ethyl-1-methyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]pyrazolo[3,4-d]pyrimidin-4-amine —— C18H28N6O
6-ethyl-1-methyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]pyrazolo[3,4-d]pyrimidin-4-amine
—— 6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[[(3S)-oxolan-3-yl]methyl]imidazo[1,2-a]pyrazine-2-carboxamide —— C19H22N4O4
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[[(3S)-oxolan-3-yl]methyl]imidazo[1,2-a]pyrazine-2-carboxamide
—— 6-[[(4-Tert-butylphenyl)methyl-methylamino]methyl]-2,3-dihydro-[1,4]dioxino[2,3-f]indole-7,8-dione —— C23H26N2O4
6-[[(4-Tert-butylphenyl)methyl-methylamino]methyl]-2,3-dihydro-[1,4]dioxino[2,3-f]indole-7,8-dione
—— (6R)-2-(pyridin-2-ylmethyl)-8-[3-(1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N6O2
(6R)-2-(pyridin-2-ylmethyl)-8-[3-(1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-amino-2-methylpropanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6R)-8-(2-amino-2-methylpropanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-benzyl-8-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6S)-2-benzyl-8-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2,2-dimethylpropanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O2
(6R)-8-(2,2-dimethylpropanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O4
(6S)-8-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one