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—— (6S)-5-(1,3-benzodioxol-5-ylmethyl)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H30N4O5
(6S)-5-(1,3-benzodioxol-5-ylmethyl)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-[(2-ethoxyphenyl)methyl]-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O4
(6R)-N-cyclohexyl-5-[(2-ethoxyphenyl)methyl]-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-6-methyl-5-(4-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H28N4O2S
(6R)-N-cyclohexyl-6-methyl-5-(4-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H29FN4O2S
(6R)-N-cycloheptyl-5-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-benzyl-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H28N4O2S
(6S)-5-benzyl-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H28N4O3S
(6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-5-(4-ethylphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O3
(6S)-N-cycloheptyl-5-(4-ethylphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-5-(4-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H28N4O3
(6S)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-5-(4-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-(3-chloro-4-methoxyphenyl)-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27ClN4O3S
(6R)-5-(3-chloro-4-methoxyphenyl)-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S2
(6R)-N-cycloheptyl-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-5-(4-fluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27FN4O2S
(6S)-N-cycloheptyl-5-(4-fluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-(2,3-dimethylphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S
(6S)-N-cyclohexyl-5-(2,3-dimethylphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-6-methyl-5-[(2-methylphenyl)methyl]-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S
(6S)-N-cyclohexyl-6-methyl-5-[(2-methylphenyl)methyl]-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-2-(furan-2-yl)-5-[(3-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O4
(6S)-N-cyclohexyl-2-(furan-2-yl)-5-[(3-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-phenylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H34N4O3
(6S)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-phenylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(2-phenylethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3
(6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(2-phenylethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-5-(4-ethoxyphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O4
(6R)-N-cycloheptyl-5-(4-ethoxyphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-bromo-N-(6-tert-butyl-3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-phenylquinoline-4-carboxamide —— C29H28BrN3O2S
6-bromo-N-(6-tert-butyl-3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-phenylquinoline-4-carboxamide
—— (6S)-5-(1,3-benzodioxol-5-ylmethyl)-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H28N4O4S
(6S)-5-(1,3-benzodioxol-5-ylmethyl)-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-2-(furan-2-yl)-5-(furan-2-ylmethyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H28N4O4
(6S)-N-cycloheptyl-2-(furan-2-yl)-5-(furan-2-ylmethyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-(3-{[(4-Cyanophenyl)carbamoyl]amino}phenyl)-N,N,8-trimethyl-2H,3H,4H,6H-pyrimido[2,1-B][1,3]thiazine-7-carboxamide —— C25H26N6O2S
6-(3-{[(4-Cyanophenyl)carbamoyl]amino}phenyl)-N,N,8-trimethyl-2H,3H,4H,6H-pyrimido[2,1-B][1,3]thiazine-7-carboxamide
—— (6S)-5-(3-chloro-4-methylphenyl)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27ClN4O3
(6S)-5-(3-chloro-4-methylphenyl)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-(2,4-dimethylphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3
(6R)-N-cyclohexyl-5-(2,4-dimethylphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-[(2-fluorophenyl)methyl]-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27FN4O3
(6S)-N-cyclohexyl-5-[(2-fluorophenyl)methyl]-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-[(2-chlorophenyl)methyl]-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H29ClN4O3
(6S)-5-[(2-chlorophenyl)methyl]-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-benzyl-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H28N4O2S
(6R)-5-benzyl-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-(4-ethylphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S
(6R)-N-cyclohexyl-5-(4-ethylphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-[(3-fluorophenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27FN4O2S
(6S)-N-cyclohexyl-5-[(3-fluorophenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27ClN4O2S
(6R)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-(3,5-dimethylphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3
(6R)-N-cyclohexyl-5-(3,5-dimethylphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-(4-chlorophenyl)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27ClN4O3
(6S)-5-(4-chlorophenyl)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27ClN4O2S
(6S)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-5-[(3-methoxyphenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O3S
(6R)-N-cycloheptyl-5-[(3-methoxyphenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-6-methyl-5-(4-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S
(6S)-N-cycloheptyl-6-methyl-5-(4-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-5-[(3-methoxyphenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O3S
(6S)-N-cycloheptyl-5-[(3-methoxyphenyl)methyl]-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-6-methyl-5-(2-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S
(6R)-N-cycloheptyl-6-methyl-5-(2-methylphenyl)-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-(3-methoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H28N4O3S
(6S)-N-cyclohexyl-5-(3-methoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-Tert-butyl-2-[(3-pentoxybenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C25H34N2O3S
6-Tert-butyl-2-[(3-pentoxybenzoyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-N-cyclohexyl-6-methyl-4-oxo-5-(3-phenylpropyl)-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O2S
(6R)-N-cyclohexyl-6-methyl-4-oxo-5-(3-phenylpropyl)-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-(2,4-difluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H24F2N4O2S
(6S)-N-cyclohexyl-5-(2,4-difluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-chloro-N-[(1S)-3-methyl-1-phenylbutyl]pyridine-3-carboxamide —— C17H19ClN2O
6-chloro-N-[(1S)-3-methyl-1-phenylbutyl]pyridine-3-carboxamide
—— (6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-phenylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O3
(6R)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-phenylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— [6-(4-Pyrimidin-2-ylpiperazine-1-carbonyl)pyridin-3-yl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone —— C23H25N9O2
[6-(4-Pyrimidin-2-ylpiperazine-1-carbonyl)pyridin-3-yl]-(4-pyrimidin-2-ylpiperazin-1-yl)methanone
—— (6S)-N-cyclohexyl-5-(4-ethoxyphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O4
(6S)-N-cyclohexyl-5-(4-ethoxyphenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-chloro-N-[(1R)-3-methyl-1-phenylbutyl]pyridine-3-carboxamide —— C17H19ClN2O
6-chloro-N-[(1R)-3-methyl-1-phenylbutyl]pyridine-3-carboxamide
—— 6-[6-(3-hydroxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-8-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid —— C33H34N2O7
6-[6-(3-hydroxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-8-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid
—— (6R)-N-cyclohexyl-5-(2-fluorophenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H25FN4O3
(6R)-N-cyclohexyl-5-(2-fluorophenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-chloro-N-[(1R)-1-(4-methoxyphenyl)propyl]pyridine-3-carboxamide —— C16H17ClN2O2
6-chloro-N-[(1R)-1-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
—— 6-(4-hydroxynaphthalen-1-yl)-1,3,7,10-tetraoxo-6a,9-diphenyl-4,6,10a,11,11a,11b-hexahydro-3aH-naphtho[2,3-e]isoindole-2-carboxamide —— C39H30N2O6
6-(4-hydroxynaphthalen-1-yl)-1,3,7,10-tetraoxo-6a,9-diphenyl-4,6,10a,11,11a,11b-hexahydro-3aH-naphtho[2,3-e]isoindole-2-carboxamide
—— (6R)-N-cyclohexyl-2-(furan-2-yl)-5-(furan-2-ylmethyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C23H26N4O4
(6R)-N-cyclohexyl-2-(furan-2-yl)-5-(furan-2-ylmethyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide