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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C23H28N4O2S
N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— 2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C24H23N3O2S
2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C23H28N4O2S
N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— 2-phenyl-5-propyl-2,3-dihydro-1,5-benzothiazepin-4(5H)-one —— C18H19NOS
2-phenyl-5-propyl-2,3-dihydro-1,5-benzothiazepin-4(5H)-one
—— 2-(4-Methoxyphenyl)-5-propyl-2,3-dihydro-1,5-benzothiazepin-4-one —— C19H21NO2S
2-(4-Methoxyphenyl)-5-propyl-2,3-dihydro-1,5-benzothiazepin-4-one
—— 5-ethyl-2-phenyl-2,3-dihydrobenzo[b][1,4]thiazepin-4(5H)-one —— C17H17NOS
5-ethyl-2-phenyl-2,3-dihydrobenzo[b][1,4]thiazepin-4(5H)-one
—— N-methyl-N-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H25N3O4S2
N-methyl-N-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-methyl-N-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H25N3O4S2
N-methyl-N-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 4-(1,3-Benzothiazol-2-yl)-2-(4-methoxyphenyl)-2,5-dihydro-1,5-benzothiazepine —— C23H18N2OS2
4-(1,3-Benzothiazol-2-yl)-2-(4-methoxyphenyl)-2,5-dihydro-1,5-benzothiazepine
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]urea —— C26H25N3O2S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]urea
—— 1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]urea —— C26H25N3O2S
1-(5-ethyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)-3-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]urea
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(4-fluorophenyl)imidazole-4-carboxylate —— C22H20FN3O3S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(4-fluorophenyl)imidazole-4-carboxylate
—— (2S)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-2-phenoxypropanamide —— C25H24N2O4S
(2S)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-2-phenoxypropanamide
—— (2R)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-2-phenoxypropanamide —— C25H24N2O4S
(2R)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-2-phenoxypropanamide
—— (3S)-1-(3,4-dimethylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide —— C29H29N3O3S
(3S)-1-(3,4-dimethylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide
—— N-[(2R)-3-methyl-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]butan-2-yl]furan-2-carboxamide —— C26H27N3O4S
N-[(2R)-3-methyl-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]butan-2-yl]furan-2-carboxamide
—— (3R)-1-(3,4-dimethylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide —— C29H29N3O3S
(3R)-1-(3,4-dimethylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide
—— (3S)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)-1-phenylpyrrolidine-3-carboxamide —— C27H25N3O3S
(3S)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)-1-phenylpyrrolidine-3-carboxamide
—— N-[(2S)-3-methyl-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]butan-2-yl]furan-2-carboxamide —— C26H27N3O4S
N-[(2S)-3-methyl-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]butan-2-yl]furan-2-carboxamide
—— N-[(2R)-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]propan-2-yl]benzamide —— C26H25N3O3S
N-[(2R)-1-oxo-1-[(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)amino]propan-2-yl]benzamide
—— (3S)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-5-oxo-1-phenylpyrrolidine-3-carboxamide —— C27H25N3O4S
(3S)-N-[5-(2-methoxyethyl)-6-oxobenzo[b][1,4]benzothiazepin-2-yl]-5-oxo-1-phenylpyrrolidine-3-carboxamide
—— (3S)-1-(4-methylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide —— C28H27N3O3S
(3S)-1-(4-methylphenyl)-5-oxo-N-(6-oxo-5-propan-2-ylbenzo[b][1,4]benzothiazepin-2-yl)pyrrolidine-3-carboxamide
—— N-[[(2S)-1,4-dioxan-2-yl]methyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C19H19N3O4S
N-[[(2S)-1,4-dioxan-2-yl]methyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— N-[[(2R)-1,4-dioxan-2-yl]methyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C19H19N3O4S
N-[[(2R)-1,4-dioxan-2-yl]methyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— N-[(2R)-1-(furan-2-yl)propan-2-yl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C21H19N3O3S
N-[(2R)-1-(furan-2-yl)propan-2-yl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— N-[(2S)-1-(furan-2-yl)propan-2-yl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C21H19N3O3S
N-[(2S)-1-(furan-2-yl)propan-2-yl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— 1-[7-[(3R)-3-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C26H33N3O3S2
1-[7-[(3R)-3-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 5-[(4-Methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylic acid —— C22H17NO3S2
5-[(4-Methylsulfanylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylic acid
—— 10-(3-Chlorobenzyl)-11-oxo-N-(2-thienylmethyl)-10,11-dihydrodibenzo[B,F][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C26H19ClN2O4S2
10-(3-Chlorobenzyl)-11-oxo-N-(2-thienylmethyl)-10,11-dihydrodibenzo[B,F][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 10-(3-chlorobenzyl)-N-(4-methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C29H23ClN2O5S
10-(3-chlorobenzyl)-N-(4-methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 10-(3-Chlorobenzyl)-11-oxo-N-(1,2,3,4-tetrahydro-1-naphthalenyl)-10,11-dihydrodibenzo[B,F][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C31H25ClN2O4S
10-(3-Chlorobenzyl)-11-oxo-N-(1,2,3,4-tetrahydro-1-naphthalenyl)-10,11-dihydrodibenzo[B,F][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— N-butyl-10-(3-chlorobenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C25H23ClN2O4S
N-butyl-10-(3-chlorobenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— N-(2-chlorobenzyl)-10-(3-chlorobenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C28H20Cl2N2O4S
N-(2-chlorobenzyl)-10-(3-chlorobenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 10-(3-chlorobenzyl)-N-cyclopropyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C24H19ClN2O4S
10-(3-chlorobenzyl)-N-cyclopropyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 5-[(3-Chlorophenyl)methyl]-3-(4-cyclohexylpiperazin-4-ium-1-carbonyl)-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C31H33ClN3O4S+
5-[(3-Chlorophenyl)methyl]-3-(4-cyclohexylpiperazin-4-ium-1-carbonyl)-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— 10-(3-chlorobenzyl)-N-cyclohexyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C27H25ClN2O4S
10-(3-chlorobenzyl)-N-cyclohexyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 5-[(3-chlorophenyl)methyl]-6,11,11-trioxo-N-(2-pyrrolidin-1-ium-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27ClN3O4S+
5-[(3-chlorophenyl)methyl]-6,11,11-trioxo-N-(2-pyrrolidin-1-ium-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 10-(3-Chlorobenzyl)-8-[(4-cyclohexyl-1-piperazinyl)carbonyl]dibenzo[B,F][1,4]thiazepin-11(10H)-one 5,5-dioxide —— C31H32ClN3O4S
10-(3-Chlorobenzyl)-8-[(4-cyclohexyl-1-piperazinyl)carbonyl]dibenzo[B,F][1,4]thiazepin-11(10H)-one 5,5-dioxide
—— 10-(3-chlorobenzyl)-N-cyclopentyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C26H23ClN2O4S
10-(3-chlorobenzyl)-N-cyclopentyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— N-benzyl-10-(3-chlorobenzyl)-N-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C29H23ClN2O4S
N-benzyl-10-(3-chlorobenzyl)-N-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 10-(3-Chlorobenzyl)-11-oxo-N-[2-(1-pyrrolidinyl)ethyl]-10,11-dihydrodibenzo[B,F][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C27H26ClN3O4S
10-(3-Chlorobenzyl)-11-oxo-N-[2-(1-pyrrolidinyl)ethyl]-10,11-dihydrodibenzo[B,F][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 10-(3-chlorobenzyl)-N-[3-(diisobutylamino)propyl]-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C32H38ClN3O4S
10-(3-chlorobenzyl)-N-[3-(diisobutylamino)propyl]-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— 3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1R)-1-phenylethyl]propanamide —— C23H21N3O2S
3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1R)-1-phenylethyl]propanamide
—— N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide —— C25H23N3O4S
N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide
—— 3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1S)-1-phenylethyl]propanamide —— C23H21N3O2S
3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)-N-[(1S)-1-phenylethyl]propanamide
—— N-[(2R)-butan-2-yl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide —— C19H21N3O2S
N-[(2R)-butan-2-yl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide
—— N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide —— C25H23N3O4S
N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide
—— N-[(2S)-butan-2-yl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide —— C19H21N3O2S
N-[(2S)-butan-2-yl]-3-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)propanamide
—— ethyl 5-[4-methoxy-3-[[(3R)-3-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]phenyl]-1,2-oxazole-3-carboxylate —— C23H24N2O6S2
ethyl 5-[4-methoxy-3-[[(3R)-3-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]phenyl]-1,2-oxazole-3-carboxylate
—— (3R)-N-(2,5-dimethylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3R)-N-(2,5-dimethylphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide