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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [2-hydroxy-4-(methylideneamino)phenyl]-(7-methoxy-3,5-dihydro-2H-1,4-benzothiazepin-4-yl)methanone —— C18H18N2O3S
[2-hydroxy-4-(methylideneamino)phenyl]-(7-methoxy-3,5-dihydro-2H-1,4-benzothiazepin-4-yl)methanone
—— 2,2,2-trifluoro-1-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]ethanone —— C12H12F3NO2S
2,2,2-trifluoro-1-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]ethanone
—— 7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepine-4-carbaldehyde —— C11H13NO2S
7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepine-4-carbaldehyde
—— benzyl 4-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepine-4-carbonyl]piperazine-1-carboxylate —— C23H27N3O4S
benzyl 4-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepine-4-carbonyl]piperazine-1-carboxylate
—— 1-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]ethanone —— C12H15NO2S
1-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]ethanone
—— methyl 7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepine-4-carboxylate —— C12H15NO3S
methyl 7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepine-4-carboxylate
—— (6aR)-2-(hydroxymethyl)-6a,7,8,11-tetrahydro-6H-pyrrolo[2,1-c][1,4]benzothiazepin-9-one —— C13H15NO2S
(6aR)-2-(hydroxymethyl)-6a,7,8,11-tetrahydro-6H-pyrrolo[2,1-c][1,4]benzothiazepin-9-one
—— [7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]-morpholin-4-ylmethanone —— C15H20N2O3S
[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]-morpholin-4-ylmethanone
—— 1-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]prop-2-en-1-one —— C13H15NO2S
1-[7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzothiazepin-4-yl]prop-2-en-1-one
—— (11S,11aS)-11-(2-ethoxyphenyl)-11,11a-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11S,11aS)-11-(2-ethoxyphenyl)-11,11a-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11R,11aS)-11-(2-ethoxyphenyl)-11,11a-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11R,11aS)-11-(2-ethoxyphenyl)-11,11a-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— Benzo[b][1,4]benzothiazepine-9-carbonyl chloride —— C14H8ClNOS
Benzo[b][1,4]benzothiazepine-9-carbonyl chloride
—— 7-Chlorobenzo[b][1,4]benzothiazepine-9-carboxamide —— C14H9ClN2OS
7-Chlorobenzo[b][1,4]benzothiazepine-9-carboxamide
—— methyl 4-[(11R,11aS)-12-oxo-11,11a-dihydroindeno[2,1-c][1,5]benzothiazepin-11-yl]benzoate —— C24H17NO3S
methyl 4-[(11R,11aS)-12-oxo-11,11a-dihydroindeno[2,1-c][1,5]benzothiazepin-11-yl]benzoate
—— [[(3S)-2,2-dimethyl-4-oxo-3,5-dihydro-1,5-benzothiazepin-3-yl]amino]methyl-[(2S)-1-oxopropan-2-yl]carbamic acid —— C16H21N3O4S
[[(3S)-2,2-dimethyl-4-oxo-3,5-dihydro-1,5-benzothiazepin-3-yl]amino]methyl-[(2S)-1-oxopropan-2-yl]carbamic acid
—— [(1S)-1-[[(3R)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-2,2-dimethyl-4-oxo-3H-1,5-benzothiazepin-3-yl]amino]ethyl]-(1-oxopropan-2-yl)carbamic acid —— C34H32N6O4S
[(1S)-1-[[(3R)-5-[[2-cyano-1-(2-cyanophenyl)indol-3-yl]methyl]-2,2-dimethyl-4-oxo-3H-1,5-benzothiazepin-3-yl]amino]ethyl]-(1-oxopropan-2-yl)carbamic acid
—— 2,2-dimethyl-4,5-dihydro-3H-1,5-benzothiazepin-3-amine —— C11H16N2S
2,2-dimethyl-4,5-dihydro-3H-1,5-benzothiazepin-3-amine
—— (2,2-Dimethyl-4-oxo-3,5-dihydro-1,5-benzothiazepin-3-yl)carbamic acid —— C12H14N2O3S
(2,2-Dimethyl-4-oxo-3,5-dihydro-1,5-benzothiazepin-3-yl)carbamic acid
—— [[(3R)-2,2-dimethyl-4-oxo-3,5-dihydro-1,5-benzothiazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate —— C16H21N3O4S
[[(3R)-2,2-dimethyl-4-oxo-3,5-dihydro-1,5-benzothiazepin-3-yl]amino] N-methyl-N-[(2S)-1-oxopropan-2-yl]carbamate
—— (11R)-11-(2,3,4,5-tetramethylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C26H23NOS
(11R)-11-(2,3,4,5-tetramethylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11S)-11-(2,3,4,5-tetramethylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C26H23NOS
(11S)-11-(2,3,4,5-tetramethylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (6S,6aR)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C21H21NO2S
(6S,6aR)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (6R,6aS)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C21H21NO2S
(6R,6aS)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (11R)-11-(3-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11R)-11-(3-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11S)-11-(3-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11S)-11-(3-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (6S,6aS)-9,9-dimethyl-6-naphthalen-1-yl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C25H23NOS
(6S,6aS)-9,9-dimethyl-6-naphthalen-1-yl-6,6a,8,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (11R)-11-(4-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11R)-11-(4-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11S)-11-(4-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11S)-11-(4-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— N,N-dihydroxy-3-[4-(4-methylphenyl)-2,3-dihydro-1,5-benzothiazepin-2-yl]aniline —— C22H20N2O2S
N,N-dihydroxy-3-[4-(4-methylphenyl)-2,3-dihydro-1,5-benzothiazepin-2-yl]aniline
—— (6S,6aR,9R)-9-phenyl-6-pyridin-3-yl-6a,8,9,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C24H20N2OS
(6S,6aR,9R)-9-phenyl-6-pyridin-3-yl-6a,8,9,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (11S)-11-(2-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11S)-11-(2-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11R)-11-(2-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C24H19NO2S
(11R)-11-(2-ethoxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (5R)-1-methyl-5-phenyl-5,6-dihydropyrano[4,3-b][1,5]benzothiazepin-4-one —— C19H15NO2S
(5R)-1-methyl-5-phenyl-5,6-dihydropyrano[4,3-b][1,5]benzothiazepin-4-one
—— (5S)-1-methyl-5-phenyl-5,6-dihydropyrano[4,3-b][1,5]benzothiazepin-4-one —— C19H15NO2S
(5S)-1-methyl-5-phenyl-5,6-dihydropyrano[4,3-b][1,5]benzothiazepin-4-one
—— (11S)-11-(4-methylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C23H17NOS
(11S)-11-(4-methylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11R)-11-(4-methylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C23H17NOS
(11R)-11-(4-methylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— 7-[(3-chloro-6-methyl-1H-benzo[c][2,1]benzothiazepin-11-yl)amino]heptanoic acid —— C21H25ClN2O2S
7-[(3-chloro-6-methyl-1H-benzo[c][2,1]benzothiazepin-11-yl)amino]heptanoic acid
—— (11S)-11-(4-methylsulfanylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C23H17NOS2
(11S)-11-(4-methylsulfanylphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11R)-11-(5-bromo-2-hydroxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C22H14BrNO2S
(11R)-11-(5-bromo-2-hydroxyphenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11R)-11-(2-chlorophenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C22H14ClNOS
(11R)-11-(2-chlorophenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11S)-11-(2-chlorophenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C22H14ClNOS
(11S)-11-(2-chlorophenyl)-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— (11R)-11-(4-tert-butylphenyl)-10,10-dioxo-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one —— C26H23NO3S
(11R)-11-(4-tert-butylphenyl)-10,10-dioxo-5,11-dihydroindeno[2,1-c][1,5]benzothiazepin-12-one
—— 3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2-hydroxyethyl)benzamide —— C33H35ClN4O4S
3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2-hydroxyethyl)benzamide
—— 3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoic acid —— C31H30ClN3O4S
3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoic acid
—— 3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2,3-dihydroxypropyl)benzamide —— C34H37ClN4O5S
3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2,3-dihydroxypropyl)benzamide
—— 3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2-hydroxy-2-methylpropyl)benzamide —— C35H39ClN4O4S
3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2-hydroxy-2-methylpropyl)benzamide
—— 3-[[3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid —— C34H35ClN4O5S
3-[[3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoyl]amino]propanoic acid
—— 2-[[3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethyl-trimethylazanium —— C36H43ClN5O3S+
2-[[3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethyl-trimethylazanium
—— 3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2-methylsulfonylethyl)benzamide —— C34H37ClN4O5S2
3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]-N-(2-methylsulfonylethyl)benzamide
—— 2-[[3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethanesulfonic acid —— C33H35ClN4O6S2
2-[[3-[[4-[5-[4-(3-chloro-2-methylphenoxy)butanoyl]-3,4-dihydro-2H-1,5-benzothiazepin-9-yl]pyrazol-1-yl]methyl]benzoyl]amino]ethanesulfonic acid