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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R)-3-methyl-7-(4-propylpiperazin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C17H25N3O3S2
(3R)-3-methyl-7-(4-propylpiperazin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-N-[2-(furan-2-ylmethylsulfanyl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H20N2O4S3
(3S)-N-[2-(furan-2-ylmethylsulfanyl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-[2-[[(2R)-butan-2-yl]-(thiophen-2-ylmethyl)amino]ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H27N3O3S3
N-[2-[[(2R)-butan-2-yl]-(thiophen-2-ylmethyl)amino]ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-2-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O4S2
(2S)-2-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(3,4-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14F2N2O3S2
(3S)-N-(3,4-difluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(4-ethoxyphenyl)-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O4S2
(2S)-N-(4-ethoxyphenyl)-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H18N2O5S2
(2R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-butyl-N-ethyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H24N2O3S2
(3S)-N-butyl-N-ethyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[3-[benzyl(ethyl)amino]propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O3S2
(2S)-N-[3-[benzyl(ethyl)amino]propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H25N3O3S2
(2R)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H25N3O3S2
(3R)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[3-(N-ethylanilino)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O3S2
(2R)-N-[3-(N-ethylanilino)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(3-chloro-4-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17ClN2O4S2
(3S)-N-(3-chloro-4-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[(4-chlorophenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17ClN2O3S2
(3R)-N-[(4-chlorophenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-(3-propan-2-yloxypropyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H24N2O4S2
(3R)-3-methyl-4-oxo-N-(3-propan-2-yloxypropyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-(2,4,6-trimethylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(3R)-3-methyl-4-oxo-N-(2,4,6-trimethylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-N-(2-morpholin-4-ylethyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H23N3O4S2
(3S)-3-methyl-N-(2-morpholin-4-ylethyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-7-[4-(furan-2-carbonyl)piperazin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H21N3O5S2
(2R)-7-[4-(furan-2-carbonyl)piperazin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-N-(4-cyanophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15N3O3S2
(2S)-N-(4-cyanophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-2-methyl-4-oxo-N-(4-sulfamoylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H17N3O5S3
(2R)-2-methyl-4-oxo-N-(4-sulfamoylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-cyclohexyl-N-(furan-2-ylmethyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H26N2O4S2
(2S)-N-cyclohexyl-N-(furan-2-ylmethyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-7-morpholin-4-ylsulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C14H18N2O4S2
(3R)-3-methyl-7-morpholin-4-ylsulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-3-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H16N2O3S2
(3R)-3-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H23N3O4S2
(3R)-3-methyl-4-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[(2-methoxyphenyl)methyl]-2-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C24H31N3O4S2
(2S)-N-[(2-methoxyphenyl)methyl]-2-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(3-bromophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H15BrN2O3S2
(3R)-N-(3-bromophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[2-(furan-2-ylmethylsulfanyl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H20N2O4S3
(3R)-N-[2-(furan-2-ylmethylsulfanyl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-butyl-N-ethyl-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H24N2O3S2
(2S)-N-butyl-N-ethyl-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-2-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H16N2O3S2
(2R)-2-methyl-4-oxo-N-phenyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-7-(4-ethylpiperazin-1-yl)sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C16H23N3O3S2
(3R)-7-(4-ethylpiperazin-1-yl)sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-N-(2,3-dimethylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3S)-N-(2,3-dimethylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(3-chloro-2-methylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17ClN2O3S2
(3S)-N-(3-chloro-2-methylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[(2,5-dimethylphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(2S)-N-[(2,5-dimethylphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(furan-2-ylmethyl)-N,3-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H18N2O4S2
(3R)-N-(furan-2-ylmethyl)-N,3-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-7-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C25H31N3O3S2
(2R)-7-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-2-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2R)-N-(3-cyanophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15N3O3S2
(2R)-N-(3-cyanophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2S)-2-ethyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H20N2O3S3
7-[[(2S)-2-ethyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2S)-2-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H27N3O3S2
(2S)-2-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N,N-diethyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C14H20N2O3S2
(3R)-N,N-diethyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-N-(3-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H18N2O3S2
(3S)-3-methyl-N-(3-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[[5-(azepan-1-ylmethyl)furan-2-yl]methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O4S2
(3S)-N-[[5-(azepan-1-ylmethyl)furan-2-yl]methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2S)-2-ethyl-6-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H22N2O4S2
7-[[(2S)-2-ethyl-6-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2R)-2-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O4S2
(2R)-2-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-ethyl-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C12H16N2O3S2
(2S)-N-ethyl-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-7-(4-cyclopentylpiperazin-1-yl)sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H27N3O3S2
(3S)-7-(4-cyclopentylpiperazin-1-yl)sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2R)-2-methyl-4-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H21N3O5S3
(2R)-2-methyl-4-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[3-(furan-2-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H20N2O4S2
(2R)-N-[3-(furan-2-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[[1-(furan-2-ylmethyl)piperidin-4-yl]methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O4S2
(2S)-N-[[1-(furan-2-ylmethyl)piperidin-4-yl]methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— methyl 3-[N-[[(2R)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate —— C20H22N2O5S2
methyl 3-[N-[[(2R)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate
—— (3S)-N-[2-(azepan-1-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H27N3O3S2
(3S)-N-[2-(azepan-1-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide