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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11R)-N-(3-butylsulfanylpropyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H29FN2O3S2
(11R)-N-(3-butylsulfanylpropyl)-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C25H22N2O4S
(11R)-5-benzyl-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-benzyl-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O4S
(11S)-5-benzyl-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[3-(diethylamino)propyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H35N3O3S
(11S)-N-[3-(diethylamino)propyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21FN2O3S
(11R)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C30H32N2O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-chlorophenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-3-[(3R,5S)-3,5-dimethylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-benzyl-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O4S
(11S)-5-benzyl-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(azepane-1-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O3S
(11S)-3-(azepane-1-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— 10-allyl-N-(3-methylbutyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C22H24N2O2S
10-allyl-N-(3-methylbutyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— (11S)-N-[2-(diethylamino)ethyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28FN3O3S
(11S)-N-[2-(diethylamino)ethyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23FN2O4S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H26FN3O4S
(11R)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-3-(azepane-1-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O3S
(11R)-3-(azepane-1-carbonyl)-5-[(2-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(4-fluorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O3S
(11R)-5-[(4-fluorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H27FN2O3S
(11S)-3-[(3R,5R)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H26FN3O4S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-N,N-diethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11R)-5-[(4-chlorophenyl)methyl]-N,N-diethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C32H28N2O3S
(11S)-3-(3,4-dihydro-1H-isoquinoline-2-carbonyl)-5-[(2,5-dimethylphenyl)methyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-N-[2-(4-benzylpiperazin-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H32N4O3S
(11R)-N-[2-(4-benzylpiperazin-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 10-allyl-11-oxo-N-propyl-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C20H20N2O2S
10-allyl-11-oxo-N-propyl-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— (11R)-5-benzyl-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H20N2O4S
(11R)-5-benzyl-N-(furan-2-ylmethyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-chlorophenyl)methyl]-N-(3-ethoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H25ClN2O4S
(11R)-5-[(4-chlorophenyl)methyl]-N-(3-ethoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 10-allyl-N-benzyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide —— C24H20N2O2S
10-allyl-N-benzyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
—— (11R)-N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11R)-N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C28H26FN3O4S
(11S)-5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C28H27FN2O4S
3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(4-fluorophenyl)methyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— 5-[(2-fluorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one —— C27H25FN2O4S
5-[(2-fluorophenyl)methyl]-3-[(2R)-2-methylpiperidine-1-carbonyl]-11,11-dioxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-benzyl-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O4S
(11R)-5-benzyl-6,11-dioxo-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H28N2O3S
(11S)-5-benzyl-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-benzyl-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C28H26N2O5S
(11R)-5-benzyl-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H19ClN2O3S2
(11R)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[3-(diethylamino)propyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H35N3O3S
(11R)-N-[3-(diethylamino)propyl]-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C25H22N2O3S
(11S)-5-benzyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-ethyl-3-[4-(4-nitrophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C26H24N4O5S
(11S)-5-ethyl-3-[4-(4-nitrophenyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H19ClN2O3S2
(11S)-5-[(4-chlorophenyl)methyl]-6,11-dioxo-N-(thiophen-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-(2,2-dimethoxyethyl)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H28N2O5S
(11R)-N-(2,2-dimethoxyethyl)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H30N2O3S
(11S)-5-benzyl-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(4-chlorophenyl)methyl]-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C25H21ClN2O3S
(11S)-5-[(4-chlorophenyl)methyl]-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— (11S)-N-butyl-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O3S
(11S)-N-butyl-5-[(4-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-N-[(2-chlorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H20ClFN2O3S
(11R)-N-[(2-chlorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-butyl-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2O3S
(11S)-5-benzyl-N-butyl-N-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-N-[2-[bis(2-methylpropyl)amino]ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C31H37N3O3S
(11S)-5-benzyl-N-[2-[bis(2-methylpropyl)amino]ethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-chlorophenyl)methyl]-N-[(1S,2R)-2-methylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H27ClN2O4S
5-[(4-chlorophenyl)methyl]-N-[(1S,2R)-2-methylcyclohexyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H31N3O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H27FN2O3S
(11S)-5-[(2-fluorophenyl)methyl]-6,11-dioxo-N-[(2R)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23FN2O4S
(11R)-5-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-N-[2-(azepan-1-yl)ethyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H30FN3O3S
(11S)-N-[2-(azepan-1-yl)ethyl]-5-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2,5-dimethylphenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H33N3O3S
(11S)-5-[(2,5-dimethylphenyl)methyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-benzyl-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C25H22N2O4S
(11S)-5-benzyl-3-(morpholine-4-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one