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—— (6S)-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H39N7O3
(6S)-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cycloheptyl-2-N-[2-(2-methoxyphenyl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O4
(6R)-6-N-cycloheptyl-2-N-[2-(2-methoxyphenyl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5,6-dimethyl-6-N-(3-methylbutyl)-2-N-[(5-methylfuran-2-yl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C21H29N5O4
(6S)-5,6-dimethyl-6-N-(3-methylbutyl)-2-N-[(5-methylfuran-2-yl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— 6-(2-Hydroxy-4-phenylmethoxyphenyl)-8-methyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone —— C30H25NO6
6-(2-Hydroxy-4-phenylmethoxyphenyl)-8-methyl-3a,4,6,11,11a,11b-hexahydronaphtho[6,7-e]isoindole-1,3,7,10-tetrone
—— 6a-(4-chlorophenyl)-8-(4-fluoroanilino)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C39H28ClF4N3O6
6a-(4-chlorophenyl)-8-(4-fluoroanilino)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6S)-6-N-cyclopentyl-5,6-dimethyl-4-oxo-2-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H31N5O3
(6S)-6-N-cyclopentyl-5,6-dimethyl-4-oxo-2-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-2-N-(furan-2-ylmethyl)-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C20H27N5O4
(6S)-2-N-(furan-2-ylmethyl)-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— 6a-(4-chlorophenyl)-6-(3-ethoxy-2-hydroxyphenyl)-8-(4-fluoroanilino)-2-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C35H31ClFN3O6
6a-(4-chlorophenyl)-6-(3-ethoxy-2-hydroxyphenyl)-8-(4-fluoroanilino)-2-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6R)-2-N-[2-(furan-2-yl)ethyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C21H29N5O4
(6R)-2-N-[2-(furan-2-yl)ethyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— 6-[(2S)-2-methyl-3-oxo-3-piperidin-1-ylpropyl]sulfonyl-4H-1,4-benzothiazin-3-one —— C17H22N2O4S2
6-[(2S)-2-methyl-3-oxo-3-piperidin-1-ylpropyl]sulfonyl-4H-1,4-benzothiazin-3-one
—— 6a,9a-Dichloro-6-(4-hydroxy-3-methoxyphenyl)-8-methyl-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C28H23Cl2N3O8
6a,9a-Dichloro-6-(4-hydroxy-3-methoxyphenyl)-8-methyl-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(2-Hydroxy-4-phenylmethoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindole-2-carboxamide —— C31H26N2O7
6-(2-Hydroxy-4-phenylmethoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindole-2-carboxamide
—— (6R)-6-N-cyclopentyl-6-methyl-2-N-(2-morpholin-4-ylethyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H36N6O4
(6R)-6-N-cyclopentyl-6-methyl-2-N-(2-morpholin-4-ylethyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— 6a,9a-Dichloro-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-[5-(hydroxymethyl)furan-2-yl]-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C27H22Cl3F3N4O6
6a,9a-Dichloro-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-[5-(hydroxymethyl)furan-2-yl]-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6S)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-[(4-propan-2-yloxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C27H37N5O4
(6S)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-[(4-propan-2-yloxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cycloheptyl-2-N-[(2,4-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O5
(6S)-6-N-cycloheptyl-2-N-[(2,4-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-2-N-[3-(diethylamino)propyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H40N6O3
(6R)-6-N-cyclopentyl-2-N-[3-(diethylamino)propyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-butyl-6-N-cyclopentyl-6-methyl-4-oxo-2-N-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C21H33N5O3
(6R)-5-butyl-6-N-cyclopentyl-6-methyl-4-oxo-2-N-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H43N7O3
(6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-2-N-[[(2S)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C20H31N5O4
(6R)-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-2-N-[[(2S)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-[3-(2-oxopyrrolidin-1-yl)propyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H34N6O4
(6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-[3-(2-oxopyrrolidin-1-yl)propyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(diethylamino)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H40N6O3
(6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(diethylamino)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-2-N-[2-(diethylamino)ethyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H38N6O3
(6S)-6-N-cyclopentyl-2-N-[2-(diethylamino)ethyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-6-methyl-4-oxo-2-N-propan-2-yl-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C20H31N5O3
(6R)-6-N-cyclopentyl-6-methyl-4-oxo-2-N-propan-2-yl-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-6-methyl-4-oxo-5-propyl-2-N-(2-pyrrolidin-1-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H36N6O3
(6S)-6-N-cyclopentyl-6-methyl-4-oxo-5-propyl-2-N-(2-pyrrolidin-1-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-(pyrrolidine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C20H29N5O3
(6S)-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-(pyrrolidine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-6-N-cyclopentyl-6-methyl-2-N-(3-methylbutyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H35N5O3
(6R)-6-N-cyclopentyl-6-methyl-2-N-(3-methylbutyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-butyl-6-N-cyclopentyl-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H43N7O3
(6R)-5-butyl-6-N-cyclopentyl-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H37N5O3
(6S)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-2-N-(3-propan-2-yloxypropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C21H35N5O4
(6R)-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-2-N-(3-propan-2-yloxypropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— 6-[2-[(2-chlorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-(furan-2-ylmethyl)hexanamide —— C26H26ClN3O3S
6-[2-[(2-chlorophenyl)methylsulfanyl]-4-oxoquinazolin-3-yl]-N-(furan-2-ylmethyl)hexanamide
—— (6R)-6-N-cyclopentyl-6-methyl-4-oxo-5-propyl-2-N-(2-pyrrolidin-1-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H36N6O3
(6R)-6-N-cyclopentyl-6-methyl-4-oxo-5-propyl-2-N-(2-pyrrolidin-1-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— 6-[6-(2-Hydroxy-4-phenylmethoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C36H35NO8
6-[6-(2-Hydroxy-4-phenylmethoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6a,9a-Dichloro-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(1-hydroxynaphthalen-2-yl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C39H33Cl2N5O5
6a,9a-Dichloro-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(1-hydroxynaphthalen-2-yl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— (6S)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-(3-propan-2-yloxypropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H37N5O4
(6S)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-(3-propan-2-yloxypropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-[(5-methylfuran-2-yl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H29N5O4
(6R)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-[(5-methylfuran-2-yl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cycloheptyl-2-N-[(2,5-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O5
(6R)-6-N-cycloheptyl-2-N-[(2,5-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-5,6-dimethyl-2-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H31N5O3S
(6R)-6-N-cyclopentyl-5,6-dimethyl-2-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cycloheptyl-2-N-[2-(2-methoxyphenyl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O4
(6S)-6-N-cycloheptyl-2-N-[2-(2-methoxyphenyl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cycloheptyl-2-N-[(3,4-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O5
(6S)-6-N-cycloheptyl-2-N-[(3,4-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-2-N-[2-(diethylamino)ethyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H36N6O3
(6R)-6-N-cyclopentyl-2-N-[2-(diethylamino)ethyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-[(4-propan-2-yloxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C27H37N5O4
(6R)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-[(4-propan-2-yloxyphenyl)methyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-[3-(2-oxopyrrolidin-1-yl)propyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H36N6O4
(6S)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-[3-(2-oxopyrrolidin-1-yl)propyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-2-N-[2-(dimethylamino)ethyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C19H32N6O3
(6S)-2-N-[2-(dimethylamino)ethyl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-2-N-[(2R)-butan-2-yl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C19H31N5O3
(6S)-2-N-[(2R)-butan-2-yl]-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cycloheptyl-2-N-[(4-ethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O4
(6R)-6-N-cycloheptyl-2-N-[(4-ethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-(3-pyrrolidin-1-ylpropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H38N6O3
(6R)-6-N-cycloheptyl-5,6-dimethyl-4-oxo-2-N-(3-pyrrolidin-1-ylpropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-(2-morpholin-4-ylethyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H34N6O4
(6S)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-(2-morpholin-4-ylethyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cycloheptyl-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H41N7O3
(6S)-6-N-cycloheptyl-2-N-[2-(4-ethylpiperazin-1-yl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cycloheptyl-2-N-[(2,3-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O5
(6S)-6-N-cycloheptyl-2-N-[(2,3-dimethoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide