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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(4-chlorophenyl)methyl]-6,11,11-trioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23ClN2O4S
5-[(4-chlorophenyl)methyl]-6,11,11-trioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H24N2O4S
(11S)-5-[(2,5-dimethylphenyl)methyl]-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C25H21FN2O4S
(11S)-5-[(4-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C34H33N3O4S
(11S)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2-fluorophenyl)methyl]-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H19FN2O4S
(11S)-5-[(2-fluorophenyl)methyl]-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C26H23FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O3S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[2-(cyclohexen-1-yl)ethyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H27FN2O3S
(11R)-N-[2-(cyclohexen-1-yl)ethyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(4-ethylpiperazine-1-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H26FN3O3S
(11S)-3-(4-ethylpiperazine-1-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-benzyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O5S
(11S)-5-benzyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C25H21FN2O4S
(11R)-5-[(4-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— 5-[(4-fluorophenyl)methyl]-3-[(2S)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O4S
5-[(4-fluorophenyl)methyl]-3-[(2S)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-3-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C32H27ClFN3O3S
(11R)-3-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— [(2S)-oxolan-2-yl]methyl 5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C28H27NO6S
[(2S)-oxolan-2-yl]methyl 5-[(2,5-dimethylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— ethyl 4-[[(11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate —— C29H28ClN3O5S
ethyl 4-[[(11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate
—— (11S)-N-benzyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H26N2O3S
(11S)-N-benzyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H26N2O4S
(11R)-5-[(2,5-dimethylphenyl)methyl]-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— 5-[(2-fluorophenyl)methyl]-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H32FN3O4S
5-[(2-fluorophenyl)methyl]-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-3-(4-benzylpiperidine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C33H30N2O3S
(11S)-5-benzyl-3-(4-benzylpiperidine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-N-[(4-chlorophenyl)methyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H20ClFN2O3S
(11R)-N-[(4-chlorophenyl)methyl]-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— [(2R)-oxolan-2-yl]methyl 5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H22FNO6S
[(2R)-oxolan-2-yl]methyl 5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— ethyl (3R)-1-[(11S)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate —— C29H28N2O5S
ethyl (3R)-1-[(11S)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate
—— 5-benzyl-N-[(2S)-butan-2-yl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2O4S
5-benzyl-N-[(2S)-butan-2-yl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-[4-(3-chlorophenyl)piperazine-1-carbonyl]-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C33H30ClN3O3S
(11R)-3-[4-(3-chlorophenyl)piperazine-1-carbonyl]-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-(1,3-benzodioxol-5-ylmethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H21FN2O5S
(11S)-N-(1,3-benzodioxol-5-ylmethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[2-(3,4-dimethoxyphenyl)ethyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C33H32N2O5S
(11S)-N-[2-(3,4-dimethoxyphenyl)ethyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— [(2R)-oxolan-2-yl]methyl 5-benzyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H23NO6S
[(2R)-oxolan-2-yl]methyl 5-benzyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— (11S)-5-benzyl-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H24N2O3S
(11S)-5-benzyl-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-cyclohexyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H25ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-cyclohexyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C33H30FN3O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-ethyl-N-[(2-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H22N2O4S
(11R)-5-ethyl-N-[(2-methoxyphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-3-(4-ethylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H27N3O3S
(11S)-5-benzyl-3-(4-ethylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— ethyl (3R)-1-[(11R)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate —— C29H28N2O5S
ethyl (3R)-1-[(11R)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C34H33N3O4S
(11R)-5-[(2,5-dimethylphenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-benzyl-N-(4-methylcyclohexyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28N2O3S
(11R)-5-benzyl-N-(4-methylcyclohexyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-5-[(3-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C32H37N3O4S
N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-5-[(3-methylphenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl 4-[[(11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate —— C29H28ClN3O5S
ethyl 4-[[(11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate
—— (11S)-5-[(2-fluorophenyl)methyl]-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl (3R)-1-[(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate —— C29H27FN2O5S
ethyl (3R)-1-[(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperidine-3-carboxylate
—— 5-[(4-chlorophenyl)methyl]-N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H34ClN3O4S
5-[(4-chlorophenyl)methyl]-N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl 4-[[(11R)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate —— C29H29N3O5S
ethyl 4-[[(11R)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]amino]piperidine-1-carboxylate
—— (11S)-5-[(4-fluorophenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C32H28FN3O4S
(11S)-5-[(4-fluorophenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H25ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-[2-(cyclohexen-1-yl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H27ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-[2-(cyclohexen-1-yl)ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-(3-ethylphenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23ClN2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-(3-ethylphenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(3-chlorophenyl)methyl]-N-(3,5-dichlorophenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H17Cl3N2O3S
(11S)-5-[(3-chlorophenyl)methyl]-N-(3,5-dichlorophenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[(2S)-butan-2-yl]-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11S)-N-[(2S)-butan-2-yl]-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[(2R)-butan-2-yl]-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11R)-N-[(2R)-butan-2-yl]-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25ClN2O3S
(11R)-5-[(3-chlorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-(4-methylcyclohexyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H30N2O3S
(11S)-N-(4-methylcyclohexyl)-5-[(2-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide