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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (11R)-N-[2-(cyclohexen-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H26N2O3S
(11R)-N-[2-(cyclohexen-1-yl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-6,11-dioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C24H22N2O3S
(11S)-5-ethyl-6,11-dioxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-ethyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C20H20N2O3S
(11S)-5-ethyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— N-(2-methoxyphenyl)-2-[(2R)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C24H22N2O3S
N-(2-methoxyphenyl)-2-[(2R)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— (2S)-5-(2-oxo-2-piperidin-1-ylethyl)-2-phenyl-2,3-dihydro-1,5-benzothiazepin-4-one —— C22H24N2O2S
(2S)-5-(2-oxo-2-piperidin-1-ylethyl)-2-phenyl-2,3-dihydro-1,5-benzothiazepin-4-one
—— N-(3-fluorophenyl)-2-[(2S)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C23H19FN2O2S
N-(3-fluorophenyl)-2-[(2S)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-[(2R)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C22H24N2O3S
N-[[(2R)-oxolan-2-yl]methyl]-2-[(2R)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 2-[(2R)-2-methyl-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(3-methylphenyl)acetamide —— C19H20N2O2S
2-[(2R)-2-methyl-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(3-methylphenyl)acetamide
—— (2S)-2-(4-methoxyphenyl)-5-(2-morpholin-4-yl-2-oxoethyl)-2,3-dihydro-1,5-benzothiazepin-4-one —— C22H24N2O4S
(2S)-2-(4-methoxyphenyl)-5-(2-morpholin-4-yl-2-oxoethyl)-2,3-dihydro-1,5-benzothiazepin-4-one
—— 2-[(2S)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide —— C23H20N2O2S
2-[(2S)-4-oxo-2-phenyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide
—— N-(2-ethoxyphenyl)-2-[(2R)-2-methyl-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C20H22N2O3S
N-(2-ethoxyphenyl)-2-[(2R)-2-methyl-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 8-methyl-N-[(1R)-1-phenylethyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C26H26N2OS
8-methyl-N-[(1R)-1-phenylethyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2S)-butan-2-yl]-8-chloro-6-ethylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C20H21ClN2OS
N-[(2S)-butan-2-yl]-8-chloro-6-ethylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-methyl-N-[(1R,2S)-2-methylcyclohexyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H30N2OS
8-methyl-N-[(1R,2S)-2-methylcyclohexyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R)-1-phenylethyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2OS
N-[(1R)-1-phenylethyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 6-methyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C23H20N2OS
6-methyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-chloro-6-ethyl-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C21H21ClN2O2S
8-chloro-6-ethyl-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-chloro-6-ethyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21ClN2OS
8-chloro-6-ethyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2S)-butan-2-yl]-6-ethylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C20H22N2OS
N-[(2S)-butan-2-yl]-6-ethylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 6-ethyl-8-methyl-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2OS
6-ethyl-8-methyl-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2R)-butan-2-yl]-8-chloro-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C19H19ClN2OS
N-[(2R)-butan-2-yl]-8-chloro-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 6-ethyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C24H22N2OS
6-ethyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-pyridin-2-ylsulfanylethanone —— C17H18N2OS2
1-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-pyridin-2-ylsulfanylethanone
—— 1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-pyridin-2-ylsulfanylethanone —— C17H18N2OS2
1-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-pyridin-2-ylsulfanylethanone
—— N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H28N2O2S
N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-chloro-6-methyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C23H19ClN2OS
8-chloro-6-methyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 2-(2,2-dimethyl-4-oxo-3H-1,5-benzothiazepin-5-yl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C23H26N2O2S
2-(2,2-dimethyl-4-oxo-3H-1,5-benzothiazepin-5-yl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide —— C22H24N2O2S
N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide
—— (11R)-5-[(3-chlorophenyl)methyl]-3-(4-cyclohexylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C31H32ClN3O3S
(11R)-5-[(3-chlorophenyl)methyl]-3-(4-cyclohexylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— (11S)-5-[(3-chlorophenyl)methyl]-N-(2-methyl-3-nitrophenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H20ClN3O5S
(11S)-5-[(3-chlorophenyl)methyl]-N-(2-methyl-3-nitrophenyl)-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (11S)-5-[(2-methylphenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C30H26N2O3S
(11S)-5-[(2-methylphenyl)methyl]-N-[(4-methylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 2-[(2S)-2-methyl-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C12H14N2O2S
2-[(2S)-2-methyl-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— (2R)-2-methyl-1,1-dioxo-3,5-dihydro-2H-1λ6,5-benzothiazepin-4-one —— C10H11NO3S
(2R)-2-methyl-1,1-dioxo-3,5-dihydro-2H-1λ6,5-benzothiazepin-4-one
—— (5R)-7-chloro-5-phenyl-1,5-dihydro-4,1-benzothiazepin-2-one —— C15H12ClNOS
(5R)-7-chloro-5-phenyl-1,5-dihydro-4,1-benzothiazepin-2-one
—— (11S)-N-(4-bromo-2-fluorophenyl)-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H17BrClFN2O3S
(11S)-N-(4-bromo-2-fluorophenyl)-5-[(3-chlorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-6,11,11-trioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C31H27ClN2O4S
5-[(3-chlorophenyl)methyl]-6,11,11-trioxo-N-[(2S)-4-phenylbutan-2-yl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28ClN3O4S
5-[(3-chlorophenyl)methyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2R)-butan-2-yl]-5-[(3-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23FN2O2S
N-[(2R)-butan-2-yl]-5-[(3-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-fluorophenyl)methyl]benzo[b][1,4]benzothiazepin-6-one —— C28H27FN2O2S
3-[(3S,5S)-3,5-dimethylpiperidine-1-carbonyl]-5-[(3-fluorophenyl)methyl]benzo[b][1,4]benzothiazepin-6-one
—— N-[(2R)-butan-2-yl]-5-ethyl-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C20H22N2O2S
N-[(2R)-butan-2-yl]-5-ethyl-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-fluorophenyl)methyl]-6-oxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C29H23FN2O2S
5-[(2-fluorophenyl)methyl]-6-oxo-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chlorophenyl)methyl]-3-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O2S
5-[(2-chlorophenyl)methyl]-3-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one
—— N-[(1R,2R)-2-methylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H26N2O2S
N-[(1R,2R)-2-methylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chlorophenyl)methyl]-3-[(2R,6R)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one —— C28H27ClN2O2S
5-[(2-chlorophenyl)methyl]-3-[(2R,6R)-2,6-dimethylpiperidine-1-carbonyl]benzo[b][1,4]benzothiazepin-6-one
—— N-[(1S,2R)-2-methylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C24H26N2O2S
N-[(1S,2R)-2-methylcyclohexyl]-6-oxo-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-chlorophenyl)methyl]-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H23ClN2O3S
5-[(2-chlorophenyl)methyl]-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 6-oxo-N-[(1S)-1-phenylethyl]-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H22N2O2S
6-oxo-N-[(1S)-1-phenylethyl]-5-prop-2-enylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-5-[(2-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C28H28FN3O2S
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-5-[(2-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1S,2R)-2-methylcyclohexyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H30N2O2S
N-[(1S,2R)-2-methylcyclohexyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-benzyl-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O3S
5-benzyl-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide