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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-methyl-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S3
(2R)-2-methyl-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[3-(N-ethylanilino)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O3S2
(2S)-N-[3-(N-ethylanilino)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-(2-phenylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3S)-3-methyl-4-oxo-N-(2-phenylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-(pyridin-3-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H17N3O3S2
(3R)-3-methyl-4-oxo-N-(pyridin-3-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O5S2
(3S)-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(4-ethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O4S2
(3S)-N-(4-ethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-N-[(5-methylfuran-2-yl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H18N2O4S2
(3R)-3-methyl-N-[(5-methylfuran-2-yl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-N-(2-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H18N2O3S2
(3R)-3-methyl-N-(2-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[2-(furan-2-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H18N2O4S2
(3R)-N-[2-(furan-2-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-(furan-2-ylmethyl)-4-oxo-N-[(1R)-1-phenylethyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H22N2O4S2
N-(furan-2-ylmethyl)-4-oxo-N-[(1R)-1-phenylethyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[[5-(azepan-1-ylmethyl)furan-2-yl]methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O4S2
(3R)-N-[[5-(azepan-1-ylmethyl)furan-2-yl]methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H27N3O3S2
(3S)-N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(1,3-benzodioxol-5-yl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H16N2O5S2
(3S)-N-(1,3-benzodioxol-5-yl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[(3-bromophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17BrN2O3S2
(2R)-N-[(3-bromophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-cyclopentyl-2-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O3S3
(2S)-N-cyclopentyl-2-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(4-fluoro-2-methylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17FN2O3S2
(3R)-N-(4-fluoro-2-methylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-N-[3-(1,2-oxazol-5-yl)phenyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H17N3O4S2
(3R)-3-methyl-N-[3-(1,2-oxazol-5-yl)phenyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[(3-bromophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17BrN2O3S2
(2S)-N-[(3-bromophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-2-methyl-4-oxo-N-(2-pyrrolidin-1-ylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H23N3O3S2
(2R)-2-methyl-4-oxo-N-(2-pyrrolidin-1-ylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-7-morpholin-4-ylsulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C14H18N2O4S2
(3S)-3-methyl-7-morpholin-4-ylsulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-N-(2,5-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14F2N2O3S2
(3R)-N-(2,5-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H16N2O3S2
(3S)-3-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(2,5-diethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O5S2
(3S)-N-(2,5-diethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— ethyl 4-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]benzoate —— C19H20N2O5S2
ethyl 4-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]benzoate
—— (3R)-7-[4-(furan-2-carbonyl)piperazin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H21N3O5S2
(3R)-7-[4-(furan-2-carbonyl)piperazin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-7-[4-(furan-2-carbonyl)piperazin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H21N3O5S2
(2S)-7-[4-(furan-2-carbonyl)piperazin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-N-(2-ethylphenyl)-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(2S)-N-(2-ethylphenyl)-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-7-[4-[methyl(3-morpholin-4-ylpropyl)amino]piperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C23H36N4O4S2
(3S)-3-methyl-7-[4-[methyl(3-morpholin-4-ylpropyl)amino]piperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2R)-2-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H27N3O3S2
(2R)-2-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— ethyl 3-[N-[[(2S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate —— C21H24N2O5S2
ethyl 3-[N-[[(2S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate
—— (3R)-3-methyl-4-oxo-N-(2-thiophen-2-ylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H18N2O3S3
(3R)-3-methyl-4-oxo-N-(2-thiophen-2-ylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[(2,5-dimethylphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(3S)-N-[(2,5-dimethylphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(2-chloro-4,6-dimethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H19ClN2O5S2
(3R)-N-(2-chloro-4,6-dimethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— methyl 4-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]benzoate —— C18H18N2O5S2
methyl 4-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonylamino]benzoate
—— (3S)-7-(azepan-1-ylsulfonyl)-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C16H22N2O3S2
(3S)-7-(azepan-1-ylsulfonyl)-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-7-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H20N2O3S2
(3S)-7-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C15H16N2O4S2
(3R)-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(3-bromophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H15BrN2O3S2
(2R)-N-(3-bromophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-(4-propan-2-ylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(3R)-3-methyl-4-oxo-N-(4-propan-2-ylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(3,4-dimethylphenyl)-N,3-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(3S)-N-(3,4-dimethylphenyl)-N,3-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O4S2
(3S)-3-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2R)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C18H18N2O3S3
7-[[(2R)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-N-[3-[benzyl(ethyl)amino]propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O3S2
(3R)-N-[3-[benzyl(ethyl)amino]propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N,3-dimethyl-N-(3-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3S)-N,3-dimethyl-N-(3-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-7-[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C22H25N3O5S2
(2S)-7-[4-(1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-2-methyl-N-[(3-methylphenyl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(2S)-2-methyl-N-[(3-methylphenyl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[3-(furan-2-yl)propyl]-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H22N2O4S2
(2R)-N-[3-(furan-2-yl)propyl]-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[(4-bromophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17BrN2O3S2
(2S)-N-[(4-bromophenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— ethyl 3-[N-[[(2R)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate —— C21H24N2O5S2
ethyl 3-[N-[[(2R)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate
—— (3S)-3-methyl-N-[3-(1,2-oxazol-5-yl)phenyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H17N3O4S2
(3S)-3-methyl-N-[3-(1,2-oxazol-5-yl)phenyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide