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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11S)-N-cyclopentyl-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23FN2O3S
(11S)-N-cyclopentyl-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(2,2-dimethoxyethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23FN2O5S
(11R)-N-(2,2-dimethoxyethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-N-(2,2-diethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O5S
(11R)-5-benzyl-N-(2,2-diethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C26H24N2O3S
(11R)-5-benzyl-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O4S
(11S)-5-[(4-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O4S
(11R)-5-benzyl-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(3-cyclohexylsulfanylpropyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H30N2O3S2
(11R)-N-(3-cyclohexylsulfanylpropyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H29N3O3S
(11S)-5-benzyl-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11S)-5-ethyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O3S
(11S)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C23H26N2O3S
(11R)-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-benzyl-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O3S
(11S)-5-benzyl-N-cyclopentyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-butyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O3S
(11S)-N-butyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H25FN2O5S
(11R)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-benzyl-N-[(2-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H21ClN2O3S
(11R)-5-benzyl-N-[(2-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-[(2-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H21ClN2O3S
(11S)-5-benzyl-N-[(2-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C32H28N2O3S
(11R)-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[2-(diethylamino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28ClN3O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[2-(diethylamino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(2-methylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H30N2O3S
(11S)-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(2-methylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— 10-allyl-11-oxo-N-(2-phenylethyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C25H22N2O2S
10-allyl-11-oxo-N-(2-phenylethyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— 3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C28H27FN2O4S
3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— N-[(2S)-butan-2-yl]-5-[(3-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O4S
N-[(2S)-butan-2-yl]-5-[(3-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-butyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O3S
(11R)-N-butyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(2-chlorophenyl)methyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C23H19ClN2O3S
(11S)-N-[(2-chlorophenyl)methyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O4S
(11S)-5-benzyl-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N,N-dipropylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N,N-dipropylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-(2,2-diethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27ClN2O5S
(11S)-5-[(4-chlorophenyl)methyl]-N-(2,2-diethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C25H24N4O3S
(11S)-5-ethyl-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11R)-N-cyclopropyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O3S
(11R)-N-cyclopropyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H25FN2O3S
(11S)-5-[(4-fluorophenyl)methyl]-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[2-(dipropylamino)ethyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H32FN3O3S
(11S)-N-[2-(dipropylamino)ethyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(2-methylphenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C27H26N2O3S
(11R)-5-[(2-methylphenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-N,5-bis[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H20F2N2O3S
(11S)-N,5-bis[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-methylphenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C29H30N2O4S
3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-methylphenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— ethyl 4-[(11R)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperazine-1-carboxylate —— C23H25N3O5S
ethyl 4-[(11R)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperazine-1-carboxylate
—— (11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H27FN2O3S
(11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H27FN2O3S
(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-N-cyclopropyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H19ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-N-cyclopropyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21FN2O3S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-ethyl-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C25H24N4O3S
(11R)-5-ethyl-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21FN2O3S
(11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O4S
(11R)-5-benzyl-6,11-dioxo-N-(3-propan-2-yloxypropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C23H26N2O4S
3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— 10-allyl-N-cyclooctyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C25H28N2O2S
10-allyl-N-cyclooctyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O3S
(11R)-5-[(4-fluorophenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(azepane-1-carbonyl)-5-[(4-chlorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25ClN2O3S
(11R)-3-(azepane-1-carbonyl)-5-[(4-chlorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-fluorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C26H23FN2O3S
(11S)-5-[(4-fluorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one