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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(2-chloro-6-fluorophenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H22ClFN2O2S
5-[(2-chloro-6-fluorophenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[3-[(2R,6S)-2,6-dimethylpiperidin-1-yl]propyl]-6-ethyl-8-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H35N3OS
N-[3-[(2R,6S)-2,6-dimethylpiperidin-1-yl]propyl]-6-ethyl-8-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6,8-dimethylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H28N2OS
N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6,8-dimethylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-chloro-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H30ClN3OS
8-chloro-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-chloro-N-[3-[(2R,6R)-2,6-dimethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H30ClN3OS
8-chloro-N-[3-[(2R,6R)-2,6-dimethylpiperidin-1-yl]propyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(methylsulfamoyl)benzoate —— C20H22N2O5S2
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(methylsulfamoyl)benzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-methyl-2-pyridin-2-yl-1,3-thiazole-5-carboxylate —— C22H21N3O3S2
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-methyl-2-pyridin-2-yl-1,3-thiazole-5-carboxylate
—— 2-(2,4-dichloro-6-methylpyridin-3-yl)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H18Cl2N2OS
2-(2,4-dichloro-6-methylpyridin-3-yl)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 4-[(2R)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-1-oxopropan-2-yl]oxybenzonitrile —— C20H20N2O2S
4-[(2R)-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-1-oxopropan-2-yl]oxybenzonitrile
—— (2-methoxy-5-morpholin-4-ylsulfonylphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C22H26N2O5S2
(2-methoxy-5-morpholin-4-ylsulfonylphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [(3S)-1-(1,1-dioxo-1,2-benzothiazol-3-yl)piperidin-3-yl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C23H25N3O3S2
[(3S)-1-(1,1-dioxo-1,2-benzothiazol-3-yl)piperidin-3-yl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 3-(5,7-dimethyl-2-methylsulfanyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]propan-1-one —— C21H25N5OS2
3-(5,7-dimethyl-2-methylsulfanyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]propan-1-one
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C32H30N4O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— 4-methyl-3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-1,3-thiazol-2-one —— C16H18N2O2S2
4-methyl-3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-1,3-thiazol-2-one
—— [(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]methanone —— C23H28N2O3S2
[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]methanone
—— [1,6-di(propan-2-yl)pyrazolo[3,4-b]pyridin-4-yl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C23H28N4OS
[1,6-di(propan-2-yl)pyrazolo[3,4-b]pyridin-4-yl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [4-methoxy-3-[(2S)-2-methylpiperidin-1-yl]sulfonylphenyl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C24H30N2O4S2
[4-methoxy-3-[(2S)-2-methylpiperidin-1-yl]sulfonylphenyl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C32H30N4O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-11-oxo-3-(4-pyridin-2-ylpiperazine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— [4-(1,3-dithiolan-2-yl)phenyl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C20H21NOS3
[4-(1,3-dithiolan-2-yl)phenyl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— N-(3-methylphenyl)-2-[(2S)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C27H28N2O5S
N-(3-methylphenyl)-2-[(2S)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 2-[(2R)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(furan-2-ylmethyl)acetamide —— C24H24N2O5S
2-[(2R)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(furan-2-ylmethyl)acetamide
—— 2-[(2S)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(furan-2-ylmethyl)acetamide —— C24H24N2O5S
2-[(2S)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(furan-2-ylmethyl)acetamide
—— N-(4-chlorophenyl)-2-[(2R)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H23ClN2O4S
N-(4-chlorophenyl)-2-[(2R)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(3-fluorophenyl)-2-[(2S)-2-(4-methoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C24H21FN2O3S
N-(3-fluorophenyl)-2-[(2S)-2-(4-methoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[methyl-[(2-methylphenyl)methyl]amino]ethanone —— C21H26N2OS
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[methyl-[(2-methylphenyl)methyl]amino]ethanone
—— 2-[(3-methoxyphenyl)methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C21H26N2O2S
2-[(3-methoxyphenyl)methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H26N2O2S
2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[(2R)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C24H28N2O3S
2-[(2R)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 2-[(4-ethoxyphenyl)methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C22H28N2O2S
2-[(4-ethoxyphenyl)methyl-methylamino]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (11S)-5-[(2-methylphenyl)methyl]-N-(3-morpholin-4-ylpropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H31N3O4S
(11S)-5-[(2-methylphenyl)methyl]-N-(3-morpholin-4-ylpropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(3-pyrrolidin-1-ylpropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28FN3O3S
(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(3-pyrrolidin-1-ylpropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(3-pyrrolidin-1-ylpropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28FN3O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(3-pyrrolidin-1-ylpropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C26H24FN3O3S
(11R)-5-[(2-fluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-benzyl-N-(3-morpholin-4-ylpropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H29N3O4S
(11R)-5-benzyl-N-(3-morpholin-4-ylpropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-methylphenyl)methyl]-N-(3-morpholin-4-ylpropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H31N3O4S
(11R)-5-[(2-methylphenyl)methyl]-N-(3-morpholin-4-ylpropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(3-butylsulfanylpropyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C23H28N2O3S2
(11R)-N-(3-butylsulfanylpropyl)-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(3-pyrrolidin-1-ylpropyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28ClN3O3S
(11S)-5-[(3-chlorophenyl)methyl]-6,11-dioxo-N-(3-pyrrolidin-1-ylpropyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 1,3-dimethyl-2-sulfanylidene-5-[(2R)-2-(2,3,4-trimethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-1,3-diazinane-4,6-dione —— C24H25N3O5S2
1,3-dimethyl-2-sulfanylidene-5-[(2R)-2-(2,3,4-trimethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-1,3-diazinane-4,6-dione
—— 5-[(2R)-2-(4-hydroxy-3,5-dimethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C23H23N3O5S2
5-[(2R)-2-(4-hydroxy-3,5-dimethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (3S)-1-(3-chlorophenyl)-N-(5-cyclopropyl-6-oxobenzo[b][1,4]benzothiazepin-2-yl)-5-oxopyrrolidine-3-carboxamide —— C27H22ClN3O3S
(3S)-1-(3-chlorophenyl)-N-(5-cyclopropyl-6-oxobenzo[b][1,4]benzothiazepin-2-yl)-5-oxopyrrolidine-3-carboxamide
—— N-benzyl-N-methyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H31N3O4S2
N-benzyl-N-methyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-[(3-methoxyphenyl)methyl]-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H31N3O5S2
N-[(3-methoxyphenyl)methyl]-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-[(4-methoxyphenyl)methyl]-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H31N3O5S2
N-[(4-methoxyphenyl)methyl]-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-[(4-methoxyphenyl)methyl]-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H31N3O5S2
N-[(4-methoxyphenyl)methyl]-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(2-ethyl-6-methylphenyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C26H33N3O4S2
N-(2-ethyl-6-methylphenyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(2-methoxy-5-methylphenyl)-2-[(3R)-3-methyl-4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C24H29N3O5S2
N-(2-methoxy-5-methylphenyl)-2-[(3R)-3-methyl-4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(2-ethyl-6-methylphenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C26H33N3O4S2
N-(2-ethyl-6-methylphenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(2,3-dimethylphenyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H31N3O4S2
N-(2,3-dimethylphenyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(4-chlorophenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C23H26ClN3O4S2
N-(4-chlorophenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(2,4,6-trimethylphenyl)acetamide —— C26H33N3O4S2
2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(2,4,6-trimethylphenyl)acetamide