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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2R)-1-(dimethylamino)-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C15H18N2O4S
[(2R)-1-(dimethylamino)-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [(2S)-1-(ethylamino)-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C15H18N2O4S
[(2S)-1-(ethylamino)-1-oxopropan-2-yl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(4-acetamidophenyl)acetate —— C22H24N2O4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(4-acetamidophenyl)acetate
—— 3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C18H17N3O2S2
3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 3-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C18H17N3O2S2
3-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— 2-[[ethyl-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]amino]methyl]-3H-quinazolin-4-one —— C23H26N4O2S
2-[[ethyl-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]amino]methyl]-3H-quinazolin-4-one
—— 4,8-dimethyl-7-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethoxy]chromen-2-one —— C23H23NO4S
4,8-dimethyl-7-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethoxy]chromen-2-one
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(4-methyl-2-nitrophenoxy)ethanone —— C19H20N2O4S
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(4-methyl-2-nitrophenoxy)ethanone
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(4-methyl-2-nitrophenoxy)ethanone —— C19H20N2O4S
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-(4-methyl-2-nitrophenoxy)ethanone
—— [2-[2-(2-methylphenyl)ethylamino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C21H22N2O4S
[2-[2-(2-methylphenyl)ethylamino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(hexylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H24N2O4S
[2-(hexylamino)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[ethyl-[2-(ethylamino)-2-oxoethyl]amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H23N3O5S
[2-[ethyl-[2-(ethylamino)-2-oxoethyl]amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[methyl(thiophen-3-ylmethyl)amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H18N2O4S2
[2-[methyl(thiophen-3-ylmethyl)amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— (6R)-6-(2,3-dimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C21H21NO3S
(6R)-6-(2,3-dimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (6R)-6-(1,3-benzodioxol-5-yl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C20H17NO3S
(6R)-6-(1,3-benzodioxol-5-yl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (6S)-6-(3,4-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C19H15Cl2NOS
(6S)-6-(3,4-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (6R)-6-[4-[(2R)-butan-2-yl]phenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C25H29NOS
(6R)-6-[4-[(2R)-butan-2-yl]phenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]ethanone —— C25H31N3OS
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]ethanone
—— 1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]piperidin-1-ium-4-carboxamide —— C18H26N3O2S+
1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]piperidin-1-ium-4-carboxamide
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-methylsulfanylbenzoate —— C20H21NO3S2
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-methylsulfanylbenzoate
—— [4-(difluoromethoxy)-3-methoxyphenyl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H17F2NO5S
[4-(difluoromethoxy)-3-methoxyphenyl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-phenylcyclopropane-1-carboxylate —— C22H23NO3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-phenylcyclopropane-1-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-cyanobenzoate —— C20H18N2O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-cyanobenzoate
—— 2-methyl-3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]quinazolin-4-one —— C21H21N3O2S
2-methyl-3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]quinazolin-4-one
—— 5,6-dimethyl-2-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-3-oxopyridazine-4-carbonitrile —— C19H20N4O2S
5,6-dimethyl-2-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-3-oxopyridazine-4-carbonitrile
—— 5,6-dimethyl-2-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-3-oxopyridazine-4-carbonitrile —— C19H20N4O2S
5,6-dimethyl-2-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-3-oxopyridazine-4-carbonitrile
—— (5S)-5-(furan-2-yl)-2-methyl-5,11-dihydropyrano[3,4-c][1,5]benzothiazepin-4-one —— C17H13NO3S
(5S)-5-(furan-2-yl)-2-methyl-5,11-dihydropyrano[3,4-c][1,5]benzothiazepin-4-one
—— N-[2-(4-fluoroanilino)-2-oxoethyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide —— C19H18FN3O3S
N-[2-(4-fluoroanilino)-2-oxoethyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-amino-3-methylbenzoate —— C20H22N2O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-amino-3-methylbenzoate
—— 2-(4-methoxyphenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H21NO2S2
2-(4-methoxyphenyl)sulfanyl-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate —— C21H20N4O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(1,2,4-triazol-1-yl)benzoate
—— methyl 5-[2-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C19H22N2O3S
methyl 5-[2-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— 7-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylmethyl)-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H15N3OS2
7-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylmethyl)-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,4-dihydroxybenzoate —— C19H19NO5S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,4-dihydroxybenzoate
—— 2-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C16H20N4OS3
2-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]cinnolin-4-one —— C20H19N3O2S
1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]cinnolin-4-one
—— 2-[(4,5-dimethyl-1,2,4-triazol-3-yl)sulfanyl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C16H20N4OS2
2-[(4,5-dimethyl-1,2,4-triazol-3-yl)sulfanyl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[(4,5-dimethyl-1,2,4-triazol-3-yl)sulfanyl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C16H20N4OS2
2-[(4,5-dimethyl-1,2,4-triazol-3-yl)sulfanyl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 7-methoxy-4-[[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methyl]chromen-2-one —— C21H21NO3S
7-methoxy-4-[[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methyl]chromen-2-one
—— 7-methoxy-4-[[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methyl]chromen-2-one —— C21H21NO3S
7-methoxy-4-[[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methyl]chromen-2-one
—— 2-[2-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylmethyl)-4-oxoquinazolin-3-yl]acetamide —— C20H20N4O2S
2-[2-(3,4-dihydro-2H-1,5-benzothiazepin-5-ylmethyl)-4-oxoquinazolin-3-yl]acetamide
—— [3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H17N3O5S
[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-oxo-2-(thiophene-2-carbonylamino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C17H14N2O5S2
[2-oxo-2-(thiophene-2-carbonylamino)ethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethanone —— C19H19N3O3S2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-(2-methylfuran-3-yl)-1,3,4-oxadiazol-2-yl]sulfanyl]ethanone
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3,5-dimethoxybenzoate —— C21H23NO5S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3,5-dimethoxybenzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-3-(5-nitrofuran-2-yl)prop-2-enoate —— C19H18N2O6S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] (E)-3-(5-nitrofuran-2-yl)prop-2-enoate
—— N-(2-morpholin-4-ylethyl)-3,4-dihydro-2H-1,5-benzothiazepine-5-carbothioamide —— C16H23N3OS2
N-(2-morpholin-4-ylethyl)-3,4-dihydro-2H-1,5-benzothiazepine-5-carbothioamide
—— N-[[(2R)-oxolan-2-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine-5-carbothioamide —— C15H20N2OS2
N-[[(2R)-oxolan-2-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine-5-carbothioamide
—— N-[[(2S)-oxolan-2-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine-5-carbothioamide —— C15H20N2OS2
N-[[(2S)-oxolan-2-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine-5-carbothioamide
—— 2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C20H21NO3S2
2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone