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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11S)-5-benzyl-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H30N2O3S
(11S)-5-benzyl-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-N-(3-ethoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O4S
(11R)-5-benzyl-N-(3-ethoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(azepane-1-carbonyl)-5-[(4-chlorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25ClN2O3S
(11S)-3-(azepane-1-carbonyl)-5-[(4-chlorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— N-[(2R)-butan-2-yl]-5-[(3-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O4S
N-[(2R)-butan-2-yl]-5-[(3-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[2-(dimethylamino)ethyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H29N3O3S
(11S)-N-[2-(dimethylamino)ethyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28ClN3O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-N-(2,2-dimethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O5S
(11R)-5-[(4-chlorophenyl)methyl]-N-(2,2-dimethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H26N2O4S
(11R)-5-[(2-methylphenyl)methyl]-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C23H26N2O4S
3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-ethyl-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-(2,2-diethoxyethyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C22H26N2O5S
(11S)-N-(2,2-diethoxyethyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H25FN2O3S
(11R)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-N-[(2S)-butan-2-yl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2O3S
(11R)-5-benzyl-N-[(2S)-butan-2-yl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-N-(2-morpholin-4-ylethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H26FN3O4S
(11S)-5-[(4-fluorophenyl)methyl]-N-(2-morpholin-4-ylethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-cyclopropyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O3S
(11S)-N-cyclopropyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2R)-butan-2-yl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23FN2O4S
N-[(2R)-butan-2-yl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O3S
(11S)-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(2-chlorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H20ClFN2O3S
(11S)-N-[(2-chlorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C23H24N2O5S
(11R)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-cyclohexyl-5-[(2,5-dimethylphenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32N2O3S
(11S)-N-cyclohexyl-5-[(2,5-dimethylphenyl)methyl]-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N,5-dibenzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H22N2O3S
(11R)-N,5-dibenzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C30H24N2O3S
(11R)-5-benzyl-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28N2O4S
(11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-ethyl-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2O3S
(11R)-5-ethyl-N-[2-(4-methylphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(3-ethoxypropyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25FN2O4S
(11R)-N-(3-ethoxypropyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(4-chlorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H20ClFN2O3S
(11S)-N-[(4-chlorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H31N3O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O3S
(11S)-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O3S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(azepane-1-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H30N2O3S
(11R)-3-(azepane-1-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-(3-ethoxypropyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O4S
(11S)-N-(3-ethoxypropyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-[3-(diethylamino)propyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H30ClN3O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-[3-(diethylamino)propyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-benzyl-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H21ClN2O3S
(11R)-N-benzyl-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-ethyl-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11R)-5-ethyl-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H28N2O4S
N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-N-[3-[cyclohexyl(methyl)amino]propyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H35N3O3S
(11R)-5-benzyl-N-[3-[cyclohexyl(methyl)amino]propyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C23H24N2O5S
(11S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— N-cyclopentyl-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C22H22N2O2S
N-cyclopentyl-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-butyl-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C21H22N2O2S
N-butyl-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21FN2O4S
(11S)-5-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H28N2O4S
N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-5-ethyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[3-(azepan-1-yl)propyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H31N3O3S
(11R)-N-[3-(azepan-1-yl)propyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-ethyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11R)-5-ethyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H27FN2O3S
(11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O4S
(11R)-5-[(2-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-ethyl-3-[4-(4-nitrophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C26H24N4O5S
(11R)-5-ethyl-3-[4-(4-nitrophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21FN2O4S
(11S)-5-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-N-[(1R,2R)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide