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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (4-ethoxy-3-nitrophenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C19H20N2O4S
(4-ethoxy-3-nitrophenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— N-[3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-oxopropyl]-4-nitrobenzamide —— C20H21N3O4S
N-[3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-oxopropyl]-4-nitrobenzamide
—— 2-[4-(1,3-dithiolan-2-yl)phenoxy]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C21H23NO2S3
2-[4-(1,3-dithiolan-2-yl)phenoxy]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (2,5-dimethoxyphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C19H21NO3S
(2,5-dimethoxyphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [4-(1,3-dithian-2-yl)phenyl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C21H23NOS3
[4-(1,3-dithian-2-yl)phenyl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (5-ethoxy-4-methoxy-2-nitrophenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C20H22N2O5S
(5-ethoxy-4-methoxy-2-nitrophenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 2-(3-fluoro-4-methoxyphenyl)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H20FNO2S
2-(3-fluoro-4-methoxyphenyl)-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (2,3-dimethylquinoxalin-6-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C21H21N3OS
(2,3-dimethylquinoxalin-6-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (3,5-dimethyl-1,2-oxazol-4-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C16H18N2O2S
(3,5-dimethyl-1,2-oxazol-4-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 1-[(2R)-2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2,3-dihydro-1,4-benzoxazin-4-yl]ethanone —— C21H22N2O3S
1-[(2R)-2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]-2,3-dihydro-1,4-benzoxazin-4-yl]ethanone
—— [1-(2,3-dihydro-1H-inden-5-ylsulfonyl)piperidin-4-yl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C25H30N2O3S2
[1-(2,3-dihydro-1H-inden-5-ylsulfonyl)piperidin-4-yl]-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (2-fluoro-4-methoxyphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C18H18FNO2S
(2-fluoro-4-methoxyphenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— N-cyclopropyl-3-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]benzenesulfonamide —— C20H22N2O3S2
N-cyclopropyl-3-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]benzenesulfonamide
—— 3-ethyl-1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]quinazoline-2,4-dione —— C22H23N3O3S
3-ethyl-1-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]quinazoline-2,4-dione
—— 2-methyl-6-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyridazin-3-one —— C16H17N3O2S
2-methyl-6-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]pyridazin-3-one
—— (7-fluoro-3-methyl-1-benzofuran-2-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C20H18FNO2S
(7-fluoro-3-methyl-1-benzofuran-2-yl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (4-methoxy-1-phenylpyrazol-3-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C21H21N3O2S
(4-methoxy-1-phenylpyrazol-3-yl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— (4-ethoxy-3-nitrophenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C19H20N2O4S
(4-ethoxy-3-nitrophenyl)-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-1,3-thiazolidin-2-one —— C15H18N2O2S2
3-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-1,3-thiazolidin-2-one
—— 2-(furan-2-ylmethyl)-5-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]isoindole-1,3-dione —— C24H20N2O4S
2-(furan-2-ylmethyl)-5-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-5-carbonyl]isoindole-1,3-dione
—— 3-[3-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-oxopropyl]-5-thiophen-2-yl-1,3,4-oxadiazol-2-one —— C19H19N3O3S2
3-[3-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-oxopropyl]-5-thiophen-2-yl-1,3,4-oxadiazol-2-one
—— (3,5-difluorophenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C17H15F2NOS
(3,5-difluorophenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— 2,4-dimethyl-5-[3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-oxopropyl]-1H-pyrimidin-6-one —— C19H23N3O2S
2,4-dimethyl-5-[3-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-3-oxopropyl]-1H-pyrimidin-6-one
—— (2-chloro-5-methylsulfonylphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C18H18ClNO3S2
(2-chloro-5-methylsulfonylphenyl)-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [6-cyclopropyl-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazolo[3,4-b]pyridin-4-yl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C25H28N4O3S2
[6-cyclopropyl-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazolo[3,4-b]pyridin-4-yl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— [(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[5-(4-nitrophenyl)furan-2-yl]methanone —— C21H18N2O4S
[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-[5-(4-nitrophenyl)furan-2-yl]methanone
—— [6-cyclopropyl-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazolo[3,4-b]pyridin-4-yl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone —— C25H28N4O3S2
[6-cyclopropyl-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazolo[3,4-b]pyridin-4-yl]-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]methanone
—— N-(3-(2-(3,4,5-trimethoxyphenyl)-2,3-dihydrobenzo[b][1,4]thiazepin-4-yl)phenyl)acetamide —— C26H26N2O4S
N-(3-(2-(3,4,5-trimethoxyphenyl)-2,3-dihydrobenzo[b][1,4]thiazepin-4-yl)phenyl)acetamide
—— 4-[2-(1H-indol-3-yl)ethyl]-N-(4-methoxyphenyl)-3-methyl-5-oxo-2,3,4,5-tetrahydro-1,4-benzothiazepine-3-carboxamide —— C28H27N3O3S
4-[2-(1H-indol-3-yl)ethyl]-N-(4-methoxyphenyl)-3-methyl-5-oxo-2,3,4,5-tetrahydro-1,4-benzothiazepine-3-carboxamide
—— N-(2-benzoylphenyl)-10-(3-chlorobenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide —— C34H23ClN2O4S
N-(2-benzoylphenyl)-10-(3-chlorobenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetate —— C22H22N2O5S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2R)-3-oxo-4H-1,4-benzoxazin-2-yl]acetate —— C22H22N2O5S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2R)-3-oxo-4H-1,4-benzoxazin-2-yl]acetate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetate —— C22H22N2O5S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2S)-3-oxo-4H-1,4-benzoxazin-2-yl]acetate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-ethyl-5-methyl-1,2-oxazole-4-carboxylate —— C19H22N2O4S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-ethyl-5-methyl-1,2-oxazole-4-carboxylate
—— [(5S,7R)-3-chloro-1-adamantyl]-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)methanone —— C20H24ClNOS
[(5S,7R)-3-chloro-1-adamantyl]-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)methanone
—— 3-hydroxy-8-methoxy-4-(4-methoxyphenyl)-4,5-dihydro-1,5-benzothiazepin-2(3H)-one —— C17H17NO4S
3-hydroxy-8-methoxy-4-(4-methoxyphenyl)-4,5-dihydro-1,5-benzothiazepin-2(3H)-one
—— ethyl 5-methyl-3-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-4-oxothieno[2,3-d]pyrimidine-6-carboxylate —— C22H23N3O4S2
ethyl 5-methyl-3-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-4-oxothieno[2,3-d]pyrimidine-6-carboxylate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate —— C22H22N4O3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate —— C22H22N4O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 5-methyl-2-phenyltriazole-4-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-bromo-5-sulfamoylbenzoate —— C19H19BrN2O5S2
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-bromo-5-sulfamoylbenzoate
—— 2-[[5-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C25H26N4O3S2
2-[[5-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(benzylamino)-1,3-thiazole-4-carboxylate —— C23H23N3O3S2
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(benzylamino)-1,3-thiazole-4-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(benzylamino)-1,3-thiazole-4-carboxylate —— C23H23N3O3S2
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(benzylamino)-1,3-thiazole-4-carboxylate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-chloro-5-(dimethylsulfamoyl)benzoate —— C21H23ClN2O5S2
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-chloro-5-(dimethylsulfamoyl)benzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-chloro-5-(dimethylsulfamoyl)benzoate —— C21H23ClN2O5S2
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-chloro-5-(dimethylsulfamoyl)benzoate
—— 2-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]sulfanyl-3-(3-methylpyridin-2-yl)quinazolin-4-one —— C26H24N4O2S2
2-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]sulfanyl-3-(3-methylpyridin-2-yl)quinazolin-4-one
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-acetamido-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H26N2O4S2
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-acetamido-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— 2-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]sulfanyl-3-(3-methylpyridin-2-yl)quinazolin-4-one —— C26H24N4O2S2
2-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]sulfanyl-3-(3-methylpyridin-2-yl)quinazolin-4-one
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(1,3-benzothiazol-2-yl)butanoate —— C23H24N2O3S2
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(1,3-benzothiazol-2-yl)butanoate
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-[(3-methylphenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C25H28N4O2S2
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-[(3-methylphenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone