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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-methylphenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C29H30N2O4S
3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-methylphenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-(2,2-dimethoxyethyl)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O5S
(11S)-N-(2,2-dimethoxyethyl)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2,5-dimethylphenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C30H32N2O4S
5-[(2,5-dimethylphenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[(2-chlorophenyl)methyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C23H19ClN2O3S
(11R)-N-[(2-chlorophenyl)methyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28N2O4S
(11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-(2,2-dimethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2O5S
(11S)-5-benzyl-N-(2,2-dimethoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-N-(3-methoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O4S
(11R)-5-[(2,5-dimethylphenyl)methyl]-N-(3-methoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(2,2-diethoxyethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H27FN2O5S
(11R)-N-(2,2-diethoxyethyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C30H23FN2O3S
(11R)-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-chlorophenyl)methyl]-N-cyclopropyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H19ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-cyclopropyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-N-(2,2-dimethoxyethyl)-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25ClN2O5S
(11R)-5-[(4-chlorophenyl)methyl]-N-(2,2-dimethoxyethyl)-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(4-benzylpiperidine-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H28N2O3S
(11S)-3-(4-benzylpiperidine-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H27FN2O3S
(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(2,3-dihydroindole-1-carbonyl)-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H21FN2O3S
(11S)-3-(2,3-dihydroindole-1-carbonyl)-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-benzyl-N-[3-[cyclohexyl(methyl)amino]propyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H35N3O3S
(11S)-5-benzyl-N-[3-[cyclohexyl(methyl)amino]propyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-N-cycloheptyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-N-cycloheptyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O4S
N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O4S
N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C26H24N2O3S
(11S)-5-benzyl-11-oxo-3-(piperidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— 5-[(4-chlorophenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O4S
5-[(4-chlorophenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(2,5-dimethylphenyl)methyl]-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C27H26N2O3S
(11R)-5-[(2,5-dimethylphenyl)methyl]-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-[3-(azepan-1-yl)propyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H31N3O3S
(11S)-N-[3-(azepan-1-yl)propyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2,5-dimethylphenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C30H32N2O4S
5-[(2,5-dimethylphenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-3-(azepane-1-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H30N2O3S
(11S)-3-(azepane-1-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-phenylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11S)-5-benzyl-N-(3-methylbutyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C25H21FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C30H32N2O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-benzyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C25H22N2O3S
(11R)-5-benzyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-ethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H29N3O3S
(11R)-5-ethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O3S
(11S)-5-[(4-fluorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-(2,2-dimethoxyethyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23FN2O5S
(11S)-N-(2,2-dimethoxyethyl)-5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl 4-[(11R)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperazine-1-carboxylate —— C28H27N3O5S
ethyl 4-[(11R)-5-benzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carbonyl]piperazine-1-carboxylate
—— (11S)-N-benzyl-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H21ClN2O3S
(11S)-N-benzyl-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2,5-dimethylphenyl)methyl]-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C30H32N2O4S
5-[(2,5-dimethylphenyl)methyl]-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H29FN2O4S
N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-5-[(2-fluorophenyl)methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-cyclopentyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28N2O3S
(11R)-N-cyclopentyl-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O3S
(11S)-5-benzyl-6,11-dioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[3-(diethylamino)propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H30FN3O3S
(11S)-N-[3-(diethylamino)propyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-N-(2-morpholin-4-ylethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H26FN3O4S
(11R)-5-[(2-fluorophenyl)methyl]-N-(2-morpholin-4-ylethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C30H24N2O3S
(11S)-5-benzyl-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-3-(2,3-dihydroindole-1-carbonyl)-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C29H21FN2O3S
(11R)-3-(2,3-dihydroindole-1-carbonyl)-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21FN2O4S
(11R)-5-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N,5-dibenzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H22N2O3S
(11S)-N,5-dibenzyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-ethyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H29N3O4S
5-ethyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-benzyl-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H29N3O4S
5-benzyl-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-benzyl-6,11,11-trioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O4S
5-benzyl-6,11,11-trioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[2-(dipropylamino)ethyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H32FN3O3S
(11S)-N-[2-(dipropylamino)ethyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23FN2O4S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide