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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-benzyl-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C26H24N2O3S
5-benzyl-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]propyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C32H37N3O2S
N-[3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]propyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2S)-2-methyl-3-(4-methylpiperidin-1-yl)propyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C32H37N3O2S
N-[(2S)-2-methyl-3-(4-methylpiperidin-1-yl)propyl]-5-[(4-methylphenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-benzyl-N-[(2S)-butan-2-yl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H24N2O2S
5-benzyl-N-[(2S)-butan-2-yl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-methylphenyl)methyl]-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H26N2O3S
5-[(4-methylphenyl)methyl]-6-oxo-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(1R,2R)-2-methylcyclohexyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide —— C21H22N2O2S
N-[(1R,2R)-2-methylcyclohexyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(2-methylphenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C30H26N2O2S
5-[(2-methylphenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O2S
N-[(2R)-butan-2-yl]-5-[(4-chlorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— N-[(2S)-butan-2-yl]-5-[(3-chlorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C25H23ClN2O2S
N-[(2S)-butan-2-yl]-5-[(3-chlorophenyl)methyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(3-chlorophenyl)methyl]-N-[(2S)-3-(diethylamino)-2-methylpropyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C29H32ClN3O2S
5-[(3-chlorophenyl)methyl]-N-[(2S)-3-(diethylamino)-2-methylpropyl]-6-oxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— (6E)-6-[2-(2-methoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H19NO2S
(6E)-6-[2-(2-methoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-6-[2-(4-methoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H19NO2S
(6Z)-6-[2-(4-methoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-3-methoxy-6-(2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene)cyclohexa-2,4-dien-1-one —— C22H19NO2S
(6Z)-3-methoxy-6-(2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene)cyclohexa-2,4-dien-1-one
—— (6E)-5-methoxy-6-(2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene)cyclohexa-2,4-dien-1-one —— C22H19NO2S
(6E)-5-methoxy-6-(2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene)cyclohexa-2,4-dien-1-one
—— 3-[(2S)-2-(5-bromo-2-hydroxyphenyl)-7-(trifluoromethyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione —— C22H15BrF3NO4S
3-[(2S)-2-(5-bromo-2-hydroxyphenyl)-7-(trifluoromethyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione
—— 2,2-dimethyl-4-[(E)-2-thiophen-2-ylethenyl]-3H-1,5-benzothiazepine —— C17H17NS2
2,2-dimethyl-4-[(E)-2-thiophen-2-ylethenyl]-3H-1,5-benzothiazepine
—— 5-Ethyl-2-(4-fluorophenyl)-4-thiophen-2-yl-2,3-dihydro-1,5-benzothiazepin-5-ium —— C21H19FNS2+
5-Ethyl-2-(4-fluorophenyl)-4-thiophen-2-yl-2,3-dihydro-1,5-benzothiazepin-5-ium
—— 3-(4-benzyl-2,3,4,5-tetrahydropyridin-1-ium-1-yl)-1-(7-methoxy-3,5-dihydro-2H-1,4-benzothiazepin-4-yl)propan-1-one —— C25H31N2O2S+
3-(4-benzyl-2,3,4,5-tetrahydropyridin-1-ium-1-yl)-1-(7-methoxy-3,5-dihydro-2H-1,4-benzothiazepin-4-yl)propan-1-one
—— (6Z)-6-[2-(3-methoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H19NO2S
(6Z)-6-[2-(3-methoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one
—— 1,5-anhydro-2,4-dideoxy-3-O-methyl-2-{[(4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-7-yl)sulfonyl]amino}-D-threo-pentitol —— C15H20N2O5S2
1,5-anhydro-2,4-dideoxy-3-O-methyl-2-{[(4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-7-yl)sulfonyl]amino}-D-threo-pentitol
—— 1,5-anhydro-2,4-dideoxy-2-{[(4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-7-yl)sulfonyl]amino}-D-threo-pentitol —— C14H18N2O5S2
1,5-anhydro-2,4-dideoxy-2-{[(4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-7-yl)sulfonyl]amino}-D-threo-pentitol
—— (3Z)-6-methyl-3-[2-(4-nitrophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]pyran-2,4-dione —— C21H16N2O5S
(3Z)-6-methyl-3-[2-(4-nitrophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]pyran-2,4-dione
—— Diltiazem, M(O-desmethyl-desamino-HO-), AC —— C23H23NO7S
Diltiazem, M(O-desmethyl-desamino-HO-), AC
—— N-Pyrrol2-[8-chloro-2-(4-methoxyphenyl)-4-oxo-3-trimethylsilanyloxy-3,4-dihydro-2H-benzo[b][1,4]thiazepin-5-yl]ethylmorpho-2,2,2-trifluoro-N-methylacetamide —— C24H28ClF3N2O4SSi
N-Pyrrol2-[8-chloro-2-(4-methoxyphenyl)-4-oxo-3-trimethylsilanyloxy-3,4-dihydro-2H-benzo[b][1,4]thiazepin-5-yl]ethylmorpho-2,2,2-trifluoro-N-methylacetamide
—— Acetic acid, 8-chloro-5-pyrrol2-[methyl-(2,2,2-trifluoroacetyl)amino]ethylmorpho-4-oxo-2-(4-trimethylsilanyloxyphenyl)-2,3,4,5-tetrahydrobenzo[b][1,4]thiazepin-3-yl ester —— C25H28ClF3N2O5SSi
Acetic acid, 8-chloro-5-pyrrol2-[methyl-(2,2,2-trifluoroacetyl)amino]ethylmorpho-4-oxo-2-(4-trimethylsilanyloxyphenyl)-2,3,4,5-tetrahydrobenzo[b][1,4]thiazepin-3-yl ester
—— (6Z)-6-[2-(2,3-dimethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one —— C23H21NO3S
(6Z)-6-[2-(2,3-dimethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one
—— 4-(5,6-dichlorobenzimidazol-2-ylidene)-2-(3-nitrophenyl)-3,5-dihydro-2H-1,5-benzothiazepine —— C22H14Cl2N4O2S
4-(5,6-dichlorobenzimidazol-2-ylidene)-2-(3-nitrophenyl)-3,5-dihydro-2H-1,5-benzothiazepine
—— 5-(2-Dimethylaminoethyl)-3-trimethylsilanyloxy-2-(4-trimethylsilanyloxyphenyl)-2,3-dihydro-5H-benzo[b] [1,4]thiazepin-4-one —— C25H38N2O3SSi2
5-(2-Dimethylaminoethyl)-3-trimethylsilanyloxy-2-(4-trimethylsilanyloxyphenyl)-2,3-dihydro-5H-benzo[b] [1,4]thiazepin-4-one
—— (6Z)-6-[2-(2-chlorophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one —— C21H16ClNOS
(6Z)-6-[2-(2-chlorophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one
—— 1-cyclohexyl-3-[3-(1,1-dioxo-3,5-dihydro-2H-1lambda6,4-benzothiazepin-4-yl)-3-oxopropyl]urea —— C19H27N3O4S
1-cyclohexyl-3-[3-(1,1-dioxo-3,5-dihydro-2H-1lambda6,4-benzothiazepin-4-yl)-3-oxopropyl]urea
—— [2-(2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl)-2-oxoethyl] 4-acetyl-1H-pyrrole-2-carboxylate —— C19H20N2O4S
[2-(2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl)-2-oxoethyl] 4-acetyl-1H-pyrrole-2-carboxylate
—— 1-[2-(4-Benzo[b][1,4]benzothiazepin-6-ylpiperazin-1-yl)ethoxy]butan-2-ol —— C23H29N3O2S
1-[2-(4-Benzo[b][1,4]benzothiazepin-6-ylpiperazin-1-yl)ethoxy]butan-2-ol
—— 1-(4-Benzo[b][1,4]benzothiazepin-6-ylpiperazin-1-yl)-2-(2-hydroxyethoxy)ethane-1,1,2,2-tetrol —— C21H25N3O6S
1-(4-Benzo[b][1,4]benzothiazepin-6-ylpiperazin-1-yl)-2-(2-hydroxyethoxy)ethane-1,1,2,2-tetrol
—— Ethane;3-(methylamino)-5-phenyl-2,3-dihydro-1,5-benzothiazepin-4-one —— C18H22N2OS
Ethane;3-(methylamino)-5-phenyl-2,3-dihydro-1,5-benzothiazepin-4-one
—— 2-Ethyl-5-phenyl-2,3,4,5-tetrahydro-1lambda6,4-benzothiazepine 1,1-dioxide —— C17H19NO2S
2-Ethyl-5-phenyl-2,3,4,5-tetrahydro-1lambda6,4-benzothiazepine 1,1-dioxide
—— 6-Chloro-5,6-dihydrobenzo[b][1,4]benzothiazepine-3-carbonyl chloride —— C14H9Cl2NOS
6-Chloro-5,6-dihydrobenzo[b][1,4]benzothiazepine-3-carbonyl chloride
—— 3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-8-[3-methoxy-5-[3-methyl-4-(6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carbonyl)piperazin-1-yl]phenyl]-5H-benzo[b][1,4]benzothiazepin-6-one —— C52H48N6O5S2
3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-8-[3-methoxy-5-[3-methyl-4-(6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carbonyl)piperazin-1-yl]phenyl]-5H-benzo[b][1,4]benzothiazepin-6-one
—— (3Z)-3-[2-(3-hydroxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione —— C21H17NO4S
(3Z)-3-[2-(3-hydroxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione
—— 4-(2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene)cyclohexa-2,5-dien-1-one —— C21H17NOS
4-(2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene)cyclohexa-2,5-dien-1-one
—— (3Z)-3-[2-(4-fluorophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione —— C21H16FNO3S
(3Z)-3-[2-(4-fluorophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione
—— (6Z)-6-[2-(4-methylphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one —— C22H19NOS
(6Z)-6-[2-(4-methylphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,4-dien-1-one
—— 2-[2-(4-Benzo[b][1,4]benzothiazepin-6-ylpiperazin-1-yl)-1,1,2,2-tetrahydroxyethoxy]ethane-1,1,1,2,2-pentol —— C21H25N3O10S
2-[2-(4-Benzo[b][1,4]benzothiazepin-6-ylpiperazin-1-yl)-1,1,2,2-tetrahydroxyethoxy]ethane-1,1,1,2,2-pentol
—— 3-[3-(4-piperidin-1-ylpiperidin-1-yl)oxiran-2-yl]-5H-benzo[b][1,4]benzothiazepin-6-one —— C25H29N3O2S
3-[3-(4-piperidin-1-ylpiperidin-1-yl)oxiran-2-yl]-5H-benzo[b][1,4]benzothiazepin-6-one
—— 6-Amino-4-benzo[b][1,4]benzothiazepin-6-yl-1-[1,1-dihydroxy-2-(2,2,2-trihydroxyethoxy)ethyl]-6-methylpiperazine-2,2,3,3,5,5-hexol —— C22H28N4O12S
6-Amino-4-benzo[b][1,4]benzothiazepin-6-yl-1-[1,1-dihydroxy-2-(2,2,2-trihydroxyethoxy)ethyl]-6-methylpiperazine-2,2,3,3,5,5-hexol
—— 14-[(2S)-butan-2-yl]-6-thia-10,14-diazatetracyclo[8.6.1.05,17.011,16]heptadeca-1(17),2,4-triene —— C18H26N2S
14-[(2S)-butan-2-yl]-6-thia-10,14-diazatetracyclo[8.6.1.05,17.011,16]heptadeca-1(17),2,4-triene
—— 4-[3,3-dibutyl-7-(dimethylamino)-4,5-dihydro-2H-1,4-benzothiazepin-5-yl]phenol —— C25H36N2OS
4-[3,3-dibutyl-7-(dimethylamino)-4,5-dihydro-2H-1,4-benzothiazepin-5-yl]phenol
—— 6-[4-(2-Deuteriooxyethyl)piperazin-1-yl]benzo[b][1,4]benzothiazepine —— C19H21N3OS
6-[4-(2-Deuteriooxyethyl)piperazin-1-yl]benzo[b][1,4]benzothiazepine
—— 3-(6-methoxy-5,6-dihydrobenzo[b][1,4]benzothiazepin-3-yl)-N-(1-phenylbutan-2-yl)oxiran-2-amine —— C26H28N2O2S
3-(6-methoxy-5,6-dihydrobenzo[b][1,4]benzothiazepin-3-yl)-N-(1-phenylbutan-2-yl)oxiran-2-amine
—— 5H-benzo[b][1,4]benzothiazepin-6-one;ethane —— C17H21NOS
5H-benzo[b][1,4]benzothiazepin-6-one;ethane
—— (3Z)-3-[2-(4-chlorophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione —— C21H16ClNO3S
(3Z)-3-[2-(4-chlorophenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione