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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2S)-oxolan-2-yl]methyl 5-[(3-nitrophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H22N2O6S
[(2S)-oxolan-2-yl]methyl 5-[(3-nitrophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— N-(3-chloro-4-methylphenyl)-2-[(3S)-3-methyl-4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C23H26ClN3O4S2
N-(3-chloro-4-methylphenyl)-2-[(3S)-3-methyl-4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— [(2R)-oxolan-2-yl]methyl 5-[(2-chloro-6-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C26H21ClFNO4S
[(2R)-oxolan-2-yl]methyl 5-[(2-chloro-6-fluorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— N-(2-ethoxyphenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H31N3O5S2
N-(2-ethoxyphenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(2-methoxy-5-methylphenyl)-2-[(3S)-3-methyl-4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C24H29N3O5S2
N-(2-methoxy-5-methylphenyl)-2-[(3S)-3-methyl-4-oxo-7-pyrrolidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-ethyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide —— C25H31N3O4S2
N-ethyl-2-[(2S)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-phenylacetamide
—— N-(2-methoxy-5-methylphenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C25H31N3O5S2
N-(2-methoxy-5-methylphenyl)-2-[(2R)-2-methyl-4-oxo-7-piperidin-1-ylsulfonyl-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 5-acetyl-N-[(2R)-butan-2-yl]-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C15H22N2O3S2
5-acetyl-N-[(2R)-butan-2-yl]-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C24H21N3O4S
N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— (2R)-5-acetyl-2-methyl-N-(2,4,6-trimethylphenyl)-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H26N2O3S2
(2R)-5-acetyl-2-methyl-N-(2,4,6-trimethylphenyl)-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 1-[7-[(2S)-2-methylpiperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C17H24N2O3S2
1-[7-[(2S)-2-methylpiperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— (2R)-5-acetyl-N-(furan-2-ylmethyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H20N2O4S2
(2R)-5-acetyl-N-(furan-2-ylmethyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 1-[(2R)-7-(2,3-dihydroindol-1-ylsulfonyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C20H22N2O3S2
1-[(2R)-7-(2,3-dihydroindol-1-ylsulfonyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 1-[7-[[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C21H24N2O3S3
1-[7-[[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 5-acetyl-N-[(2S)-butan-2-yl]-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C15H22N2O3S2
5-acetyl-N-[(2S)-butan-2-yl]-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-5-acetyl-N-(furan-2-ylmethyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H20N2O4S2
(2S)-5-acetyl-N-(furan-2-ylmethyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 1-[7-[(2R)-2-methylpiperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C17H24N2O3S2
1-[7-[(2R)-2-methylpiperidin-1-yl]sulfonyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— 1-[(2S)-7-(2,3-dihydroindol-1-ylsulfonyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C20H22N2O3S2
1-[(2S)-7-(2,3-dihydroindol-1-ylsulfonyl)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide —— C24H21N3O4S
N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(5-oxopyrido[2,3-b][1,5]benzothiazepin-6-yl)acetamide
—— 1-[7-[[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C21H24N2O3S3
1-[7-[[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]sulfonyl]-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— ethyl 3-[N-[[(3S)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate —— C21H24N2O5S2
ethyl 3-[N-[[(3S)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate
—— 7-[[(2S)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C18H18N2O3S3
7-[[(2S)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-N-[3-[benzyl(ethyl)amino]propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O3S2
(3S)-N-[3-[benzyl(ethyl)amino]propyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[3-(dimethylamino)-4-methylphenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H23N3O3S2
(3R)-N-[3-(dimethylamino)-4-methylphenyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— methyl 3-[N-[[(2S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate —— C20H22N2O5S2
methyl 3-[N-[[(2S)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate
—— (3R)-N-[(2-ethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O4S2
(3R)-N-[(2-ethoxyphenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[(3S)-3-phenylpyrrolidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H20N2O3S2
7-[(3S)-3-phenylpyrrolidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-N-cyclohexyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H26N2O3S3
(3R)-N-cyclohexyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-(3-pyrrolidin-1-ylpropyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H25N3O3S2
(3R)-3-methyl-4-oxo-N-(3-pyrrolidin-1-ylpropyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— ethyl 3-[N-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate —— C21H24N2O5S2
ethyl 3-[N-[[(3R)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl]sulfonyl]anilino]propanoate
—— (3S)-N-(4-cyanophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15N3O3S2
(3S)-N-(4-cyanophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[(3,4-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O5S2
(2S)-N-[(3,4-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-7-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C25H31N3O3S2
(3S)-7-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-N-(1,3-benzodioxol-5-yl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H16N2O5S2
(3R)-N-(1,3-benzodioxol-5-yl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-7-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C25H31N3O3S2
(3R)-7-[4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-3-methyl-N-(2-morpholin-4-ylethyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H23N3O4S2
(3R)-3-methyl-N-(2-morpholin-4-ylethyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[(3-bromophenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H17BrN2O3S2
(3R)-N-[(3-bromophenyl)methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[2-(furan-2-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H18N2O4S2
(3S)-N-[2-(furan-2-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-N-[3-(4-methylpiperidin-1-yl)propyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H29N3O3S2
(3S)-3-methyl-N-[3-(4-methylpiperidin-1-yl)propyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S3
(3S)-3-methyl-N-[2-(4-methylsulfanylphenyl)ethyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-cyclopentyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O3S3
(3R)-N-cyclopentyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-cyclopentyl-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O4S2
(3R)-N-cyclopentyl-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2R)-2-ethyl-6-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H22N2O4S2
7-[[(2R)-2-ethyl-6-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-3-methyl-4-oxo-N-(3-pyrrolidin-1-ylpropyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H25N3O3S2
(3S)-3-methyl-4-oxo-N-(3-pyrrolidin-1-ylpropyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O4S2
(3R)-3-methyl-4-oxo-N-[(4-propan-2-yloxyphenyl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-cyclohexyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H26N2O3S3
(3S)-N-cyclohexyl-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-butyl-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H24N2O4S2
(3R)-N-butyl-N-(furan-2-ylmethyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-(4-sulfamoylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H17N3O5S3
(3R)-3-methyl-4-oxo-N-(4-sulfamoylphenyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[3-(furan-2-yl)propyl]-N,3-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H22N2O4S2
(3S)-N-[3-(furan-2-yl)propyl]-N,3-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— ethyl (3S)-3-(4-methylphenyl)-3-[(4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl)sulfonylamino]propanoate —— C21H24N2O5S2
ethyl (3S)-3-(4-methylphenyl)-3-[(4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-7-yl)sulfonylamino]propanoate