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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H14ClF3N2O3S2
(2R)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(4-ethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(2R)-N-(4-ethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-2-methyl-4-oxo-N-(pyridin-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H17N3O3S2
(2S)-2-methyl-4-oxo-N-(pyridin-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[(4-chlorophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17ClN2O3S2
(2R)-N-[(4-chlorophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(4-bromo-2-fluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14BrFN2O3S2
(2S)-N-(4-bromo-2-fluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-7-(azepan-1-ylsulfonyl)-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C16H22N2O3S2
(2S)-7-(azepan-1-ylsulfonyl)-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-N-(2,4-difluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14F2N2O3S2
(2S)-N-(2,4-difluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(4-methoxyphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H18N2O4S2
(2S)-N-(4-methoxyphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-2-methyl-N-(5-methylpyridin-2-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H17N3O3S2
(2S)-2-methyl-N-(5-methylpyridin-2-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-2-methyl-N-(6-methylpyridin-2-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H17N3O3S2
(2S)-2-methyl-N-(6-methylpyridin-2-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(2,5-difluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14F2N2O3S2
(2S)-N-(2,5-difluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(3-fluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H15FN2O3S2
(2S)-N-(3-fluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— ethyl 1-[[(2R)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]piperidine-4-carboxylate —— C18H24N2O5S2
ethyl 1-[[(2R)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]piperidine-4-carboxylate
—— (2R)-7-(4-cyclohexylpiperazin-1-yl)sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H29N3O3S2
(2R)-7-(4-cyclohexylpiperazin-1-yl)sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-N-(4-ethoxyphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O4S2
(2S)-N-(4-ethoxyphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(5-chloropyridin-2-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C15H14ClN3O3S2
(2R)-N-(5-chloropyridin-2-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(2-fluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H15FN2O3S2
(2R)-N-(2-fluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(5-chloro-2-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17ClN2O3S2
(2S)-N-(5-chloro-2-methylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-2-methyl-4-oxo-N-[3-(trifluoromethyl)phenyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15F3N2O3S2
(2R)-2-methyl-4-oxo-N-[3-(trifluoromethyl)phenyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(2,3-dimethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(2R)-N-(2,3-dimethylphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(2,4-dimethoxyphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O5S2
(2R)-N-(2,4-dimethoxyphenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(6-methoxy-1,3-benzothiazol-2-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H17N3O4S3
(2R)-N-(6-methoxy-1,3-benzothiazol-2-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-ethyl-2-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(2R)-N-ethyl-2-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-7-(1,2-dihydroimidazo[1,2-a]benzimidazol-3-ylsulfonyl)-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H18N4O3S2
(2S)-7-(1,2-dihydroimidazo[1,2-a]benzimidazol-3-ylsulfonyl)-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H19N3O4S3
(2S)-N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-[(2R)-butan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C13H18N2O3S2
N-[(2R)-butan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 4-oxo-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H20N2O3S2
4-oxo-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2S)-2-methyl-2,3-dihydroindol-1-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C18H18N2O3S2
7-[[(2S)-2-methyl-2,3-dihydroindol-1-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— N-[(2S)-butan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C13H18N2O3S2
N-[(2S)-butan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2R)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H19ClN2O4S2
7-[[(2R)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— 7-[[(2S)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H19ClN2O4S2
7-[[(2S)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— 4-oxo-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H20N2O3S2
4-oxo-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1R)-1-phenylethyl]urea —— C24H23N3O2S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1R)-1-phenylethyl]urea
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S)-1-phenylethyl]urea —— C24H23N3O2S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S)-1-phenylethyl]urea
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2S)-2-phenylpropyl]urea —— C25H25N3O2S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(2S)-2-phenylpropyl]urea
—— (2-bromo-5-methoxyphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C18H18BrNO2S
(2-bromo-5-methoxyphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (2-bromo-5-methoxyphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C18H18BrNO2S
(2-bromo-5-methoxyphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 2-(4-chlorophenyl)-10-phenyl-9,10-dihydro-1H-pyrrolo[3,4-b][1,5]benzothiazepine-1,3(2H)-dione —— C23H15ClN2O2S
2-(4-chlorophenyl)-10-phenyl-9,10-dihydro-1H-pyrrolo[3,4-b][1,5]benzothiazepine-1,3(2H)-dione
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-bromobenzoate —— C19H18BrNO3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-bromobenzoate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-bromobenzoate —— C19H18BrNO3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-bromobenzoate
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[4-(2-methylphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C26H25N5OS2
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[4-(2-methylphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[4-(2-methylphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C26H25N5OS2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[4-(2-methylphenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-methyl-4-oxophthalazine-1-carboxylate —— C22H21N3O4S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-methyl-4-oxophthalazine-1-carboxylate
—— (3,5-dimethylphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C19H21NOS
(3,5-dimethylphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-phenylmethanone —— C17H17NOS
[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-phenylmethanone
—— (3,5-dimethylphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C19H21NOS
(3,5-dimethylphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (2-fluorophenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C17H16FNOS
(2-fluorophenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (2-fluorophenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C17H16FNOS
(2-fluorophenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-phenylmethanone —— C17H17NOS
[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-phenylmethanone
—— (11R)-5-ethyl-3-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H29N3O3S
(11R)-5-ethyl-3-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one