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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-N-[2-(dimethylamino)ethyl]-N-[(3-methylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-6-carboxamide —— C20H28N4O
(6R)-N-[2-(dimethylamino)ethyl]-N-[(3-methylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-6-carboxamide
—— 6-[(2R)-2-hydroxy-3-pyrazol-1-ylpropyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C16H23N5O2
6-[(2R)-2-hydroxy-3-pyrazol-1-ylpropyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— (6S)-N-[2-(dimethylamino)ethyl]-N-[(3-methylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-6-carboxamide —— C20H28N4O
(6S)-N-[2-(dimethylamino)ethyl]-N-[(3-methylphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazole-6-carboxamide
—— 6-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C15H21N5O2
6-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C15H24N4O3
6-[(2R)-2-hydroxy-3-morpholin-4-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[2-[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-2-oxoethyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H26N4O3
6-[2-[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-2-oxoethyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(2S)-2-hydroxy-3-morpholin-4-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C15H24N4O3
6-[(2S)-2-hydroxy-3-morpholin-4-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(3R)-2-oxooxolan-3-yl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C14H19N3O3
6-[(3R)-2-oxooxolan-3-yl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-N-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]pyrazin-2-amine —— C15H14ClN5
6-chloro-N-[(1R)-1-(3-imidazol-1-ylphenyl)ethyl]pyrazin-2-amine
—— 6-[(2S)-1-(4-acetylpiperazin-1-yl)-1-oxopropan-2-yl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C17H25N5O3
6-[(2S)-1-(4-acetylpiperazin-1-yl)-1-oxopropan-2-yl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(3S)-2-oxooxolan-3-yl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C14H19N3O3
6-[(3S)-2-oxooxolan-3-yl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[2-[(S)-phenylsulfinyl]ethyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H23N3O2S
6-[2-[(S)-phenylsulfinyl]ethyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(2R)-2-hydroxy-3-pyrazol-1-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C14H19N5O2
6-[(2R)-2-hydroxy-3-pyrazol-1-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-4-N-[(3S)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrimidine-2,4-diamine —— C13H18ClN7
6-chloro-4-N-[(3S)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrimidine-2,4-diamine
—— 6-(5-methylthiophen-2-yl)-2-[2-[[(2R)-oxolan-2-yl]methoxy]ethyl]pyridazin-3-one —— C16H20N2O3S
6-(5-methylthiophen-2-yl)-2-[2-[[(2R)-oxolan-2-yl]methoxy]ethyl]pyridazin-3-one
—— [(6R)-3-pyridin-4-yl-4,5,6,7-tetrahydro-1H-indazol-6-yl]methanamine —— C13H16N4
[(6R)-3-pyridin-4-yl-4,5,6,7-tetrahydro-1H-indazol-6-yl]methanamine
—— 6-chloro-N-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]pyrazin-2-amine —— C15H14ClN5
6-chloro-N-[(1S)-1-(3-imidazol-1-ylphenyl)ethyl]pyrazin-2-amine
—— 6-[(2S)-2-hydroxy-3-pyrazol-1-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C14H19N5O2
6-[(2S)-2-hydroxy-3-pyrazol-1-ylpropyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— [(6S)-3-pyridin-4-yl-4,5,6,7-tetrahydro-1H-indazol-6-yl]methanamine —— C13H16N4
[(6S)-3-pyridin-4-yl-4,5,6,7-tetrahydro-1H-indazol-6-yl]methanamine
—— 6-[2-[(S)-phenylsulfinyl]ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H23N3O2S
6-[2-[(S)-phenylsulfinyl]ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-N-[(3S)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrazin-2-amine —— C13H17ClN6
6-chloro-N-[(3S)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrazin-2-amine
—— 6-[2-[(R)-phenylsulfinyl]ethyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H23N3O2S
6-[2-[(R)-phenylsulfinyl]ethyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(3R)-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C14H19N3O3
6-[(3R)-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[methyl-[(1R,2R)-2-(4-methylphenyl)cyclopentyl]amino]pyridine-3-carbonitrile —— C19H21N3
6-[methyl-[(1R,2R)-2-(4-methylphenyl)cyclopentyl]amino]pyridine-3-carbonitrile
—— 6-[methyl-[(1S,2R)-2-(4-methylphenyl)cyclopentyl]amino]pyridine-3-carbonitrile —— C19H21N3
6-[methyl-[(1S,2R)-2-(4-methylphenyl)cyclopentyl]amino]pyridine-3-carbonitrile
—— 6-[(2R)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H25N3O4
6-[(2R)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[[(2S)-oxan-2-yl]methyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C16H25N3O2
6-[[(2S)-oxan-2-yl]methyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-4-[[(2R)-2-hydroxy-3-methoxypropyl]amino]quinoline-3-carbonitrile —— C14H14ClN3O2
6-chloro-4-[[(2R)-2-hydroxy-3-methoxypropyl]amino]quinoline-3-carbonitrile
—— 6-[[(2R,3S)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]pyridine-3-carbonitrile —— C17H20N4S
6-[[(2R,3S)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-ethyl-N-[2-methyl-2-(1-oxo-1,4-thiazinan-4-yl)propyl]pyrimidin-4-amine —— C14H24N4OS
6-ethyl-N-[2-methyl-2-(1-oxo-1,4-thiazinan-4-yl)propyl]pyrimidin-4-amine
—— 6-[[(2R)-oxan-2-yl]methyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C16H25N3O2
6-[[(2R)-oxan-2-yl]methyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[2-[(R)-phenylsulfinyl]ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H23N3O2S
6-[2-[(R)-phenylsulfinyl]ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-N-[(3R)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrazin-2-amine —— C13H17ClN6
6-chloro-N-[(3R)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrazin-2-amine
—— 6-[(3S,5S)-5-methyl-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C15H21N3O3
6-[(3S,5S)-5-methyl-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-4-[[(2S)-2-hydroxy-3-methoxypropyl]amino]quinoline-3-carbonitrile —— C14H14ClN3O2
6-chloro-4-[[(2S)-2-hydroxy-3-methoxypropyl]amino]quinoline-3-carbonitrile
—— 6-[methyl-[(1R,2S)-2-(4-methylphenyl)cyclopentyl]amino]pyridine-3-carbonitrile —— C19H21N3
6-[methyl-[(1R,2S)-2-(4-methylphenyl)cyclopentyl]amino]pyridine-3-carbonitrile
—— 6-[(2R)-1-(4-acetylpiperazin-1-yl)-1-oxopropan-2-yl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C17H25N5O3
6-[(2R)-1-(4-acetylpiperazin-1-yl)-1-oxopropan-2-yl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C15H21N5O2
6-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[(3R,5S)-5-methyl-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C15H21N3O3
6-[(3R,5S)-5-methyl-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-[[(2R,3R)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]pyridine-3-carbonitrile —— C17H20N4S
6-[[(2R,3R)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-[2-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-2-oxoethyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H26N4O3
6-[2-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-2-oxoethyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]pyrazin-2-amine —— C9H14ClN3O2S
6-chloro-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]pyrazin-2-amine
—— 6-chloro-4-[[(2R)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]quinoline-3-carbonitrile —— C15H16ClN3OS
6-chloro-4-[[(2R)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]quinoline-3-carbonitrile
—— 6-[[(2S)-3-imidazol-1-yl-2-methylpropyl]amino]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C18H19N7O
6-[[(2S)-3-imidazol-1-yl-2-methylpropyl]amino]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[(3S)-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C14H19N3O3
6-[(3S)-2-oxooxolan-3-yl]-2-propyl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-4-[[(2S)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]quinoline-3-carbonitrile —— C15H16ClN3OS
6-chloro-4-[[(2S)-4-hydroxy-1-methylsulfanylbutan-2-yl]amino]quinoline-3-carbonitrile
—— 6-[(2S)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one —— C18H25N3O4
6-[(2S)-3-(furan-2-ylmethoxy)-2-hydroxypropyl]-2-propan-2-yl-7,8-dihydro-5H-pyrido[4,3-c]pyridazin-3-one
—— 6-chloro-4-N-[(3R)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrimidine-2,4-diamine —— C13H18ClN7
6-chloro-4-N-[(3R)-1-(1-methylpyrazol-4-yl)piperidin-3-yl]pyrimidine-2,4-diamine
—— 6,7-difluoro-N-[2-[[(2S)-oxolan-2-yl]methoxy]ethyl]quinazolin-4-amine —— C15H17F2N3O2
6,7-difluoro-N-[2-[[(2S)-oxolan-2-yl]methoxy]ethyl]quinazolin-4-amine
—— 6,7-difluoro-N-[2-[[(2R)-oxolan-2-yl]methoxy]ethyl]quinazolin-4-amine —— C15H17F2N3O2
6,7-difluoro-N-[2-[[(2R)-oxolan-2-yl]methoxy]ethyl]quinazolin-4-amine