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苯并硫氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl N-(9-amino-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-3-yl)carbamate —— C14H19N3O3S
tert-butyl N-(9-amino-4-oxo-3,5-dihydro-2H-1,5-benzothiazepin-3-yl)carbamate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(dimethylamino)-3-fluorobenzoate —— C21H23FN2O3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 4-(dimethylamino)-3-fluorobenzoate
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 6-methyl-2-oxo-1H-pyridine-3-carboxylate —— C19H20N2O4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 6-methyl-2-oxo-1H-pyridine-3-carboxylate
—— 4-[(2R)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,5-dien-1-one —— C21H17NOS
4-[(2R)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,5-dien-1-one
—— 4-[(2S)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,5-dien-1-one —— C21H17NOS
4-[(2S)-2-phenyl-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]cyclohexa-2,5-dien-1-one
—— 2-[(1R)-cyclopent-2-en-1-yl]-1-[(2R)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone —— C18H20F3NOS
2-[(1R)-cyclopent-2-en-1-yl]-1-[(2R)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]ethanone
—— [(2S)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-quinoxalin-2-ylmethanone —— C20H16F3N3OS
[(2S)-2-methyl-7-(trifluoromethyl)-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-quinoxalin-2-ylmethanone
—— 2-[(2R)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide —— C26H23F3N2O5S
2-[(2R)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide
—— N-(4-acetamidophenyl)-2-[(2R)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C28H29N3O6S
N-(4-acetamidophenyl)-2-[(2R)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— 2-[(2S)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide —— C26H23F3N2O5S
2-[(2S)-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide
—— N-(4-acetamidophenyl)-2-[(2S)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C28H29N3O6S
N-(4-acetamidophenyl)-2-[(2S)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(3-acetamidophenyl)-2-[(2R)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C28H29N3O6S
N-(3-acetamidophenyl)-2-[(2R)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— N-(3-acetamidophenyl)-2-[(2S)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide —— C28H29N3O6S
N-(3-acetamidophenyl)-2-[(2S)-4-oxo-2-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,5-benzothiazepin-5-yl]acetamide
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2S)-oxolan-2-yl]acetate —— C18H23NO4S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-[(2S)-oxolan-2-yl]acetate
—— [(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(2-methyl-1,3-thiazol-5-yl)methanone —— C15H16N2OS2
[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(2-methyl-1,3-thiazol-5-yl)methanone
—— [(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(2-methyl-1,3-thiazol-5-yl)methanone —— C15H16N2OS2
[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-(2-methyl-1,3-thiazol-5-yl)methanone
—— N-cyclopropyl-N-[(2R)-3-methylbutan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide —— C18H24N2O2S
N-cyclopropyl-N-[(2R)-3-methylbutan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide
—— N-cyclopropyl-N-[(2S)-3-methylbutan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide —— C18H24N2O2S
N-cyclopropyl-N-[(2S)-3-methylbutan-2-yl]-4-oxo-3,5-dihydro-2H-1,5-benzothiazepine-7-carboxamide
—— (3E)-3-[2-(4-ethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione —— C23H21NO4S
(3E)-3-[2-(4-ethoxyphenyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-ylidene]-6-methylpyran-2,4-dione
—— [2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(2H-indazol-3-yl)acetate —— C21H21N3O3S
[2-[(2S)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl] 2-(2H-indazol-3-yl)acetate
—— 3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(5-pyridin-3-yl-1,2-oxazol-3-yl)methanone —— C18H15N3O2S
3,4-dihydro-2H-1,5-benzothiazepin-5-yl-(5-pyridin-3-yl-1,2-oxazol-3-yl)methanone
—— N-(2-fluorophenyl)-2-(2-(furan-2-yl)-4-oxo-3,4-dihydrobenzo[b][1,4]thiazepin-5(2H)-yl)acetamide —— C21H17FN2O3S
N-(2-fluorophenyl)-2-(2-(furan-2-yl)-4-oxo-3,4-dihydrobenzo[b][1,4]thiazepin-5(2H)-yl)acetamide
—— 2-[2-(furan-2-yl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide —— C19H17N3O4S
2-[2-(furan-2-yl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-5-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
—— N-benzyl-2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)acetamide —— C20H22N2O4S
N-benzyl-2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)acetamide
—— 3-(Azepane-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C22H24N2O3S
3-(Azepane-1-carbonyl)-5-ethyl-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— Methyl 5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C24H21NO4S
Methyl 5-[(2,5-dimethylphenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— 5-ethyl-6,11,11-trioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C22H19N3O4S
5-ethyl-6,11,11-trioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-Ethyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one —— C20H20N2O3S
5-Ethyl-11-oxo-3-(pyrrolidine-1-carbonyl)benzo[b][1,4]benzothiazepin-6-one
—— N-[3-(4-ethylpiperazin-1-yl)propyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide —— C23H28N4O2S
N-[3-(4-ethylpiperazin-1-yl)propyl]-6-oxo-5H-benzo[b][1,4]benzothiazepine-3-carboxamide
—— 2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)-N-(2-methoxyethyl)acetamide —— C16H22N2O5S
2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)-N-(2-methoxyethyl)acetamide
—— N-butyl-10-ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide —— C20H22N2O4S
N-butyl-10-ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
—— N-cyclopentyl-2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)acetamide —— C18H24N2O4S
N-cyclopentyl-2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)acetamide
—— 5-Ethyl-3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C25H23N3O5S
5-Ethyl-3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— N-cyclopropyl-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C19H18N2O3S
N-cyclopropyl-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— ethyl 4-{[(4-oxo-3,4-dihydro-1,5-benzothiazepin-5(2H)-yl)acetyl]amino}piperidine-1-carboxylate —— C19H25N3O4S
ethyl 4-{[(4-oxo-3,4-dihydro-1,5-benzothiazepin-5(2H)-yl)acetyl]amino}piperidine-1-carboxylate
—— N-[2-(2,5-dimethoxyphenyl)ethyl]-2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)acetamide —— C23H28N2O6S
N-[2-(2,5-dimethoxyphenyl)ethyl]-2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)acetamide
—— 5-ethyl-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C22H19N3O3S
5-ethyl-6,11-dioxo-N-(pyridin-2-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— 2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)-N-[(4-fluorophenyl)methyl]acetamide —— C20H21FN2O4S
2-(2,2-dimethyl-1,1,4-trioxo-3H-1lambda6,5-benzothiazepin-5-yl)-N-[(4-fluorophenyl)methyl]acetamide
—— 5-ethyl-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C23H25N3O4S
5-ethyl-6,11-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— Methyl 5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxylate —— C22H16FNO4S
Methyl 5-[(2-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxylate
—— 5-[(2-Fluorophenyl)methyl]-6,11-dioxo-3-benzo[b][1,4]benzothiazepinecarboxylic acid —— C21H14FNO4S
5-[(2-Fluorophenyl)methyl]-6,11-dioxo-3-benzo[b][1,4]benzothiazepinecarboxylic acid
—— 2-(1,1,4-triketo-2,2-dimethyl-3H-1,5-benzothiazepin-5-yl)acetic acid —— C13H15NO5S
2-(1,1,4-triketo-2,2-dimethyl-3H-1,5-benzothiazepin-5-yl)acetic acid
—— 5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide —— C27H26FN3O3S
5-[(4-fluorophenyl)methyl]-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
—— (1-oxido-4-oxo-3,4-dihydro-1,5-benzothiazepin-5(2H)-yl)acetic acid —— C11H11NO4S
(1-oxido-4-oxo-3,4-dihydro-1,5-benzothiazepin-5(2H)-yl)acetic acid
—— N-butyl-5-ethyl-N-methyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide —— C21H24N2O4S
N-butyl-5-ethyl-N-methyl-6,11,11-trioxobenzo[b][1,4]benzothiazepine-3-carboxamide
—— 5-[(4-Chlorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one —— C26H24ClN3O3S
5-[(4-Chlorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-11-oxobenzo[b][1,4]benzothiazepin-6-one
—— 5-Cycloheptyl-6-oxobenzo[b][1,4]benzothiazepine-2,3-dicarbonitrile —— C22H19N3OS
5-Cycloheptyl-6-oxobenzo[b][1,4]benzothiazepine-2,3-dicarbonitrile
—— 5-Cyclopentyl-6-oxobenzo[b][1,4]benzothiazepine-2,3-dicarbonitrile —— C20H15N3OS
5-Cyclopentyl-6-oxobenzo[b][1,4]benzothiazepine-2,3-dicarbonitrile
—— N-(4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-7-yl)furan-2-carboxamide —— C14H12N2O3S
N-(4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-7-yl)furan-2-carboxamide
—— 10-(4-Methylphenyl)-11-oxo-10,11-dihydrodibenzo[B,F][1,4]thiazepine-7,8-dicarbonitrile —— C22H13N3OS
10-(4-Methylphenyl)-11-oxo-10,11-dihydrodibenzo[B,F][1,4]thiazepine-7,8-dicarbonitrile