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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11S)-5-[(3-chlorophenyl)methyl]-N-(2-methylphenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H21ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-(2-methylphenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 6,7,10-trimethyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H26N2OS
6,7,10-trimethyl-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 6,7,10-trimethyl-N-[(2R)-1-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2OS
6,7,10-trimethyl-N-[(2R)-1-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 6,7,10-trimethyl-N-[(2S)-1-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2OS
6,7,10-trimethyl-N-[(2S)-1-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-(2-methylphenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H21ClN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-N-(2-methylphenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (2S)-N-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2,2-dimethyl-4-oxo-3H-1,5-benzothiazepin-5-yl)propanamide —— C24H30N2O4S
(2S)-N-[2-(3,4-dimethoxyphenyl)ethyl]-2-(2,2-dimethyl-4-oxo-3H-1,5-benzothiazepin-5-yl)propanamide
—— N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O2S2
N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O2S2
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(4-methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20FN3O3S
(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-ethyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H27N3O3S
(11R)-5-ethyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H23N3O3S
(11S)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20FN3O3S
(11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H21N3O3S
(11S)-5-benzyl-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H25N3O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-ethyl-3-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C28H29N3O4S
5-ethyl-3-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20FN3O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H27N3O3S
(11S)-5-ethyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H29N3O3S
(11R)-5-benzyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20FN3O3S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H21N3O3S
(11R)-5-benzyl-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H21N3O3S
(11S)-5-benzyl-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H23N3O3S
(11R)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H25N3O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20FN3O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H21N3O3S
(11R)-5-benzyl-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H29N3O3S
(11S)-5-benzyl-N-[2-(N-ethylanilino)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H20FN3O3S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide —— C26H25N3O4S
N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide
—— N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide —— C25H32N4O2S
N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide
—— N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide —— C25H32N4O2S
N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)butanamide
—— 5-[(2-chloro-6-fluorophenyl)methyl]-3-[(2S,6R)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one —— C28H26ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-3-[(2S,6R)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one
—— 5-[(2-chloro-6-fluorophenyl)methyl]-3-[(2R,6R)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one —— C28H26ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-3-[(2R,6R)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one
—— 3-[(2R,6R)-2,6-dimethylpiperidine-1-carbonyl]-5-[(4-ethoxyphenyl)methyl]benzo[b][1,4]benzothiazepin-6-one —— C30H32N2O3S
3-[(2R,6R)-2,6-dimethylpiperidine-1-carbonyl]-5-[(4-ethoxyphenyl)methyl]benzo[b][1,4]benzothiazepin-6-one
—— 5-[(4-ethoxyphenyl)methyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H35N3O3S
5-[(4-ethoxyphenyl)methyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H28ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-ethoxyphenyl)methyl]-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H35N3O3S
5-[(4-ethoxyphenyl)methyl]-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(2S,6R)-2,6-dimethylpiperidine-1-carbonyl]-5-[(4-ethoxyphenyl)methyl]benzo[b][1,4]benzothiazepin-6-one —— C30H32N2O3S
3-[(2S,6R)-2,6-dimethylpiperidine-1-carbonyl]-5-[(4-ethoxyphenyl)methyl]benzo[b][1,4]benzothiazepin-6-one
—— N-[(2R)-butan-2-yl]-5-[(2-chloro-6-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H22ClFN2O2S
N-[(2R)-butan-2-yl]-5-[(2-chloro-6-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]-5-[(4-ethoxyphenyl)methyl]benzo[b][1,4]benzothiazepin-6-one —— C30H32N2O3S
3-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]-5-[(4-ethoxyphenyl)methyl]benzo[b][1,4]benzothiazepin-6-one
—— 5-[(2-chloro-6-fluorophenyl)methyl]-3-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one —— C28H26ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-3-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one
—— 5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H28ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chloro-6-fluorophenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClFN3O2S
5-[(2-chloro-6-fluorophenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chloro-6-fluorophenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClFN3O2S
5-[(2-chloro-6-fluorophenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2S)-butan-2-yl]-5-[(2-chloro-6-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H22ClFN2O2S
N-[(2S)-butan-2-yl]-5-[(2-chloro-6-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-methoxyphenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C30H26N2O3S
5-[(3-methoxyphenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H28ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-methoxyphenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H30N2O3S
5-[(3-methoxyphenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O3S
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(3-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H28ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chloro-6-fluorophenyl)methyl]-6-oxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H22ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-6-oxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide