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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-N-(furan-2-ylmethyl)-2-methyl-N-(3-morpholin-4-ylpropyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O5S2
(2R)-N-(furan-2-ylmethyl)-2-methyl-N-(3-morpholin-4-ylpropyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[3-(azepan-1-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H29N3O3S2
(2R)-N-[3-(azepan-1-yl)propyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-(3,4-difluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14F2N2O3S2
(2R)-N-(3,4-difluorophenyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-cyclopentyl-N-(furan-2-ylmethyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O4S2
(2S)-N-cyclopentyl-N-(furan-2-ylmethyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H23N3O4S2
(3S)-3-methyl-4-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-7-[[3-[(4-fluorophenyl)methyl]-1,3-diazinan-1-yl]sulfonyl]-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C21H24FN3O3S2
(3R)-7-[[3-[(4-fluorophenyl)methyl]-1,3-diazinan-1-yl]sulfonyl]-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-3-methyl-N-[4-(1,2-oxazol-5-yl)phenyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H17N3O4S2
(3S)-3-methyl-N-[4-(1,2-oxazol-5-yl)phenyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C15H16N2O3S3
(3R)-3-methyl-4-oxo-N-(thiophen-2-ylmethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(3-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H18N2O4S2
(3R)-N-(3-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 4-oxo-N-[(1R)-1-thiophen-2-ylbutyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H20N2O3S3
4-oxo-N-[(1R)-1-thiophen-2-ylbutyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(3-cyanophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H15N3O3S2
(3S)-N-(3-cyanophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[[(2S)-2-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C18H18N2O4S2
7-[[(2S)-2-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]sulfonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-3-methyl-7-[4-[methyl(3-morpholin-4-ylpropyl)amino]piperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C23H36N4O4S2
(3R)-3-methyl-7-[4-[methyl(3-morpholin-4-ylpropyl)amino]piperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2R)-N-(3,4-dimethylphenyl)-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O3S2
(2R)-N-(3,4-dimethylphenyl)-N,2-dimethyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-benzyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H18N2O3S2
(3S)-N-benzyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-3-methyl-4-oxo-N-(2-pyrrolidin-1-ylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H23N3O3S2
(3S)-3-methyl-4-oxo-N-(2-pyrrolidin-1-ylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H20N2O5S2
N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[2-[benzyl(ethyl)amino]ethyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O3S2
(2R)-N-[2-[benzyl(ethyl)amino]ethyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[(3,4-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O5S2
(2R)-N-[(3,4-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[[4-(dimethylamino)phenyl]methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H23N3O3S2
(3S)-N-[[4-(dimethylamino)phenyl]methyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-benzyl-3-methyl-4-oxo-N-propan-2-yl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O3S2
(3S)-N-benzyl-3-methyl-4-oxo-N-propan-2-yl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-(2-fluorophenyl)-2-methyl-4-oxo-N-propyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H21FN2O3S2
(2S)-N-(2-fluorophenyl)-2-methyl-4-oxo-N-propyl-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H20N2O5S2
N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-N-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N,2-dimethyl-4-oxo-N-[(1-phenylpyrazol-4-yl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H22N4O3S2
(2S)-N,2-dimethyl-4-oxo-N-[(1-phenylpyrazol-4-yl)methyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-7-[4-[2-(4-chlorophenoxy)ethyl]piperazin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C22H26ClN3O4S2
(3S)-7-[4-[2-(4-chlorophenoxy)ethyl]piperazin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-7-[4-[2-(4-chlorophenoxy)ethyl]piperazin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C22H26ClN3O4S2
(3R)-7-[4-[2-(4-chlorophenoxy)ethyl]piperazin-1-yl]sulfonyl-3-methyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3R)-3-methyl-4-oxo-N-(2-phenylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3R)-3-methyl-4-oxo-N-(2-phenylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-benzyl-3-methyl-4-oxo-N-(2-phenylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C25H26N2O3S2
(3S)-N-benzyl-3-methyl-4-oxo-N-(2-phenylethyl)-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(2-chloro-4-fluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H14ClFN2O3S2
(3R)-N-(2-chloro-4-fluorophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-N-[(2,5-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O5S2
(2S)-N-[(2,5-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-7-(4-methylpiperidin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C16H22N2O3S2
(3R)-3-methyl-7-(4-methylpiperidin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (2R)-N-[(2,5-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C19H22N2O5S2
(2R)-N-[(2,5-dimethoxyphenyl)methyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2S)-2-methyl-7-(4-piperidin-1-ylpiperidin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H29N3O3S2
(2S)-2-methyl-7-(4-piperidin-1-ylpiperidin-1-yl)sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— 7-[(3R)-3-phenylpyrrolidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C19H20N2O3S2
7-[(3R)-3-phenylpyrrolidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-3-methyl-N-[(3-methylphenyl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3S)-3-methyl-N-[(3-methylphenyl)methyl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(furan-2-ylmethyl)-3-methyl-N-(2-morpholin-4-ylethyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C21H27N3O5S2
(3S)-N-(furan-2-ylmethyl)-3-methyl-N-(2-morpholin-4-ylethyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— 7-[(3S)-3-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C24H29N3O3S2
7-[(3S)-3-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)piperidin-1-yl]sulfonyl-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (3S)-N,N-diethyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C14H20N2O3S2
(3S)-N,N-diethyl-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(furan-2-ylmethyl)-3-methyl-N-(3-morpholin-4-ylpropyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C22H29N3O5S2
(3R)-N-(furan-2-ylmethyl)-3-methyl-N-(3-morpholin-4-ylpropyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-3-methyl-4-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H21N3O5S3
(3R)-3-methyl-4-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(2,5-diethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C20H24N2O5S2
(3R)-N-(2,5-diethoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[(2-methoxyphenyl)methyl]-2-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C24H31N3O4S2
(2R)-N-[(2-methoxyphenyl)methyl]-2-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N,3-dimethyl-N-(4-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H20N2O3S2
(3R)-N,3-dimethyl-N-(4-methylphenyl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H18N2O5S2
(3R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-(3-bromophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H15BrN2O3S2
(3S)-N-(3-bromophenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-[2-(furan-2-yl)ethyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C16H18N2O4S2
(2R)-N-[2-(furan-2-yl)ethyl]-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-[2-(azepan-1-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C18H27N3O3S2
(3R)-N-[2-(azepan-1-yl)ethyl]-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3S)-N-[(2-methoxyphenyl)methyl]-3-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C24H31N3O4S2
(3S)-N-[(2-methoxyphenyl)methyl]-3-methyl-N-(1-methylpiperidin-4-yl)-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (2R)-N-ethyl-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C12H16N2O3S2
(2R)-N-ethyl-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide
—— (3R)-N-(2-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide —— C17H18N2O4S2
(3R)-N-(2-methoxyphenyl)-3-methyl-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-sulfonamide