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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-[(3-methylphenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone —— C25H28N4O2S2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-[[5-[(3-methylphenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethanone
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-(phenylcarbamoyl)piperidine-4-carboxylate —— C25H29N3O4S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-(phenylcarbamoyl)piperidine-4-carboxylate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-(phenylcarbamoyl)piperidine-4-carboxylate —— C25H29N3O4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 1-(phenylcarbamoyl)piperidine-4-carboxylate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-chloro-3-(methylsulfamoyl)benzoate —— C20H21ClN2O5S2
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-chloro-3-(methylsulfamoyl)benzoate
—— [2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(2-methoxyphenoxy)propanoate —— C22H25NO5S
[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(2-methoxyphenoxy)propanoate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(2-methoxyphenoxy)propanoate —— C22H25NO5S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 3-(2-methoxyphenoxy)propanoate
—— (3aS,7aS)-2-[2-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)-2-oxoethyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione —— C19H22N2O3S
(3aS,7aS)-2-[2-(3,4-dihydro-2H-1,5-benzothiazepin-5-yl)-2-oxoethyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione
—— 2-[4-(2-hydroxyethyl)piperazin-1-yl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H27N3O2S
2-[4-(2-hydroxyethyl)piperazin-1-yl]-1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (3S)-N-[4-[(4-ethylpiperazin-1-yl)methyl]phenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C23H30N4O3S2
(3S)-N-[4-[(4-ethylpiperazin-1-yl)methyl]phenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[4-[(4-ethylpiperazin-1-yl)methyl]phenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C23H30N4O3S2
(3R)-N-[4-[(4-ethylpiperazin-1-yl)methyl]phenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[3-(4-benzylpiperazin-1-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C24H32N4O3S2
(2R)-N-[3-(4-benzylpiperazin-1-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[3-(4-benzylpiperazin-1-yl)propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C24H32N4O3S2
(3R)-N-[3-(4-benzylpiperazin-1-yl)propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H28N4O3S2
(3S)-3-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H28N4O3S2
(3R)-3-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 1-(3,5-dimethylphenyl)-5-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]pyrazolo[3,4-d]pyrimidin-4-one —— C25H25N5O2S
1-(3,5-dimethylphenyl)-5-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]pyrazolo[3,4-d]pyrimidin-4-one
—— 7-[[4-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C23H27N5O2S2
7-[[4-[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 2-[2-(2,3-Dimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-4-yl]phenol —— C23H21NO3S
2-[2-(2,3-Dimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-4-yl]phenol
—— N-[(4-fluorophenyl)methyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide —— C21H15FN2O2S
N-[(4-fluorophenyl)methyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-{[4-(3-Chlorophenyl)piperazino]carbonyl}dibenzo[B,F][1,4]thiazepin-11(10H)-one —— C24H20ClN3O2S
8-{[4-(3-Chlorophenyl)piperazino]carbonyl}dibenzo[B,F][1,4]thiazepin-11(10H)-one
—— N-(1,3-benzodioxol-5-ylmethyl)-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide —— C22H16N2O4S
N-(1,3-benzodioxol-5-ylmethyl)-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-(2-methylcyclohexyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C21H22N2O2S
N-(2-methylcyclohexyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— 8-{[4-(2,3-Dimethylphenyl)piperazino]carbonyl}dibenzo[B,F][1,4]thiazepin-11(10H)-one —— C26H25N3O2S
8-{[4-(2,3-Dimethylphenyl)piperazino]carbonyl}dibenzo[B,F][1,4]thiazepin-11(10H)-one
—— 8-{[3-Methyl-4-(4-methylphenyl)piperazino]carbonyl}dibenzo[B,F][1,4]thiazepin-11(10H)-one —— C26H25N3O2S
8-{[3-Methyl-4-(4-methylphenyl)piperazino]carbonyl}dibenzo[B,F][1,4]thiazepin-11(10H)-one
—— N-hexyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C20H22N2O2S
N-hexyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— 3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-5H-benzo[b][1,4]benzothiazepin-6-one —— C25H23N3O3S
3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-5H-benzo[b][1,4]benzothiazepin-6-one
—— 4-(Furan-2-yl)-2-(4-methylphenyl)-2,3-dihydro-1,5-benzothiazepine —— C20H17NOS
4-(Furan-2-yl)-2-(4-methylphenyl)-2,3-dihydro-1,5-benzothiazepine
—— 2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C22H31N3O5S2
2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C22H31N3O5S2
2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-(3-fluorophenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C23H26FN3O4S2
N-(3-fluorophenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C22H31N3O5S2
2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-cyclohexyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C23H33N3O4S2
N-cyclohexyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-methyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide —— C24H29N3O4S2
N-methyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide
—— 2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(2-methylphenyl)acetamide —— C24H29N3O4S2
2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(2-methylphenyl)acetamide
—— N-(3-fluorophenyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C23H26FN3O4S2
N-(3-fluorophenyl)-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— [(2S)-oxolan-2-yl]methyl 5-[(4-cyanophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C27H22N2O4S
[(2S)-oxolan-2-yl]methyl 5-[(4-cyanophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— N-[[(2R)-oxolan-2-yl]methyl]-2-(4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl)acetamide —— C20H27N3O5S2
N-[[(2R)-oxolan-2-yl]methyl]-2-(4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl)acetamide
—— 2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C22H31N3O5S2
2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— ethyl 5-[(2R)-1-(2-chloroanilino)-1-oxopropan-2-yl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C25H21ClN2O4S
ethyl 5-[(2R)-1-(2-chloroanilino)-1-oxopropan-2-yl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— 2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide —— C23H27N3O4S2
2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide
—— 2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide —— C23H27N3O4S2
2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide
—— N-cyclohexyl-N-methyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C24H35N3O4S2
N-cyclohexyl-N-methyl-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-cyclohexyl-N-methyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C24H35N3O4S2
N-cyclohexyl-N-methyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-cyclohexyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C23H33N3O4S2
N-cyclohexyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-methyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide —— C24H29N3O4S2
N-methyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide
—— [(2R)-oxolan-2-yl]methyl 6-oxo-5-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxylate —— C25H22N2O4S
[(2R)-oxolan-2-yl]methyl 6-oxo-5-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxylate
—— [(2S)-oxolan-2-yl]methyl 5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H22FNO4S
[(2S)-oxolan-2-yl]methyl 5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— [(2R)-oxolan-2-yl]methyl 5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H22FNO4S
[(2R)-oxolan-2-yl]methyl 5-[(4-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— [(2S)-oxolan-2-yl]methyl 5-[(3-chlorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H22ClNO4S
[(2S)-oxolan-2-yl]methyl 5-[(3-chlorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— [(2R)-oxolan-2-yl]methyl 5-[(4-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C27H25NO5S
[(2R)-oxolan-2-yl]methyl 5-[(4-methoxyphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— [(2R)-oxolan-2-yl]methyl 5-[2-(furan-2-ylmethylamino)-2-oxoethyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H24N2O6S
[(2R)-oxolan-2-yl]methyl 5-[2-(furan-2-ylmethylamino)-2-oxoethyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate