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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O4S
5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O4S
5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O4S
5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O2S
N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O2S
N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O2S
N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H28N2O2S
N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H28N2O2S
N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O2S
5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O2S
5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3S)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O2S
5-[(3-chlorophenyl)methyl]-N-[(1S,2S,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29ClN2O2S
5-[(3-chlorophenyl)methyl]-N-[(1R,2S,3R)-2,3-dimethylcyclohexyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (1S,10R)-1-methyl-17-oxa-9-thia-2-azatetracyclo[8.7.1.03,8.011,16]octadeca-3,5,7,11,13,15-hexaene —— C16H15NOS
(1S,10R)-1-methyl-17-oxa-9-thia-2-azatetracyclo[8.7.1.03,8.011,16]octadeca-3,5,7,11,13,15-hexaene
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(2-amino-2-oxoethoxy)benzoate —— C21H22N2O5S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(2-amino-2-oxoethoxy)benzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-chloro-2-fluorobenzoate —— C19H17ClFNO3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-chloro-2-fluorobenzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,3-dimethylquinoxaline-6-carboxylate —— C23H23N3O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2,3-dimethylquinoxaline-6-carboxylate
—— 1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S,2S,3S)-2,3-dimethylcyclohexyl]urea —— C29H31N3O2S
1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S,2S,3S)-2,3-dimethylcyclohexyl]urea
—— 1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S,2S,3R)-2,3-dimethylcyclohexyl]urea —— C29H31N3O2S
1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S,2S,3R)-2,3-dimethylcyclohexyl]urea
—— 1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1R,2S,3S)-2,3-dimethylcyclohexyl]urea —— C29H31N3O2S
1-(5-benzyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1R,2S,3S)-2,3-dimethylcyclohexyl]urea
—— [(1R)-2-(cyclopropylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C21H20N2O4S
[(1R)-2-(cyclopropylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [(1R)-2-(diethylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C22H24N2O4S
[(1R)-2-(diethylamino)-2-oxo-1-phenylethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— (11R)-5-[(4-chlorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-N-[(1S,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-N-[3-[(3R,5S)-3,5-dimethylpiperidin-1-yl]propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H34FN3O3S
(11R)-N-[3-[(3R,5S)-3,5-dimethylpiperidin-1-yl]propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-N-[(1R,2S)-2-methylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H34FN3O3S
(11R)-N-[3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27FN2O3S
(11R)-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27FN2O3S
(11R)-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— [2-[methyl-(4-methylcyclohexyl)amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H26N2O4S
[2-[methyl-(4-methylcyclohexyl)amino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(2-fluorophenyl)methyl-methylamino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C20H19FN2O4S
[2-[(2-fluorophenyl)methyl-methylamino]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C21H26N2O4S
[2-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-1-yl]-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-(azocan-1-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C19H24N2O4S
[2-(azocan-1-yl)-2-oxoethyl] 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [5-(furan-2-yl)-1,2-oxazol-3-yl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate —— C18H14N2O5S
[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl 4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxylate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(5-methylpyrazol-1-yl)benzoate —— C23H23N3O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(5-methylpyrazol-1-yl)benzoate
—— (6R)-9,9-dimethyl-6-(4-methylsulfanylphenyl)-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C22H23NOS2
(6R)-9,9-dimethyl-6-(4-methylsulfanylphenyl)-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (6S)-6-[4-[(2S)-butan-2-yl]phenyl]-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C23H25NOS
(6S)-6-[4-[(2S)-butan-2-yl]phenyl]-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (6S)-6-[4-[(2R)-butan-2-yl]phenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C25H29NOS
(6S)-6-[4-[(2R)-butan-2-yl]phenyl]-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (6S)-6-(1,3-benzodioxol-5-yl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C20H17NO3S
(6S)-6-(1,3-benzodioxol-5-yl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (6R)-6-(3-methoxy-4-propoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C25H29NO3S
(6R)-6-(3-methoxy-4-propoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (6R)-6-(2,4-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C19H15Cl2NOS
(6R)-6-(2,4-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]ethanone —— C25H31N3OS
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]ethanone
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-hydroxy-4-methoxybenzoate —— C20H21NO5S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-hydroxy-4-methoxybenzoate
—— 5-[2-(4-bromophenyl)sulfonylethyl]-3,4-dihydro-2H-1,5-benzothiazepine —— C17H18BrNO2S2
5-[2-(4-bromophenyl)sulfonylethyl]-3,4-dihydro-2H-1,5-benzothiazepine
—— (2S)-N-methyl-4-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H25N3O3S
(2S)-N-methyl-4-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N-methyl-N-[2-(2-methylsulfanylanilino)-2-oxoethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide —— C20H21N3O3S2
N-methyl-N-[2-(2-methylsulfanylanilino)-2-oxoethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide
—— 2-(4-methoxyphenyl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C19H21NO2S2
2-(4-methoxyphenyl)sulfanyl-1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— N-[2-(2,5-dimethylanilino)-2-oxoethyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide —— C21H23N3O3S
N-[2-(2,5-dimethylanilino)-2-oxoethyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide